Sfoglia per Autore
SYNTHESIS OF SOME 2-ARYL-1,2,4-TRIAZOLO[1,5-C][1,3]BENZOXAZIN-5-ONES AS TOOLS TO DEFINE THE ESSENTIAL PHARMACOPHORIC DESCRIPTORS OF A BENZODIAZEPINE RECEPTOR LIGAND.
1995 D. CATARZI; L. CECCHI; V. COLOTTA; G. FILACCHIONI; F. VARANO; C. MARTINI; L. GIUSTI; A. LUCACCHINI
Hydrogen bonding power and benzodiazepine receptor affinity relationships of 2-phenyl and 2-carbethoxy- tricyclic derivatives
1995 Daniela Catarzi; Lucia Cecchi; Vittoria Colotta; Guido Filacchioni; Flavia Varano
Structure-activity relationship studies of novel pyrazolo[1,5-c][1,3]benzoxazines: synthesis and benzodiazepine receptor affinity.
1996 F. VARANO; D. CATARZI; V. COLOTTA; L. CECCHI; G.FILACCHIONI; A. GALLI; C. COSTAGLI
Synthesis and binding activity of some pyrazolo[1,5-c]quinazolines as tools to verify an optional binding site of a benzodiazepine receptor ligand.
1996 V. COLOTTA; D. CATARZI; F. VARANO; L. CECCHI; G.FILACCHIONI; A. GALLI; C. COSTAGLI
Benzodiazepine binding activity of some tricyclic heteroarometic systems to define the hydrogen bonding strength of the proton donors of the receptor site.
1996 V. COLOTTA; D. CATARZI; F. VARANO; F. MELANI; G.FILACCHIONI; L. CECCHI; A. GALLI; C. COSTAGLI
Tricyclic heteroaromatic systems. 1,2,4-triazolo[4,3-a]quinoxalines and 1,2,4-triazino[4,3-a]quinoxalines: synthesis and central benzodiazepine receptor activity.
1997 V. COLOTTA; D. CATARZI; F. VARANO; L. CECCHI; G. FILACCHIONI; A. GALLI; C. COSTAGLI.
Tricyclic heteroaromatic systems. Pyrazolo[3,4-c]quinolin-4-ones and pyrazolo[3,4-c]quinoline-1,4-diones: synthesis and benzodiazepine receptor activity.
1997 D. CATARZI; V. COLOTTA; F. VARANO; L. CECCHI; G.FILACCHIONI; A. GALLI; C. COSTAGLI
Tricyclic Heteroaromatic systems. 3-Substituted 1,2,3,5,6,7-hexahydro-2,5,6-trioxopyrazino[1,2,3-de]quinoxalines as novel antagonists at the glycine-NMDA site.
1997 F. VARANO; D. CATARZI; V. COLOTTA; L. CECCHI; G. FILACCHIONI; A. GALLI; C. COSTAGLI.
Synthesis and biological evaluation of a series of quinazoline-2-carboxylic acids and quinazolin-2,4-diones as glycine-NMDA antagonists: a pharmacophore model based approach.
1997 V. COLOTTA; D. CATARZI; F. VARANO; L. CECCHI; G.FILACCHIONI; A. GALLI; C. COSTAGLI
Tricyclic heteroaromatic systems. Synthesis and benzodiazepine receptor affinity of 2-substituted-1-benzopyrano[3,4-d]oxazol-4-ones, -thiazol-4-ones, and –imidazol-4-ones.
1998 V. COLOTTA; D. CATARZI; F. VARANO; L. CECCHI; G. FILACCHIONI; C. MARTINI; L. GIUSTI; A. LUCACCHINI
Synthesis and A1 and A2A binding activity of some pyrano[2,3-c]pyrazol-4-ones.
1998 V. COLOTTA; D. CATARZI; F. VARANO; F. MELANI; G.FILACCHIONI; L. CECCHI; L. TRINCAVELLI; C. MARTINI; A. LUCACCHINI
Synthesis of 2-substituted-3,4-dihydro-3-oxo-6,8-dichloro-2H-1,4-benzothiazin-1,1-dioxides and 1-oxides as glycine-NMDA receptor antagonists.
1998 F. VARANO; D. CATARZI; V. COLOTTA; L. CECCHI; G.FILACCHIONI; A. GALLI; C. COSTAGLI
1,2,4-triazolo[4,3-a]quinoxalin-1-one as a framework to obtain potent and selective A1, A2A and A3 adenosine receptor antagonists
1999 Vittoria Colotta; Daniela Catarzi; Flavia Varano; Letizia Trincavelli
4-Oxo-1,2,4-triazolo[1,5-a]quinoxalin-2-carboxylic acid derivatives: antagonists of the Glycine/NMDA and AMPA receptors.
1999 Daniela Catarzi; Vittoria Colotta; Flavia Varano; Chiara Costagli
Synthesis, glycine/NMDA and AMPA binding activity of some new 2,5,6-trioxopyrazino[1,2,3-de]quinoxalines and of their restricted analogs 2,5-dioxo- and 4,5-dioxoimidazo[1,5,4-de]quinoxalines.
1999 F. VARANO; D. CATARZI; V. COLOTTA; L. CECCHI; G.FILACCHIONI; A. GALLI; C. COSTAGLI
4,5-Dihydro-1,2,4-triazolo[1,5-a]quinoxalin-4-ones. Excitatory amino acid antagonists with combined glycine/NMDA and AMPA receptor affinity
1999 D. CATARZI; V. COLOTTA; F. VARANO; L. CECCHI; G. FILACCHIONI; A. GALLI; C. COSTAGLI
4-Amino-6-benzylamino-1,2-dihydro-2-phenyl-1,2,4-triazolo[4,3-a] quinoxalin-1-one: a new A2A adenosine receptor antagonist with high selectivity versus A1 receptors.
1999 V. COLOTTA; D. CATARZI; F. VARANO; L. CECCHI; G. FILACCHIONI; C. MARTINI; L. TRINCAVELLI; A. LUCACCHINI
4,5-Dihydro-2-phenyl-1,2,4-triazolo[1,5-a]quinoxaline derivatives as highly potent and selective A3 adenosine receptor antagonists
2000 Daniela Catarzi; Vittoria Colotta; Flavia Varano; Letizia Trincavelli
Tricyclic heteroaromatic system. 5,6-dihydro-5-oxo-pyrazolo[1,5-c]quinazolines as excitatory amino acid antagonists
2000 Flavia Varano; Daniela Catarzi; Vittoria Colotta; Chiara Costagli
Benzosubstituted 2-phenyl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones. Synthesis and binding activity on adenosine receptors
2000 Vittoria Colotta; Daniela Catarzi; Flavia Varano; Letizia Trincavelli
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