Sfoglia per Autore
Platinum(II) Complexes with O,S Bidentate Ligands: Biophysical Characterization, Antiproliferative Activity, and Crystallographic Evidence of Protein Binding
2015 Mügge, Carolin; Marzo, Tiziano; Massai, Lara; Hildebrandt, Jana; Ferraro, Giarita; Rivera-Fuentes, Pablo; Metzler-Nolte, Nils; Merlino, Antonello; Messori, Luigi; Weigand, Wolfgang
Evidence that the antiproliferative effects of auranofin in Saccharomyces cerevisiae arise from inhibition of mitochondrial respiration
2015 Gamberi, T; Fiaschi, T; Modesti, A; Massai, L; Messori, L; Balzi, M; Magherini, F.
Interactions of selected gold(III) complexes with DNA G quadruplexes
2015 P. Gratteri; L. Massai; E. Michelucci; R. Rigo; L. Messori; M. A. Cinellu; C. Musetti; C. Sissi; C. Bazzicalupi
Reactions of Cytotoxic Metallodrugs with Lysozyme in pure DMSO explored through UV-Vis Absorption Spectroscopy and ESI MS
2015 Tiziano Marzo; Aleksandar Savić; Lara Massai; Elena Michelucci; Tibor J. Sabo; Sanja Grguric-Šipka; Luigi Messori
Interaction of anticancer Ru(III) complexes with single stranded and duplex DNA model systems
2015 Musumeci, Domenica; Rozza, Lucia; Merlino, Antonello; Paduano, Luigi; Marzo, Tiziano; Massai, Lara; Messori, Luigi; Montesarchio, Daniela
Reactions of model proteins with aurothiomalate, a clinically established gold(I) drug: The comparison with auranofin
2015 Farivash Darabi; Tiziano Marzo; Lara Massai; Federica Scaletti; Elena Michelucci; Luigi Messori
Antiproliferative properties and biomolecular interactions of three Pd(II) and Pt(II) complexes
2016 Massai, Lara; Pratesi, Alessandro; Bogojeski, Jovana; Banchini, Marco; Pillozzi, Serena; Messori, Luigi; Bugarčić, Živadin D
Elucidating the reactivity of Pt(II) complexes with (O,S) bidentate ligands towards DNA model systems
2016 Mügge, Carolin; Musumeci, Domenica; Michelucci, Elena; Porru, Francesca; Marzo, Tiziano; Massai, Lara; Messori, Luigi; Weigand, Wolfgang; Montesarchio, Daniela
Organogold(III) compounds as experimental anticancer agents: chemical and biological profiles
2016 Massai, Lara; Cirri, Damiano; Michelucci, Elena; Bartoli, Gianluca; Guerri, Annalisa; Cinellu, Maria A.; Cocco, Fabio; Gabbiani, Chiara; Messori, Luigi
A first-in-class and a fished out anticancer platinum compound:: Cis -[PtCl2(NH3)2] and cis -[PtI2(NH3)2] compared for their reactivity towards DNA model systems
2016 Musumeci, Domenica; Platella, Chiara; Riccardi, Claudia; Merlino, Antonello; Marzo, Tiziano; Massai, Lara; Messori, Luigi; Montesarchio, Daniela
Cytotoxic properties of a new organometallic platinum(II) complex and its gold(I) heterobimetallic derivatives.
2016 Serratrice, M; Maiore, L; Zucca, A; Stoccoro, S; Landini, I; Mini, E; Massai, L; Ferraro, G; Merlino, A; Messori, L; Cinellu, Ma
Determinants for Tight and Selective Binding of a Medicinal Dicarbene Gold(I) Complex to a Telomeric DNA G-Quadruplex: a Joint ESI MS and XRD Investigation
2016 Bazzicalupi, Carla; Ferraroni, Marta; Papi, Francesco; Massai, Lara; Bertrand, Benoît; Messori, Luigi; Gratteri, Paola; Casini, Angela
Gold compounds as cysteine protease inhibitors: perspectives for pharmaceutical application as antiparasitic agents
2017 Massai, Lara; Messori, Luigi; Micale, Nicola; Schirmeister, Tanja; Maes, Louis; Fregona, Dolores; Cinellu, Maria Agostina; Gabbiani, Chiara*
Na/K-ATPase as a target for anticancer metal based drugs: insights into molecular interactions with selected gold(iii) complexes
2017 Bondžić, Aleksandra M.; Janjić, Goran V.; Dramićanin, Miroslav D.; Messori, Luigi; Massai, Lara; Parac Vogt, Tatjana N.; Vasić, Vesna M.
[Au(9-methylcaffein-8-ylidene)2]+/DNA Tel23 System: Solution, Computational, and Biological Studies
2017 Papi, Francesco; Bazzicalupi, Carla; Ferraroni, Marta; Massai, Lara; Bertrand, Benoit; Gratteri, Paola; Colangelo, Donato; Messori, Luigi
Cell and Cell-Free Mechanistic Studies on Two Gold(III) Complexes with Proven Antitumor Properties
2017 Nardon, Chiara; Boscutti, Giulia; Gabbiani, Chiara; Massai, Lara; Pettenuzzo, Nicolò; Fassina, Ambrogio; Messori, Luigi; Fregona, Dolores*
Selection and characterization of a human ovarian cancer cell line resistant to auranofin
2017 Landini, I; Lapucci, A; Pratesi, A; Massai, L; Napoli, C; Perrone, G; Pinzani, P; Messori, L; Mini, E; Nobili, S.
Antiproliferative effects of two gold(I)-N-heterocyclic carbene complexes in A2780 human ovarian cancer cells: A comparative proteomic study
2018 Magherini, Francesca; Fiaschi, Tania; Valocchia, Elisa; Becatti, Matteo; Pratesi, Alessandro; Marzo, Tiziano; Massai, Lara; Gabbiani, Chiara; Landini, Ida; Nobili, Stefania; Mini, Enrico; Messori, Luigi; Modesti, Alessandra; Gamberi, Tania*
The cisplatin/serum albumin system: A reappraisal
2019 Massai, Lara; Pratesi, Alessandro; Gailer, Jurgen; Marzo, Tiziano; Messori, Luigi
Replacement of the Thiosugar of Auranofin with Iodide Enhances the Anticancer Potency in a Mouse Model of Ovarian Cancer
2019 Tiziano Marzo, Lara Massai, Alessandro Pratesi, Matteo Stefanini, Damiano Cirri, Francesca Magherini, Matteo Becatti, Ida Landini, Stefania Nobili, Enrico Mini, Olivia Crociani, Annarosa Arcangeli, Serena Pillozzi, Tania Gamberi, Luigi Messori
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Platinum(II) Complexes with O,S Bidentate Ligands: Biophysical Characterization, Antiproliferative Activity, and Crystallographic Evidence of Protein Binding | 2015 | Mügge, Carolin; Marzo, Tiziano; Massai, Lara; Hildebrandt, Jana; Ferraro, Giarita; Rivera-Fuentes, Pablo; Metzler-Nolte, Nils; Merlino, Antonello; Messori, Luigi; Weigand, Wolfgang | |
Evidence that the antiproliferative effects of auranofin in Saccharomyces cerevisiae arise from inhibition of mitochondrial respiration | 2015 | Gamberi, T; Fiaschi, T; Modesti, A; Massai, L; Messori, L; Balzi, M; Magherini, F. | |
Interactions of selected gold(III) complexes with DNA G quadruplexes | 2015 | P. Gratteri; L. Massai; E. Michelucci; R. Rigo; L. Messori; M. A. Cinellu; C. Musetti; C. Sissi; C. Bazzicalupi | |
Reactions of Cytotoxic Metallodrugs with Lysozyme in pure DMSO explored through UV-Vis Absorption Spectroscopy and ESI MS | 2015 | Tiziano Marzo; Aleksandar Savić; Lara Massai; Elena Michelucci; Tibor J. Sabo; Sanja Grguric-Šipka; Luigi Messori | |
Interaction of anticancer Ru(III) complexes with single stranded and duplex DNA model systems | 2015 | Musumeci, Domenica; Rozza, Lucia; Merlino, Antonello; Paduano, Luigi; Marzo, Tiziano; Massai, Lara; Messori, Luigi; Montesarchio, Daniela | |
Reactions of model proteins with aurothiomalate, a clinically established gold(I) drug: The comparison with auranofin | 2015 | Farivash Darabi; Tiziano Marzo; Lara Massai; Federica Scaletti; Elena Michelucci; Luigi Messori | |
Antiproliferative properties and biomolecular interactions of three Pd(II) and Pt(II) complexes | 2016 | Massai, Lara; Pratesi, Alessandro; Bogojeski, Jovana; Banchini, Marco; Pillozzi, Serena; Messori, Luigi; Bugarčić, Živadin D | |
Elucidating the reactivity of Pt(II) complexes with (O,S) bidentate ligands towards DNA model systems | 2016 | Mügge, Carolin; Musumeci, Domenica; Michelucci, Elena; Porru, Francesca; Marzo, Tiziano; Massai, Lara; Messori, Luigi; Weigand, Wolfgang; Montesarchio, Daniela | |
Organogold(III) compounds as experimental anticancer agents: chemical and biological profiles | 2016 | Massai, Lara; Cirri, Damiano; Michelucci, Elena; Bartoli, Gianluca; Guerri, Annalisa; Cinellu, Maria A.; Cocco, Fabio; Gabbiani, Chiara; Messori, Luigi | |
A first-in-class and a fished out anticancer platinum compound:: Cis -[PtCl2(NH3)2] and cis -[PtI2(NH3)2] compared for their reactivity towards DNA model systems | 2016 | Musumeci, Domenica; Platella, Chiara; Riccardi, Claudia; Merlino, Antonello; Marzo, Tiziano; Massai, Lara; Messori, Luigi; Montesarchio, Daniela | |
Cytotoxic properties of a new organometallic platinum(II) complex and its gold(I) heterobimetallic derivatives. | 2016 | Serratrice, M; Maiore, L; Zucca, A; Stoccoro, S; Landini, I; Mini, E; Massai, L; Ferraro, G; Merlino, A; Messori, L; Cinellu, Ma | |
Determinants for Tight and Selective Binding of a Medicinal Dicarbene Gold(I) Complex to a Telomeric DNA G-Quadruplex: a Joint ESI MS and XRD Investigation | 2016 | Bazzicalupi, Carla; Ferraroni, Marta; Papi, Francesco; Massai, Lara; Bertrand, Benoît; Messori, Luigi; Gratteri, Paola; Casini, Angela | |
Gold compounds as cysteine protease inhibitors: perspectives for pharmaceutical application as antiparasitic agents | 2017 | Massai, Lara; Messori, Luigi; Micale, Nicola; Schirmeister, Tanja; Maes, Louis; Fregona, Dolores; Cinellu, Maria Agostina; Gabbiani, Chiara* | |
Na/K-ATPase as a target for anticancer metal based drugs: insights into molecular interactions with selected gold(iii) complexes | 2017 | Bondžić, Aleksandra M.; Janjić, Goran V.; Dramićanin, Miroslav D.; Messori, Luigi; Massai, Lara; Parac Vogt, Tatjana N.; Vasić, Vesna M. | |
[Au(9-methylcaffein-8-ylidene)2]+/DNA Tel23 System: Solution, Computational, and Biological Studies | 2017 | Papi, Francesco; Bazzicalupi, Carla; Ferraroni, Marta; Massai, Lara; Bertrand, Benoit; Gratteri, Paola; Colangelo, Donato; Messori, Luigi | |
Cell and Cell-Free Mechanistic Studies on Two Gold(III) Complexes with Proven Antitumor Properties | 2017 | Nardon, Chiara; Boscutti, Giulia; Gabbiani, Chiara; Massai, Lara; Pettenuzzo, Nicolò; Fassina, Ambrogio; Messori, Luigi; Fregona, Dolores* | |
Selection and characterization of a human ovarian cancer cell line resistant to auranofin | 2017 | Landini, I; Lapucci, A; Pratesi, A; Massai, L; Napoli, C; Perrone, G; Pinzani, P; Messori, L; Mini, E; Nobili, S. | |
Antiproliferative effects of two gold(I)-N-heterocyclic carbene complexes in A2780 human ovarian cancer cells: A comparative proteomic study | 2018 | Magherini, Francesca; Fiaschi, Tania; Valocchia, Elisa; Becatti, Matteo; Pratesi, Alessandro; Marzo, Tiziano; Massai, Lara; Gabbiani, Chiara; Landini, Ida; Nobili, Stefania; Mini, Enrico; Messori, Luigi; Modesti, Alessandra; Gamberi, Tania* | |
The cisplatin/serum albumin system: A reappraisal | 2019 | Massai, Lara; Pratesi, Alessandro; Gailer, Jurgen; Marzo, Tiziano; Messori, Luigi | |
Replacement of the Thiosugar of Auranofin with Iodide Enhances the Anticancer Potency in a Mouse Model of Ovarian Cancer | 2019 | Tiziano Marzo, Lara Massai, Alessandro Pratesi, Matteo Stefanini, Damiano Cirri, Francesca Magherini, Matteo Becatti, Ida Landini, Stefania Nobili, Enrico Mini, Olivia Crociani, Annarosa Arcangeli, Serena Pillozzi, Tania Gamberi, Luigi Messori |
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