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Benzodiazepine receptor ligands. Part III. Synthesis and biological evaluation of 2 and/or 3-substituted pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides. 1999 G. GUERRINI; A. COSTANZO; F. BRUNI; G. CICIANI; S. SELLERI; P. GRATTERI; B. COSTA; C. MARTINI; A. LUCACCHINI
Benzodiazepine receptor ligands. 4.Synthesis, and pharmacological evaluation of 3-hetroaryl-8-chloro pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides. 1999 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; S. SELLERI; B. COSTA; C. MARTINI; A. LUCACCHINI; P. MALMBERG AIELLO; A. IPPONI
Benzodiazepine receptor ligands. 4. Synthesis and pharmacological evaluation of 3-heteroaryl-8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5- oxides 1999 Costanzo A.; Guerrini G.; Ciciani G.; Bruni F.; Selleri S.; Costa B.; Martini C.; Lucacchini A.; Malmberg Aiello P.; Ipponi A.
Synthesis and BZR affinity of pyrazolo [ 1,5-a ] pyrimidine derivatives. Part 2:Further Investigation on the 3-aryl substituents. 2000 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. MALBERG; C. LAMBERTI; B. COSTA; C. MARTINI
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective Peripheral Benzodiazepine Receptor ligands 2001 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; B. COSTA; C. MARTINI
Benzodiazepine receptor ligands. 6. New 3-(2-,3- or 4-substituted benzyloxycarbonyl) derivatives of 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide receptor affinity and In vivo testing C. Martini, P. Malmberg Aiello 2001 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; C. COSTAGLI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG AIELLO
Synthesis and pharmacological evaluation of 3-(2-furyl)- and 3-(3-furyl)-(-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxides, new 3-heteroaryl substituted benzodiazepine receptor ligands. 2002 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; C. COSTAGLI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG AIELLO
BENZODIAZEPINE RECEPTOR LIGANDS. 7. SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF NEW 3-ESTERS OF THE 8-CHLOROPYRAZOLO[5,1-C][1,2,4]BENZOTRIAZINE 5-OXIDE. 3-(2- THIENYLMETHOXYCARBONYL) DERIVATIVE: AN ANXIOSELECTIVE AGENT IN RODENTS. 2002 F. BRUNI; P. MALMBERG; A. COSTANZO; G. CICIANI; G. GUERRINI; S. SELLERI; C. COSTAGLI; C. MARTINI; B. COSTA; F. BESNARD
Synthesis and Benzodiazepine Receptor Affinity of Pyrazolo [1,5-a]pyrimidine Derivatives.3. New 6-(3-Thienyl) Series as a1 Selective Ligands 2003 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; P.GRATTERI; C.BONACCINI; P.MALMBERG AIELLO; F.BESNARD; S.RENARD; B. COSTA; C. MARTINI
Insight into 2-phenylpyrazolo[1,5-a]pyrimidin-3-yl acetamides as Peripheral Benzodiazepine Receptor Ligands: synthesis, biological evaluation and 3D-QSAR investigation. 2005 S. SELLERI; P. GRATTERI; C. COSTAGLI; C. BONACCINI; A. COSTANZO; F. MELANI; G. GUERRINI; G. CICIANI; B. COSTA; C. MARTINI; F. BRUNI; F. SPINETTI
Cytotoxic activity of 3-nitropyrazolo[5,1-c][1,2,4]benzotriazine derivatives: a new series of anti-proliferative agents. 2005 M. CORONNELLO; G. CICIANI; E. MINI; G. GUERRINI; B. CACIAGLI; S. SELLERI; A. COSTANZO; T. MAZZEI
A novel selective GABA-A alpha1 receptor agonist displaying sedative and anxiolytic-like properties in rodents. 2005 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. GRATTERI; F. BESNARD; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; M. MONTALI; J. FOHLIN
Benzodiazepine receptor ligands. 8. Synthesis and pharamcological evaluation of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide 3- and 8-disubstituted: high affinity ligands endowed with inverse-agonist pharmacological efficacy. 2006 G. GUERRINI; A. COSTANZO; G. CICIANI; F. BRUNI; S. SELLERI; C. COSTAGLI; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; F. BESNARD
Novel 3-iodo-8-ethoxypyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide as promising lead for design of alpha5-inverse agonist, useful tools for therapy of mnemonic damage. 2007 G. GUERRINI; G. CICIANI; G. CAMBI; F. BRUNI; S. SELLERI; F. BESNARD; M. MONTALI; C. MARTINI; C. GHELARDINI; N. GALEOTTI; A. COSTANZO
Novel 3-aroylpyrazolo[5,1-c][1,2,4] benzotriazines 5-oxides 8-substituted, ligands at GABAA/benzodiazepine receptor complex: synthesis, pharmacological and molecular modelling studies. 2008 G. Guerrini; G. Ciciani; G. Cambi; F. Bruni; S. Selleri; F. Melani; M. Montali; C. Martini; C. Ghelardini; M. Norcini; A. Costanzo
Synthesis of new pyrazolo[5,1-c][1,2,4]benzotriazines, pyrazolo[5,1-c]pyrido[4,3-e][1,2,4]triazines and their open analogues as cytotoxic agents in normoxic and hypoxic conditions. 2008 G. Ciciani; M. Coronnello; G. Guerrini; S.Selleri; M.Cantore; P. Failli; E. Mini; A. Costanzo
Synthesis, in vivo evaluation, and molecular modeling studies of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide derivatives. Identification of a bifunctional hydrogen bond area related to the inverse-agonism 2009 G. Guerrini; G. Ciciani; G. Cambi; F. Bruni; S.Selleri; C. Guarino; F. Melani; M. Montali; C: Martini; C. Ghelardini; M. Norcini; A. Costanzo
ChemInform Abstract: Reactivity of 7‐(2‐Dimethylaminovinyl)pyrazolo(1,5‐a)pyrimidines: Synthesis of Pyrazolo(1,5‐a)pyrido(3,4‐e)pyrimidine Derivatives as Potential Benzodiazepine Receptor Ligands. Part 1 2010 BRUNI, F.; SELLERI, S.; COSTANZO, A.; GUERRINI, G.; CASILLI, M. L.
ChemInform Abstract: Pyrazolo(1,5‐a)pyrido(3,4‐e)pyrimidin‐6‐ones. Part 1. Synthesis and in vitro Antimicrobial Evaluation 2010 BRUNI, F.; SELLERI, S.; COSTANZO, A.; GUERRINI, G.; CASILLI, M. L.; SACCO, C.; DONATO, R.
New fluoro derivatives of the pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide system: evaluation of fluorine binding properties in the benzodiazepine site on gamma-aminobutyrric acid type A (GABAA) receptor. Design, synthesis, biological evaluation, and molecular modeling investigation. 2010 G. Guerrini; G. Ciciani; F. Bruni; S. Selleri; C. Guarino; F. Melani; M. Montali; S. Daniele; C. Martini; C. Ghelardini; M. Norcini; S. Ciattini; A. Costanzo
Mostrati risultati da 41 a 60 di 63
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