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Amino acids as building blocks for carbonic anhydrase inhibitors 2018 Chiaramonte, Niccolò*; Romanelli, Maria Novella; Teodori, Elisabetta; Supuran, Claudiu T.
Designing selective modulators for the nicotinic receptor subtypes: challenges and opportunities 2018 Dina Manetti, Cristina Bellucci, Niccolo` Chiaramonte, Silvia Dei, Elisabetta Teodori, Maria Novella Romanelli
Design and synthesis of aminoester heterodimers containing flavone or chromone moieties as modulators of P-glycoprotein-based multidrug resistance (MDR) 2018 Silvia, Dei; Maria Novella Romanelli, ; Dina, Manetti; Niccolò, Chiaramonte; Marcella, Coronnello; Milena, Salerno; Elisabetta, Teodori
2-Benzylpiperazine: a new scaffold for potent human Carbonic Anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents. 2018 Niccolò Chiaramonte, Silvia Bua, Marta Ferraroni, Alessio Nocentini, Alessandro Bonardi, Gian Luca Bartolucci, Maria Concetta Durante, Laura Lucarini, Donata Chiapponi, Silvia Dei, Dina Manetti, Elisabetta Teodori, Paola Gratteri, Emanuela Masini, Claudiu T. Supuran, Maria Novella Romanelli
Investigation of piperazines as human carbonic anhydrase I, II, IV and VII activators 2018 Angeli, Andrea; Chiaramonte, Niccolò; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T
New Rigid Nicotine Analogues, Carrying a Norbornane Moiety, Are Potent Agonists of α7 and α3∗ Nicotinic Receptors 2019 Dina Manetti*† , Alexandra Garifulina‡, Gian Luca Bartolucci , Carla Bazzicalupi§ , Cristina Bellucci†, Niccolò Chiaramonte†, Silvia Dei†, Lorenzo Di Cesare Mannelli∥, Carla Ghelardini∥, Paola Gratteri⊥ , Ekaterina Spirova‡, Irina Shelukhina‡, Elisabetta Teodori†, Katia Varani#, Victor Tsetlin‡, Maria Novella Romanelli†
Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug-resistance (MDR) modulators 2019 Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Marcella Coronnello, Niccolò Chiaramonte, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Chatchanok Udomtanakunchai, Nicola Antonio Colabufo, Gian luca Bartolucci, Ottavia Spiga, Milena Salerno, Elisabetta Teodori
Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine 2020 Niccolò Chiaramonte, Soumia Maach, Caterina Biliotti, Andrea Angeli, Gian luca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T. Supuran, Maria Novella Romanelli
Design, synthesis and preliminary biological evaluation of modulators of metalloenzymes 2020 Niccolò Chiaramonte
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers 2020 Braconi L.; Bartolucci G.; Contino M.; Chiaramonte N.; Giampietro R.; Manetti D.; Perrone M.G.; Romanelli M.N.; Colabufo N.A.; Riganti C.; Dei S.; Teodori E.
Carbonic Anhydrase IV Selective Inhibitors Counteract the Development of Colitis-Associated Visceral Pain in Rats 2021 Lucarini E., Nocentini A., Bonardi A., Chiaramonte N., Parisio C., Micheli L., Toti A., Ferrara V., Carrino D., Pacini A., Romanelli M.N., Supuran C.T., Ghelardini C., Di Cesare Mannelli L.
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators 2022 Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N.
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity 2022 Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N.
Dual HDAC–BRD4 inhibitors endowed with antitumor and antihyperalgesic activity 2022 Maach S.; Chiaramonte N.; Borgonetti V.; Sarno F.; Pierucci F.; Dei S.; Teodori E.; Altucci L.; Meacci E.; Galeotti N.; Romanelli M.N.
Mostrati risultati da 1 a 14 di 14
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