Sfoglia per Autore
Unexpected agonistic activity in a series of muscarinic antagonists
1999 P. Angeli; C. Bellucci; S. Dei; F. Gualtieri; D. Manetti; G. Marucci; R. Matucci; M.N.Romanelli; S. Scapecchi; E. Teodori
Hybridized and isosteric analogs of N1-acetyl-N4-dimethyl-piperazinium iodide (ADMP) and N1-phenyl-N4-dimethyl-piperazinium iodide (DMPP) with central nicotinic action
1999 D. MANETTI; A. BARTOLINI; P. BOREA; C. BELLUCCI; S. DEI; C. GHELARDINI; F. GUALTIERI; M. ROMANELLI; S. SCAPECCHI; E. TEODORI; K. VARANI
Antisense knockdowns of M1 receptors induces transient anterograde amnesia in mice
1999 GHELARDINI C.; GALEOTTI N.; MATUCCI R.; BELLUCCI C.; GUALTIERI F.; CAPACCIOLI S.; QUATTRONE A.; BARTOLINI A.
1,4-Diazabicyclo[4.3.0]nonan-9-ones and 1,4-diamidopiperazines as new classes of highly potent nootropic drugs
2000 D. Manetti; C. Ghelardini; A. Bartolini; C. Bellucci; S. Dei; N. Galeotti; F. Gualtieri; M.N. Romanelli; S Scapecchi; E. Teodori
1,4-Diazabicyclo[4.3.0]nonan-9-ones as a new class of highly potent nootropic drugs
2000 Dina Manetti; Carla Ghelardini; Alessandro Bartolini; Cristina Bellucci; Silvia Dei; Nicoletta Galeotti; Fulvio Gualtieri; Maria Novella Romanelli; Serena Scapecchi; Elisabetta Teodori
Design, synthesis and preliminary pharmacological evaluation of 1,4-diazabicyclo[4.3.0]nonan-9-ones as a new class of highly potent nootropic drugs.
2000 D. MANETTI; C. GHELARDINI; A. BARTOLINI; C. BELLUCCI; S. DEI; N. GALEOTTI; F. GUALTIERI; M.N. ROMANELLI; S. SCAPECCHI; E. TEODORI
Piperazine derivatives possessing nootropic activity
2001 A Bartolini; C Bellucci; N Galeotti; C Ghelardini; F Gualtieri; D Manetti
Structure-activity relationships in 2,2-diphenyl-2-ethylthioacetic acid esters: unexpected agonistic activity in a series of muscarinic antagonists.
2001 Scapecchi, Serena; Marucci, G.; Matucci, Rosanna; Angeli, P.; Bellucci, Cristina; Buccioni, M.; Dei, Silvia; Gualtieri, Fulvio; Manetti, Dina; Romanelli, MARIA NOVELLA; Teodori, Elisabetta
(1,3-Dioxolane)- and (1,3-oxathiolane)-2-pyrrolidines: molecular hybrids with potential anti-Alzheimer activity
2001 Silvia Dei; Elisabetta Teodori; Cristina Bellucci; Fulvio Gualtieri; Luca Guandalini; Rosanna Matucci; Serena Scapecchi; Katia Varani; Marta Ferraroni
Sintesi e affinità per i recettori colinergici degli stereoisomeri della 1-metil-2-(2-metil-1,3-diossolan-4-il)pirrolidina, della 1-metil-2-(2-metil-1,3-ossatiolan-5-il)pirrolidina e dei loro iodometilati
2002 Silvia Dei; Cristina Bellucci; Michela Buccioni; Marta Ferraroni; Fulvio Gualtieri; Luca Guandalini; Dina Manetti; Rosanna Matucci; Maria Novella Romanelli; Serena Scapecchi; Katia Varani; Elisabetta Teodori
Highly chiral muscarinic ligands: synthesis and affinity of diastereomeric and enantiomeric isomers of 1-methyl-2-(2-methyl-1,3-oxathiolane-5-yl)pyrrolidine 3-sulfoxides and their methyl iodides
2003 Serena Scapecchi; Cecilia Martelli; Elisabetta Martini; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Luca Guandalini; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori
Molecular modulation of muscarinic antagonists. Synthesis and pharmacological profile of 2,2-diphenyl-2-ethylthioacetic acid and 3,3-diphenyl-3-ethylthiopropionic acid derivatives characterized by a dipeptide spacer
2003 Serena Scapecchi; Piero Angeli; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Cecilia Martelli; Gabriella Marucci; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori
Design, synthesis and preliminary pharmacological evaluation of alkylderivatives of 4-aminopiperidine as N-type calcium channels blockers
2003 Elisabetta Teodori; Elisabetta Baldi; Cristina Bellucci; Silvia Dei; Carla Ghelardini; Fulvio Gualtieri; Rosanna Matucci; Maria Novella Romanelli; Serena Scapecchi
Synthesis and Cholinergic Affinity of Diastereomeric and Enantiomeric Isomers of 1-Methyl-2-(2-methyl-1,3-dioxolan-4-yl)-pyrrolidine, 1-Methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine and of Their Iodomethylates
2003 Dei, Silvia; Bellucci, Cristina; Buccioni, M.; Ferraroni, Marta; Gualtieri, Fulvio; Guandalini, Luca; Manetti, Dina; Matucci, Rosanna; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Teodori, Elisabetta
MOLECULAR MODULATION OF MUSCARINIC ANTAGONISTS. SYNTHESIS AND PHARMACOLOGICAL PROFILE OF 2,2-DIPHENYL-2-ETHYLTHIOACETIC AND 3,3-DIPHENYL-3-ETHYLTHIOPROPIONIC ACID DERIVATIVES CHARACTERIZED BY A DIPEPTIDE SPACER
2004 S. SCAPECCHI; C. MARTELLI; P. ANGELI; C. BELLUCCI; M. BUCCIONI; S. DEI; F. GUALTIERI; G. MARUCCI; R. MATUCCI; M. ROMANELLI; E. TEODORI
Modulazione molecolare di antagonisti muscarinici. Sintesi e valutazione farmacologica preliminare di esteri amminoalchil piperazinici e piperidinici dell'acido 2,2-difenil-2-etiltioacetico
2004 S. Scapecchi; E. Martini; C. Bellucci; S. Dei; L. Guandalini; D. Manetti; C. Martelli; G. Marucci; R. Matucci
Synthesis and pharmacological characterization of diastereomeric and enantiomeric isomers of 1-methyl-2-(2-methyl-1,3-oxathiolane-5-yl)pyrrolidine 3-sulfoxides and their methyl iodides
2004 Serena Scapecchi; Cecilia Martelli; Elisabetta Martini; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori
MOLECULAR MODULATION OF MUSCARINIC ANTAGONISTS. SYNTHESIS AND AFFINITY PROFILE OF 2,2-DIPHENYL-2-ETHYLTHIO-ACETIC ACID ESTERS DESIGNED TO PROBE THE BINDING SITE CAVITY
2004 S. SCAPECCHI; E. MARTINI; C. BELLUCCI; M. BUCCIONI; S. DEI; L. GUANDALINI; D. MANETTI; C. MARTELLI; G. MARUCCI; R. MATUCCI
Design, synthesis and preliminary pharmacological evaluation of 4-aminopiperidine derivatives as N-type calcium channel blockers active on pain and neuropathic pain
2004 Teodori, Elisabetta; Baldi, Elisabetta; Dei, Silvia; Gualtieri, Fulvio; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Bellucci, Cristina; Ghelardini, Carla; Matucci, Rosanna
Muscarinic subtype affinity and functional activity profile of 1-methyl-2-(2-methyl-1,3-dioxolan-4-yl)pyrrolidine and 1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine derivatives.
2005 Dei, Silvia; Angeli, P.; Bellucci, Cristina; Buccioni, M.; Gualtieri, Fulvio; Marucci, G.; Manetti, Dina; Matucci, Rosanna; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Teodori, Elisabetta
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Unexpected agonistic activity in a series of muscarinic antagonists | 1999 | P. Angeli; C. Bellucci; S. Dei; F. Gualtieri; D. Manetti; G. Marucci; R. Matucci; M.N.Romanelli; S. Scapecchi; E. Teodori | |
Hybridized and isosteric analogs of N1-acetyl-N4-dimethyl-piperazinium iodide (ADMP) and N1-phenyl-N4-dimethyl-piperazinium iodide (DMPP) with central nicotinic action | 1999 | D. MANETTI; A. BARTOLINI; P. BOREA; C. BELLUCCI; S. DEI; C. GHELARDINI; F. GUALTIERI; M. ROMANELLI; S. SCAPECCHI; E. TEODORI; K. VARANI | |
Antisense knockdowns of M1 receptors induces transient anterograde amnesia in mice | 1999 | GHELARDINI C.; GALEOTTI N.; MATUCCI R.; BELLUCCI C.; GUALTIERI F.; CAPACCIOLI S.; QUATTRONE A.; BARTOLINI A. | |
1,4-Diazabicyclo[4.3.0]nonan-9-ones and 1,4-diamidopiperazines as new classes of highly potent nootropic drugs | 2000 | D. Manetti; C. Ghelardini; A. Bartolini; C. Bellucci; S. Dei; N. Galeotti; F. Gualtieri; M.N. Romanelli; S Scapecchi; E. Teodori | |
1,4-Diazabicyclo[4.3.0]nonan-9-ones as a new class of highly potent nootropic drugs | 2000 | Dina Manetti; Carla Ghelardini; Alessandro Bartolini; Cristina Bellucci; Silvia Dei; Nicoletta Galeotti; Fulvio Gualtieri; Maria Novella Romanelli; Serena Scapecchi; Elisabetta Teodori | |
Design, synthesis and preliminary pharmacological evaluation of 1,4-diazabicyclo[4.3.0]nonan-9-ones as a new class of highly potent nootropic drugs. | 2000 | D. MANETTI; C. GHELARDINI; A. BARTOLINI; C. BELLUCCI; S. DEI; N. GALEOTTI; F. GUALTIERI; M.N. ROMANELLI; S. SCAPECCHI; E. TEODORI | |
Piperazine derivatives possessing nootropic activity | 2001 | A Bartolini; C Bellucci; N Galeotti; C Ghelardini; F Gualtieri; D Manetti | |
Structure-activity relationships in 2,2-diphenyl-2-ethylthioacetic acid esters: unexpected agonistic activity in a series of muscarinic antagonists. | 2001 | Scapecchi, Serena; Marucci, G.; Matucci, Rosanna; Angeli, P.; Bellucci, Cristina; Buccioni, M.; Dei, Silvia; Gualtieri, Fulvio; Manetti, Dina; Romanelli, MARIA NOVELLA; Teodori, Elisabetta | |
(1,3-Dioxolane)- and (1,3-oxathiolane)-2-pyrrolidines: molecular hybrids with potential anti-Alzheimer activity | 2001 | Silvia Dei; Elisabetta Teodori; Cristina Bellucci; Fulvio Gualtieri; Luca Guandalini; Rosanna Matucci; Serena Scapecchi; Katia Varani; Marta Ferraroni | |
Sintesi e affinità per i recettori colinergici degli stereoisomeri della 1-metil-2-(2-metil-1,3-diossolan-4-il)pirrolidina, della 1-metil-2-(2-metil-1,3-ossatiolan-5-il)pirrolidina e dei loro iodometilati | 2002 | Silvia Dei; Cristina Bellucci; Michela Buccioni; Marta Ferraroni; Fulvio Gualtieri; Luca Guandalini; Dina Manetti; Rosanna Matucci; Maria Novella Romanelli; Serena Scapecchi; Katia Varani; Elisabetta Teodori | |
Highly chiral muscarinic ligands: synthesis and affinity of diastereomeric and enantiomeric isomers of 1-methyl-2-(2-methyl-1,3-oxathiolane-5-yl)pyrrolidine 3-sulfoxides and their methyl iodides | 2003 | Serena Scapecchi; Cecilia Martelli; Elisabetta Martini; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Luca Guandalini; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori | |
Molecular modulation of muscarinic antagonists. Synthesis and pharmacological profile of 2,2-diphenyl-2-ethylthioacetic acid and 3,3-diphenyl-3-ethylthiopropionic acid derivatives characterized by a dipeptide spacer | 2003 | Serena Scapecchi; Piero Angeli; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Cecilia Martelli; Gabriella Marucci; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori | |
Design, synthesis and preliminary pharmacological evaluation of alkylderivatives of 4-aminopiperidine as N-type calcium channels blockers | 2003 | Elisabetta Teodori; Elisabetta Baldi; Cristina Bellucci; Silvia Dei; Carla Ghelardini; Fulvio Gualtieri; Rosanna Matucci; Maria Novella Romanelli; Serena Scapecchi | |
Synthesis and Cholinergic Affinity of Diastereomeric and Enantiomeric Isomers of 1-Methyl-2-(2-methyl-1,3-dioxolan-4-yl)-pyrrolidine, 1-Methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine and of Their Iodomethylates | 2003 | Dei, Silvia; Bellucci, Cristina; Buccioni, M.; Ferraroni, Marta; Gualtieri, Fulvio; Guandalini, Luca; Manetti, Dina; Matucci, Rosanna; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Teodori, Elisabetta | |
MOLECULAR MODULATION OF MUSCARINIC ANTAGONISTS. SYNTHESIS AND PHARMACOLOGICAL PROFILE OF 2,2-DIPHENYL-2-ETHYLTHIOACETIC AND 3,3-DIPHENYL-3-ETHYLTHIOPROPIONIC ACID DERIVATIVES CHARACTERIZED BY A DIPEPTIDE SPACER | 2004 | S. SCAPECCHI; C. MARTELLI; P. ANGELI; C. BELLUCCI; M. BUCCIONI; S. DEI; F. GUALTIERI; G. MARUCCI; R. MATUCCI; M. ROMANELLI; E. TEODORI | |
Modulazione molecolare di antagonisti muscarinici. Sintesi e valutazione farmacologica preliminare di esteri amminoalchil piperazinici e piperidinici dell'acido 2,2-difenil-2-etiltioacetico | 2004 | S. Scapecchi; E. Martini; C. Bellucci; S. Dei; L. Guandalini; D. Manetti; C. Martelli; G. Marucci; R. Matucci | |
Synthesis and pharmacological characterization of diastereomeric and enantiomeric isomers of 1-methyl-2-(2-methyl-1,3-oxathiolane-5-yl)pyrrolidine 3-sulfoxides and their methyl iodides | 2004 | Serena Scapecchi; Cecilia Martelli; Elisabetta Martini; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori | |
MOLECULAR MODULATION OF MUSCARINIC ANTAGONISTS. SYNTHESIS AND AFFINITY PROFILE OF 2,2-DIPHENYL-2-ETHYLTHIO-ACETIC ACID ESTERS DESIGNED TO PROBE THE BINDING SITE CAVITY | 2004 | S. SCAPECCHI; E. MARTINI; C. BELLUCCI; M. BUCCIONI; S. DEI; L. GUANDALINI; D. MANETTI; C. MARTELLI; G. MARUCCI; R. MATUCCI | |
Design, synthesis and preliminary pharmacological evaluation of 4-aminopiperidine derivatives as N-type calcium channel blockers active on pain and neuropathic pain | 2004 | Teodori, Elisabetta; Baldi, Elisabetta; Dei, Silvia; Gualtieri, Fulvio; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Bellucci, Cristina; Ghelardini, Carla; Matucci, Rosanna | |
Muscarinic subtype affinity and functional activity profile of 1-methyl-2-(2-methyl-1,3-dioxolan-4-yl)pyrrolidine and 1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine derivatives. | 2005 | Dei, Silvia; Angeli, P.; Bellucci, Cristina; Buccioni, M.; Gualtieri, Fulvio; Marucci, G.; Manetti, Dina; Matucci, Rosanna; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Teodori, Elisabetta |
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