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N-Bridgehead polycyclic compounds by sequential rearrangement-annulation of isoxazoline-5-spirocyclopropanes. 6. A general synthetic method of 5,6-dihydro-7(8H)- and 2,3,5,6-tetrahydro-7(1H)-indolizinones 1992 E. OCCHIATO; A. GUARNA; A. BRANDI; A. GOTI; F. DE SARLO
HIGH-PERFORMANCE LIQUID CHROMATOGRAPHIC DETERMINATION OF 3,5-DIMETHYLHYPPURIC ACID IN THE OCCUPATIONAL EXPOSURE TO TRIMETHYLBENZENES 1992 E. OCCHIATO; S. BUSINI; P. BAVAZZANO
Pharmacokinetics of 4-hydroxyandrostenedione in man after intramuscular injection of different formulations and the effect of this drug on plasma aromatizable androgens and 17beta-estradiol concentrations. 1993 Danza G; Muratori M; Guarna A; Occhiato EG; Sadri R; Serio M
ENANTIOSELECTIVE SYNTHESIS OF INDOLIZINE DERIVATIVES BY REARRANGEMENT-CYCLIZATION OF ISOXAZOLINE-5-SPIROCYCLOPROPANES 1993 E. OCCHIATO; A. GUARNA; M. SPINETTI
Rearrangement of isoxazoline-5-spirocyclopropanes. Part 9. Synthesis of medium-size azaheterocycles 1993 E. OCCHIATO; A. GUARNA; F. DE SARLO; A. BRANDI; A. GOTI; P. PAOLI; P. DAPPORTO
BAKER'S YEAST REDUCTION OF PROCHIRAL G-NITROKETONES: ENANTIOSELECTIVE SYNTHESIS OF (S)-4-NITROALCOHOLS 1995 A. GUARNA; E. OCCHIATO; D. SCARPI; L. SPINETTI; M. VALLECCHI
Baker's yeast reduction of prochiral g-nitro ketones. II. Straightforward enantioselective synthesis of 2,7-dimethyl-1,6-dioxaspiro[4.4]nonanes 1995 E. OCCHIATO; A. GUARNA; F. DE SARLO; D. SCARPI
ASYMMETRIC HYDROGENATION OF PROCHIRAL G-NITROKETONES BY RUTHENIUM COMPLEXES 1996 D. SCARPI; G. MENCHI; E. OCCHIATO; A. GUARNA
PROBING ENZYME STEREOSPECIFICITY. INHIBITION OF A-CHYMOTRYPSIN AND SUBTILISIN CARLSBERG BY CHIRAL AMINE- AND AMINOALCOHOL-DERIVATIVES 1996 E. OCCHIATO; J. JONES
SYNTHESIS OF ENANTIOPURE 2,7-DIARYL-1,6-DIOXASPIRO[4.4]NONANES VIA ENANTIOSELECTIVE REDUCTION OF PROCHIRAL G-NITROKETONES BY DIISOPINOCAMPHEYLCHLOROBORANE (DIP-CLTM) 1996 E. OCCHIATO; D. SCARPI; G. MENCHI; A. GUARNA
19-nor-10-azasteroids: a novel class of inhibitors for human steroid 5alpha-reductases 1 and 2 1997 A. GUARNA; C. BELLE; F. MACHETTI; E. OCCHIATO; A. H. PAYNE; C. CASSIANI; A; COMERCI; G. DANZA; A. DE BELLIS; S. DINI; A. MARRUCCI; M. SERIO
19-nor-10-azasteroids, a new class of steroid 5a-reductase inhibitors. 2. X-ray structure, molecular modeling, conformational analysis of 19-nor-10-azasteroids and comparison with 4-azasteroids and 6-azasteroids 1997 A. GUARNA; E. OCCHIATO; F. MACHETTI; G. DANZA; M. SERIO; P. PAOLI; A. MARRUCCI
Synthesis of benzo[c]quinolizin-3-ones: selective non steroidal inhibitors of steroid 5a-Reductase 1 1998 A. GUARNA; E. G. OCCHIATO; D. SCARPI; R. TSAI; G. DANZA; A. COMERCI; R. MANCINA; M. SERIO
Process for the synthesis of (1H)-benzo[c]quinolizin-3-ones derivatives 1998 GUARNA A; SERIO M; E. OCCHIATO
5A-REDUCTASE INHIBITORS, CHEMICAL AND CLINICAL MODELS 1998 A. GUARNA; E. OCCHIATO; G. DANZA; A. CONTI; M. SERIO
5alpha-reductase ihnibitors, chemical and clinical models 1998 A. GUARNA; E.G. OCCHIATO; G. DANZA; A. CONTI; M. SERIO
MICROBIAL BIOTRANFORMATIONS IN WATER/ORGANIC SOLVENT SYSTEM. ENANTIOSELECTIVE REDUCTION OF AROMATIC B- AND G-NITROKETONES 1998 F. MOLINARI; E. OCCHIATO; A. GUARNA; F. ARAGOZZINI
STEREOSELECTIVITY IN THE TICL4-CATALYSED REEACTION OF DANISHEFSKY¿S DIENE WITH A N-(ACYLOXY)IMINIUM ION: SYNTHESIS OF 5A VERSUS 5B D1(2)-19-NOR-10-AZASTEROIDS. PART 4 1998 E. OCCHIATO; D. SCARPI; F. MACHETTI; A. GUARNA
A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5-REDUCTASE INHIBITORS. 3.1 SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-17B-ACETYLOXY-(5B)-10-AZAESTR-1-EN-3-ONE 1998 A. GUARNA; E. OCCHIATO; F. MACHETTI; D. SCARPI
Synthesis and reactivity of bicycles derived from tartaric acids and alfa-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid 1999 A. GUARNA; A. GUIDI; F. MACHETTI; G. MENCHI; E. OCCHIATO; D. SCARPI; S. SISI; A. TRABOCCHI
Mostrati risultati da 1 a 20 di 126
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