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Synthesis and carbonic anhydrase inhibitory effects of new N-glycosylsulfonamides incorporating the phenol moiety 2016 Riafrecha, Leonardo E.; Bua, Silvia; Supuran, Claudiu T.; Colinas, Pedro A.
Advances in New Psychoactive Substances Identification: The U.R.I.To.N Consortium 2017 Bertol, Elisabetta; Vaiano, Fabio; Mari, Francesco; Di Milia, Maria Grazia; Bua, Silvia; Supuran, Claudiu Trandafir; Carta, Fabrizio
Inhibition of Malassezia globosa carbonic anhydrase with phenols 2017 Entezari Heravi, Yeganeh; Bua, Silvia; Nocentini, Alessio; Del Prete, Sonia; Saboury, Ali Akbar; Sereshti, Hassan; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T
Benzenesulfonamide bearing imidazothiadiazole and thiazolotriazole scaffolds as potent tumor associated human carbonic anhydrase IX and XII inhibitors 2017 Kumar, Rajiv; Bua, Silvia; Ram, Sita; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T; Sharma, Pawan K.
Investigating the antiplasmodial activity of primary sulfonamide compounds identified in open source malaria data 2017 Fisher, Gillian M.; Bua, Silvia; Del Prete, Sonia; Arnold, Megan S.J.; Capasso, Clemente; Supuran, Claudiu T.; Andrews, Katherine T.; Poulsen, Sally-Ann
Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives 2017 Bozdag, Murat; Bua, Silvia; Osman, Sameh M; AlOthman, Zeid; Supuran, Claudiu T
Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous Bases 2017 Nocentini, Alessio; Bua, Silvia; Lomelino, Carrie L.; Mckenna, Robert; Menicatti, Marta; Bartolucci, Gianluca; Tenci, Barbara; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Gratteri, Paola; Supuran, Claudiu T.
Novel indolin-2-one-based sulfonamides as carbonic anhydrase inhibitors: Synthesis, in vitro biological evaluation against carbonic anhydrases isoforms I, II, IV and VII and molecular docking studies 2017 Eldehna, Wagdy M; Al-Ansary, Ghada H.; Bua, Silvia; Nocentini, Alessio; Gratteri, Paola; Altoukhy, Ayman; Ghabbour, Hazem; Ahmed, Hanaa Y.; Supuran, Claudiu T.
Novel sulfamide-containing compounds as selective carbonic anhydrase i inhibitors 2017 Berrino, Emanuela; Bua, Silvia; Mori, Mattia; Botta, Maurizio; Murthy, Vallabhaneni S.; Vijayakumar, Vijayaparthasarathi; Tamboli, Yasinalli; Bartolucci, Gianluca; Mugelli, Alessandro; Cerbai, Elisabetta; Supuran, Claudiu T.; Carta, Fabrizio
Synthesis and biological evaluation of benzenesulphonamide-bearing 1,4,5-trisubstituted-1,2,3-triazoles possessing human carbonic anhydrase I, II, IV, and IX inhibitory activity 2017 Kumar, Rajiv; Sharma, Vikas; Bua, Silvia; Supuran, Claudiu T; Sharma, Pawan K
Synthesis and human/bacterial carbonic anhydrase inhibition with a series of sulfonamides incorporating phthalimido moieties 2017 Mohamed, Menshawy A; Abdel-Aziz, Alaa A-M; Sakr, Helmy M; El-Azab, Adel S; Bua, Silvia; Supuran, Claudiu T
Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis 2017 Bua, Silvia; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Ghelardini, Carla; Bartolucci, Gianluca; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio
Improving the carbonic anhydrase inhibition profile of the sulfamoylphenyl pharmacophore by attachment of carbohydrate moieties 2017 Riafrecha, Leonardo E.; Bua, Silvia; Supuran, Claudiu T.; Colinas, Pedro A.
P-glycoprotein and carbonic anhydrases hybrid inhibitors: a new strategy to reverse multidrug resistance (MDR) in cancer cells 2018 E. Teodori, M. Coronnello, S. Bua, L. Braconi, D. Manetti, M.N. Romanelli, C. Supuran, S. Dei
APPLICATION OF LINEAR EQUATIONS DECONVOLUTION ANALYSIS (LEDA) ALGORITHM IN ION TRAP MASS SPECTROMETRY: RESOLUTION OF ISOMERIC PAIRS OF CARBONIC ANHYDRASE AND CYCLOOXYGENASE HYBRIDS INHIBITORS 2018 Donato Squillaci; Marta Menicatti; Silvia Bua; Claudiu T. Supuran; Gian Luca Bartolucci
STABILITY STUDY IN PLASMA OF NOVEL ESTER-LINKED NSAID - CARBONIC ANHYDRASE INHIBITOR HYBRIDS 2018 Silvia Bua; Marta Menicatti; Paola Gratteri; Alessio Nocentini; Claudiu T. Supuran; Gian Luca Bartolucci
Comparison of the Anion Inhibition Profiles of the α-CA Isoforms (SpiCA1, SpiCA2 and SpiCA3) from the Scleractinian Coral Stylophora pistillata 2018 Del Prete, Sonia; Bua, Silvia; Zoccola, Didier; Alasmary, Fatmah A S; AlOthman, Zeid; Alqahtani, Linah S; Techer, Nathalie; Supuran, Claudiu T; Tambutté, Sylvie; Capasso, Clemente
Synthesis, structure and bioactivity of primary sulfamate-containing natural products 2018 Mujumdar, Prashant; Bua, Silvia; Supuran, Claudiu T.; Peat, Thomas S.; Poulsen, Sally-Ann*
Novel hydrazido benzenesulfonamides-isatin conjugates: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies 2018 Mahmoud F. Abo-Ashour; Wagdy M. Eldehna; Alessio Nocentini; Hany S. Ibrahim; Silvia Bua; Sahar M. Abou-Seri; Claudiu T. Supuran
Natural Polyphenols Selectively Inhibit β-Carbonic Anhydrase from the Dandruff-Producing Fungus Malassezia globosa: Activity and Modeling Studies 2018 Nocentini, Alessio; Bua, Silvia; Del Prete, Sonia; Heravi, Yeganeh Entezari; Saboury, Ali A; Karioti, Anastasia; Bilia, Anna Rita; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T
Mostrati risultati da 1 a 20 di 104
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