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BAKER'S YEAST REDUCTION OF PROCHIRAL G-NITROKETONES: ENANTIOSELECTIVE SYNTHESIS OF (S)-4-NITROALCOHOLS 1995 A. GUARNA; E. OCCHIATO; D. SCARPI; L. SPINETTI; M. VALLECCHI
Baker's yeast reduction of prochiral g-nitro ketones. II. Straightforward enantioselective synthesis of 2,7-dimethyl-1,6-dioxaspiro[4.4]nonanes 1995 E. OCCHIATO; A. GUARNA; F. DE SARLO; D. SCARPI
ASYMMETRIC HYDROGENATION OF PROCHIRAL G-NITROKETONES BY RUTHENIUM COMPLEXES 1996 D. SCARPI; G. MENCHI; E. OCCHIATO; A. GUARNA
SYNTHESIS OF ENANTIOPURE 2,7-DIARYL-1,6-DIOXASPIRO[4.4]NONANES VIA ENANTIOSELECTIVE REDUCTION OF PROCHIRAL G-NITROKETONES BY DIISOPINOCAMPHEYLCHLOROBORANE (DIP-CLTM) 1996 E. OCCHIATO; D. SCARPI; G. MENCHI; A. GUARNA
Synthesis of benzo[c]quinolizin-3-ones: selective non steroidal inhibitors of steroid 5a-Reductase 1 1998 A. GUARNA; E. G. OCCHIATO; D. SCARPI; R. TSAI; G. DANZA; A. COMERCI; R. MANCINA; M. SERIO
STEREOSELECTIVITY IN THE TICL4-CATALYSED REEACTION OF DANISHEFSKY¿S DIENE WITH A N-(ACYLOXY)IMINIUM ION: SYNTHESIS OF 5A VERSUS 5B D1(2)-19-NOR-10-AZASTEROIDS. PART 4 1998 E. OCCHIATO; D. SCARPI; F. MACHETTI; A. GUARNA
A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5-REDUCTASE INHIBITORS. 3.1 SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-17B-ACETYLOXY-(5B)-10-AZAESTR-1-EN-3-ONE 1998 A. GUARNA; E. OCCHIATO; F. MACHETTI; D. SCARPI
Synthesis and reactivity of bicycles derived from tartaric acids and alfa-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid 1999 A. GUARNA; A. GUIDI; F. MACHETTI; G. MENCHI; E. OCCHIATO; D. SCARPI; S. SISI; A. TRABOCCHI
A SHORT AND EFFICIENT ROUTE TO ENANTIOPURE 3,5-DIARYLPYRROLIZIDINES 1999 D. SCARPI; E. OCCHIATO; A. GUARNA
Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1 2000 A. GUARNA; F. MACHETTI; E. OCCHIATO; D. SCARPI; A. COMERCI; G. DANZA; R. MANCINA; M. SERIO; K. HARDY
MODIFICATION OF THE AZA-ROBINSON ANNULATION FOR THE SYNTHESIS OF 4-METHYL-BENZO[C]QUINOLIZIN-3-ONES, POTENT INHIBITORS OF STEROID 5A-REDUCTASE 1 2000 A. GUARNA; F. MACHETTI; E. OCCHIATO; D. SCARPI; E. LOMBARDI
Stereoselective Meisenheimer Rearrangement using BTAa's as Chiral Auxiliaries 2000 A. GUARNA; E. OCCHIATO; D. SCARPI; M. PIZZETTI; S. SISI
3-Aza-6,8-dioxabicyclo (3,2,1) octanes and analogues and combinatorial libraries 2000 GUARNA A; E. OCCHIATO; SCARPI D; MENCHI G; MACHETTI F
Synthesis of 8-Chloro-benzo[c]quinolizin-3-ones as Potent andSelective Inhibitors of Human Steroid 5-alpha-Reductase 1 2000 A. Guarna; E. G. Occhiato; D. Scarpi; C. Zorn; G. Danza; A. Comerci; R. Mancina; M. Serio
Introduction of the New Dipeptide Isostere 7-Endo-BtA as Reverse Turn Inducer in a Bowman-Birk Proteinase Inhibitor: Synthesis and Conformational Analysis 2001 SCARPI D.; OCCHIATO E.G.; TRABOCCHI A.; LEATHERBARROW R.J.; BRAUER A.B.E.; NIEVO M.; A. GUARNA
Effect of C-Ring Modifications in Benzo[c]quinolizin-3-ones, New Selective Inhibitors of Human 5a-Reductase 1 2001 A. GUARNA; E.G. OCCHIATO; F. MACHETTI; A. TRABOCCHI; D. SCARPI; G. DANZA; R. MANCINA; A. COMERCI; M. SERIO
Synthesis of 17b-N-Substituted 19-Nor-10-Azasteroids as Inhibitors of Human 5a-Reductase I and II 2002 D. SCARPI; E. OCCHIATO; G. DANZA; M. SERIO; A. GUARNA
Synthesis of New Enantiopure Bicycles gamma/delta-Amino Acid (BTKa), Derived from Tartaric Acid and alfa-Aminoacetophenone 2002 A.GUARNA; I.BUCELLI; F.MACHETTI; G. MENCHI; E.G.OCCHIATO; D.SCARPI; A.TRABOCCHI
Inhibition of Human beta-Tryptase by Bowman-Birk Inhibitor Derived Peptides 2002 D.SCARPI; J.D.MCBRIDE; R. J.LEATHERBARROW
Synthesis of New Molecular Scaffolds: 3-Aza-7,9-Dioxa-Bicyclo[4.2.1]Nonane (8-exo BTKa) and 3-Aza-8,10-Dioxa-Bicyclo[5.2.1]Decane (9-exo BTKa) Carboxylic Acids 2004 D. SCARPI; D. STRANGES; L. CECCHI; A. GUARNA
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