Sfoglia per Autore
Structural Investigation of 3,5-Disubstituted Isoxazoles by1H-Nuclear Magnetic Resonance
2003 Sechi, Mario; Sannia, Luciano; Orecchioni, Maria; Carta, Fabrizio; Paglietti, Giuseppe; Neamati, Nouri
Design and synthesis of novel dihydroxyindole-2-carboxylic acids as HIV-1 integrase inhibitors
2004 Sechi, Mario*; Angotzi, Gianfranco; Dallocchio, Roberto; Dessi, Alessandro; Carta, Fabrizio; Sannia, Luciano; Mariani, Alberto; Fiori, Stefano; Sanchez, Tino; Movsessian, Leah; Plasencia, Carmen; Neamati, Nouri
Design and synthesis of novel indole β-diketo acid derivatives as HIV-1 integrase inhibitors
2004 Sechi, Mario*; Derudas, Massimiliano; Dallocchio, Roberto; Dessì, Alessandro; Bacchi, Alessia; Sannia, Luciano; Carta, Fabrizio; Palomba, Michele; Ragab, Omar; Chan, Carney; Shoemaker, Robert; Sei, Shizuko; Dayam, Raveendra; Neamati, Nouri
Design of novel bioisosteres of β-diketo acid inhibitors of HIV-1 integrase
2005 Sechi, Mario*; Sannia, Luciano; Carta, Fabrizio; Palomba, Michele; Dallocchio, Roberto; Dessì, Alessandro; Derudas, Massimiliano; Zawahir, Zahrah; Neamati, Nouri
From ligand to complexes. Part 2. Remarks on human immunodeficiency virus type 1 integrase inhibition by β-diketo acid metal complexes
2008 Bacchi, Alessia; Biemmi, Mariano; Carcelli, Mauro; Carta, Fabrizio; Compari, Carlotta; Fisicaro, Emilia; Rogolino, Dominga; Sechi, Mario*; Sippel, Martin; Sotriffer, Christoph A.; Sanchez, Tino W.; Neamati, Nouri
Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides.
2009 A. Maresca;F. Carta;D. Vullo;A. Scozzafava;C. T. Supuran
Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c.
2009 F. Carta;A. Maresca;A. S. Covarrubias;S. L. Mowbray;T. A. Jones;C. T. Supuran
Carbonic anhydrase inhibitors. Diazenylbenzenesulfonamides are potent and selective inhibitors of the tumor-associated isozymes IX and XII over the cytosolic isoforms I and II.
2009 F. Carta;A. Maresca;A. Scozzafava;D. Vullo;C. T. Supuran
Carbonic anhydrase inhibitors: inhibition of cytosolic carbonic anhydrase isozymes II and VII with simple aromatic sulfonamides and some azo dyes.
2009 F. Carta;B. Pothen;A. Maresca;M. Tiwari;V. Singh;C. T. Supuran
Design, synthesis, molecular modeling, and anti-HIV-1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes
2009 Sechi, M; Carta, F; Sannia, L; Dallocchio, R; Dessi, A; Al-Safi, RI; Neamati, N
The β-carbonic anhydrases from Mycobacterium tuberculosis as drug targets
2010 Nishimori I.; Minakuchi T.; Maresca A.; Carta F.; Scozzafava A.; Supuran C.T.
Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule.
2010 F. Carta;C. Temperini;A. Innocenti;A. Scozzafava;K. Kaila;C. T. Supuran
NOVEL SULFONAMIDE COMPOUNDS FOR INHIBITION OF METASTATIC TUMOR GROWTH
2010 SUPURAN CLAUDIU; DEDHAR SHOUKAT; MCDONALD PAUL; CARTA FABRIZIO
CARBONIC ANHYDRASE INHIBITORS WITH ANTIMETASTATIC ACTIVITY
2010 SUPURAN CLAUDIU, DEDHAR SHOUKAT, CARTA FABRIZIO, WINUM JEAN-YVES, MCDONALD PAUL C
Searching for intermediates in Prins cyclisations: The 2-oxa-5-adamantyl carbocation
2010 Alder, Roger W.*; Carta, Fabrizio; Reed, Christopher A.; Stoyanova, Irina; Willis, Christine L.
The β-carbonic anhydrases from Mycobacterium tuberculosis as drug targets.
2010 I. Nishimori;T. Minakuchi;A. Maresca;F. Carta;A. Scozzafava;C. T. Supuran
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.
2011 F. Carta;V. Garaj;A. Maresca;J. Wagner;B. S. Avvaru;A. H. Robbins;A. Scozzafava;R. McKenna;C. T. Supuran
CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE
2011 claudiu supuran, andrea scozzafava, fabrizio carta
Targeting Tumor Hypoxia: Suppression of Breast TumorGrowth and Metastasis by Novel Carbonic Anhydrase IX Inhibitors
2011 Y.Lou; P.C. McDonald; A.Oloumi; S.Chia; C.Ostlund; A. Ahmadi; A.Kyle; U.auf dem Keller; S.Leung; D.Huntsman; B.Clarke; B.W.Sutherland; D.Waterhouse; M.Bally; C.Roskelley; C.M. Overall; A.Minchinton; F.Pacchiano; F. Carta; A.Scozzafava; N.Touisni; J.-Y.Winum; C.T. Supuran; S.Dedhar
Dithiocarbamates strongly inhibit the β-class carbonic anhydrases from Mycobacterium tuberculosis.
2011 A. Maresca;F. Carta;D. Vullo;C. T. Supuran
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Structural Investigation of 3,5-Disubstituted Isoxazoles by1H-Nuclear Magnetic Resonance | 2003 | Sechi, Mario; Sannia, Luciano; Orecchioni, Maria; Carta, Fabrizio; Paglietti, Giuseppe; Neamati, Nouri | |
Design and synthesis of novel dihydroxyindole-2-carboxylic acids as HIV-1 integrase inhibitors | 2004 | Sechi, Mario*; Angotzi, Gianfranco; Dallocchio, Roberto; Dessi, Alessandro; Carta, Fabrizio; Sannia, Luciano; Mariani, Alberto; Fiori, Stefano; Sanchez, Tino; Movsessian, Leah; Plasencia, Carmen; Neamati, Nouri | |
Design and synthesis of novel indole β-diketo acid derivatives as HIV-1 integrase inhibitors | 2004 | Sechi, Mario*; Derudas, Massimiliano; Dallocchio, Roberto; Dessì, Alessandro; Bacchi, Alessia; Sannia, Luciano; Carta, Fabrizio; Palomba, Michele; Ragab, Omar; Chan, Carney; Shoemaker, Robert; Sei, Shizuko; Dayam, Raveendra; Neamati, Nouri | |
Design of novel bioisosteres of β-diketo acid inhibitors of HIV-1 integrase | 2005 | Sechi, Mario*; Sannia, Luciano; Carta, Fabrizio; Palomba, Michele; Dallocchio, Roberto; Dessì, Alessandro; Derudas, Massimiliano; Zawahir, Zahrah; Neamati, Nouri | |
From ligand to complexes. Part 2. Remarks on human immunodeficiency virus type 1 integrase inhibition by β-diketo acid metal complexes | 2008 | Bacchi, Alessia; Biemmi, Mariano; Carcelli, Mauro; Carta, Fabrizio; Compari, Carlotta; Fisicaro, Emilia; Rogolino, Dominga; Sechi, Mario*; Sippel, Martin; Sotriffer, Christoph A.; Sanchez, Tino W.; Neamati, Nouri | |
Carbonic anhydrase inhibitors. Inhibition of the Rv1284 and Rv3273 beta-carbonic anhydrases from Mycobacterium tuberculosis with diazenylbenzenesulfonamides. | 2009 | A. Maresca;F. Carta;D. Vullo;A. Scozzafava;C. T. Supuran | |
Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c. | 2009 | F. Carta;A. Maresca;A. S. Covarrubias;S. L. Mowbray;T. A. Jones;C. T. Supuran | |
Carbonic anhydrase inhibitors. Diazenylbenzenesulfonamides are potent and selective inhibitors of the tumor-associated isozymes IX and XII over the cytosolic isoforms I and II. | 2009 | F. Carta;A. Maresca;A. Scozzafava;D. Vullo;C. T. Supuran | |
Carbonic anhydrase inhibitors: inhibition of cytosolic carbonic anhydrase isozymes II and VII with simple aromatic sulfonamides and some azo dyes. | 2009 | F. Carta;B. Pothen;A. Maresca;M. Tiwari;V. Singh;C. T. Supuran | |
Design, synthesis, molecular modeling, and anti-HIV-1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes | 2009 | Sechi, M; Carta, F; Sannia, L; Dallocchio, R; Dessi, A; Al-Safi, RI; Neamati, N | |
The β-carbonic anhydrases from Mycobacterium tuberculosis as drug targets | 2010 | Nishimori I.; Minakuchi T.; Maresca A.; Carta F.; Scozzafava A.; Supuran C.T. | |
Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule. | 2010 | F. Carta;C. Temperini;A. Innocenti;A. Scozzafava;K. Kaila;C. T. Supuran | |
NOVEL SULFONAMIDE COMPOUNDS FOR INHIBITION OF METASTATIC TUMOR GROWTH | 2010 | SUPURAN CLAUDIU; DEDHAR SHOUKAT; MCDONALD PAUL; CARTA FABRIZIO | |
CARBONIC ANHYDRASE INHIBITORS WITH ANTIMETASTATIC ACTIVITY | 2010 | SUPURAN CLAUDIU, DEDHAR SHOUKAT, CARTA FABRIZIO, WINUM JEAN-YVES, MCDONALD PAUL C | |
Searching for intermediates in Prins cyclisations: The 2-oxa-5-adamantyl carbocation | 2010 | Alder, Roger W.*; Carta, Fabrizio; Reed, Christopher A.; Stoyanova, Irina; Willis, Christine L. | |
The β-carbonic anhydrases from Mycobacterium tuberculosis as drug targets. | 2010 | I. Nishimori;T. Minakuchi;A. Maresca;F. Carta;A. Scozzafava;C. T. Supuran | |
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies. | 2011 | F. Carta;V. Garaj;A. Maresca;J. Wagner;B. S. Avvaru;A. H. Robbins;A. Scozzafava;R. McKenna;C. T. Supuran | |
CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE | 2011 | claudiu supuran, andrea scozzafava, fabrizio carta | |
Targeting Tumor Hypoxia: Suppression of Breast TumorGrowth and Metastasis by Novel Carbonic Anhydrase IX Inhibitors | 2011 | Y.Lou; P.C. McDonald; A.Oloumi; S.Chia; C.Ostlund; A. Ahmadi; A.Kyle; U.auf dem Keller; S.Leung; D.Huntsman; B.Clarke; B.W.Sutherland; D.Waterhouse; M.Bally; C.Roskelley; C.M. Overall; A.Minchinton; F.Pacchiano; F. Carta; A.Scozzafava; N.Touisni; J.-Y.Winum; C.T. Supuran; S.Dedhar | |
Dithiocarbamates strongly inhibit the β-class carbonic anhydrases from Mycobacterium tuberculosis. | 2011 | A. Maresca;F. Carta;D. Vullo;C. T. Supuran |
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