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Mostrati risultati da 241.903 a 241.922 di 270.005
Titolo Data di pubblicazione Autore(i) File
Synthesis, biological evaluation and in silico studies with 4-benzylidene-2-phenyl-5(4H)-imidazolone-based benzenesulfonamides as novel selective carbonic anhydrase IX inhibitors endowed with anticancer activity 2019 Eldehna W.M.; Abdelrahman M.A.; Nocentini A.; Bua S.; Al-Rashood S.T.; Hassan G.S.; Bonardi A.; Almehizia A.A.; Alkahtani H.M.; Alharbi A.; Gratteri P.; Supuran C.T.
Synthesis, biological evaluation and molecular modeling of novel selective COX-2 inhibitors: sulfide, sulfoxide, and sulfone derivatives of 1,5-diarylpyrrol-3-substituted scaffold 2019 Reale A, Brogi S, Chelini A, Paolino M1, Di Capua A, Giuliani G, Cappelli A, Giorgi G, Chemi G, Grillo A, Valoti M, Sautebin L, Rossi A, Pace S, La Motta C, Di Cesare Mannelli L, Lucarini E, Ghelardini C, Anzini M
Synthesis, biological evaluation and theoretical studies of (E)-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitors 2023 Ramzan, Farhat; Nabi, Syed Ayaz; Lone, Mehak Saba; Bonardi, Alessandro; Hamid, Aabid; Bano, Sameena; Sharma, Kalicharan; Shafi, Syed; Samim, Mohammed; Javed, Kalim; Supuran, Claudiu T
Synthesis, biological evaluation, and enzyme docking simulations of 1,5-diarylpyrrole-3-alkoxyethyl ethers as selective cyclooxygenase-2 inhibitors endowed with anti-inflammatory and antinociceptive activity. 2008 Maurizio Anzini; Michele Rovini; Andrea Cappelli; Salvatore Vomero; Fabrizio Manetti; Maurizio Botta; Lidia Sautebin; Antonietta Rossi; Carlo Pergola; Carla Ghelardini; Monica Norcini; Antonio Giordani; Francesco Makovec; Paola Anzellotti; Paola Patrignani; Mariangela Biava
Synthesis, biological evaluation, and in silico studies of potential activators of apoptosis and carbonic anhydrase inhibitors on isatin-5-sulfonamide scaffold 2022 Stepan K. Krymov; Alexander M. Scherbakov; Diana I. Salnikova; Danila V. Sorokin; Lyubov G. Dezhenkova; Ivan V. Ivanov; Daniela Vullo; Viviana De Luca; Clemente Capasso; Claudiu T. Supuran; Andrey E. Shchekotikhin
Synthesis, biological evaluation, and molecular modelling studies of potent human neutrophil elastase (HNE) inhibitors 2018 Giovannoni, Maria Paola; Schepetkin, Igor A.; Quinn, Mark T.; Cantini, Niccolò; Crocetti, Letizia*; Guerrini, Gabriella; Iacovone, Antonella; Paoli, Paola; Rossi, Patrizia; Bartolucci, Gian Luca; Menicatti, Marta; Vergelli, Claudia
Synthesis, biological evaluation, and receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as kappa-opioid receptor agonists endowed with antinociceptive and antiamnesic activity. 2003 Maurizio Anzini; Laura Canullo; Carlo Braile; Andrea Cappelli; Andrea Gallelli; Salvatore Vomero; M. Cristina Menziani; Pier G De; Milena Rizzo; Simona Collina; Ornella Azzolina; Massimo Sbacchi; Carla Ghelardini; Nicoletta Galeotti
Synthesis, biological evaluation, molecular modeling, and structural analysis of new pyrazole and pyrazolone derivatives as N-formyl peptide receptors agonists 2021 Vergelli C.; Khlebnikov A.I.; Crocetti L.; Guerrini G.; Cantini N.; Kirpotina L.N.; Schepetkin I.A.; Cilibrizzi A.; Quinn M.T.; Rossi P.; Paoli P.; Giovannoni M.P.
Synthesis, carbonic anhydrase I and II inhibition studies of the 1,3,5-trisubstituted-pyrazolines 2017 Gul, Halise Inci; Mete, Ebru; Taslimi, Parham; Gulcin, Ilhami; Supuran, Claudiu T
Synthesis, carbonic anhydrase inhibition and cytotoxic activity of novel chromone-based sulfonamide derivatives 2015 Awadallah, Fadi M; El-Waei, Tamer A.; Hanna, Mona M.; Abbas, Safinaz E.; Ceruso, Mariangela; Oz, Beyza Ecem; Guler, Ozen Ozensoy; Supuran, Claudiu T.
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids 2024 Morteza Abdoli; Alessandro Bonardi; Paola Gratteri; Claudiu T Supuran; Raivis Žalubovskis
Synthesis, characterisation, biological evaluation and in silico studies of sulphonamide Schiff bases 2020 Durgun, Mustafa; Türkeş, Cüneyt; Işık, Mesut; Demir, Yeliz; Saklı, Ali; Kuru, Ali; Güzel, Abdussamat; Beydemir, Şükrü; Akocak, Suleyman; Osman, Sameh M; AlOthman, Zeid; Supuran, Claudiu T
Synthesis, characterization and application of Ni(tta)2.tmeda to MOCVD of nickel oxide thin films 2006 G. Malandrino; L. M. S. Perdicaro;G. Condorelli; I. L. Fragala; P. Rossi; P. Dapporto
Synthesis, characterization and applicative study of innovative materials for the conservation of cellulosic artifacts with an artistic and architectural interest 2017 Papacchini, Alessandra
Synthesis, characterization and basicity properties of two new oxa-aza macrobicyclic receptors. Crystal structure of a "Water Cryptate" 1994 C.Bazzicalupi; A.Bencini; A.Bianchi; V.Fusi; P.Paoletti; B.Valtancoli
Synthesis, characterization and biological activity evaluation of a dual-drug based on the antibacterial peptide lugdunin functionalized with the Carbonic Anhydrase sulfonamide inhibitor acetazolamide 2024 Quagliata, M.; Brenzini Biagioni, F.; Giovannuzzi, S.; De Luca, V.; Capasso, C.; Nocentini, A.; Supuran, C. T.; Rovero, P.; Papini, A.M
. Synthesis, characterization and biological activity evaluation of a dual-drug based on the antibacterial peptide lugdunin functionalized with the carbonic anhydrase sulfonamide inhibitor acetazolamide 2024 M. Quagliata; F. Brenzini Biagioni; S. Giovannuzzi; V. De Luca; C. Capasso; A. Nocentini; C.T. Supuran; P. Rovero; A.M. Papini
Synthesis, characterization and biological studies of sulfonamide Schiff's bases and some of their metal derivatives. 2012 Z. H. Chohan;H. A. Shad;C. T. Supuran
Synthesis, characterization and carbonic anhydrase inhibitory activity of novel benzothiazole derivatives 2016 Küçükbay, F. Zehra; Buğday, Nesrin; Küçükbay, Hasan; Tanc, Muhammet; Supuran, Claudiu T.
Synthesis, characterization and CO2 uptake of a chiral Co(II) metal-organic framework containing a thiazolidine-based spacer 2012 Rossin A; Di Credico B; Giambastiani G; Peruzzini M; Pescitelli G; Reginato G; Borfecchia E; Gianolio D; Lamberti C; Bordiga S
Mostrati risultati da 241.903 a 241.922 di 270.005
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