Sfoglia per Autore
Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors
2020 Berrino E.; Angeli A.; Zhdanov D.D.; Kiryukhina A.P.; Milaneschi A.; De Luca A.; Bozdag M.; Carradori S.; Selleri S.; Bartolucci G.; Peat T.S.; Ferraroni M.; Supuran C.T.; Carta F.
N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions
2020 Poli G.; Bozdag M.; Berrino E.; Angeli A.; Tuccinardi T.; Carta F.; Supuran C.T.
New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies
2020 Abdel-Mohsen, Heba T; El Kerdawy, Ahmed M; Omar, Mohamed A; Berrino, Emanuela; Abdelsamie, Ahmed S; El Diwani, Hoda I; Supuran, Claudiu T
Zeta-carbonic anhydrases show CS2 hydrolase activity: A new metabolic carbon acquisition pathway in diatoms?
2021 Alterio V.; Langella E.; Buonanno M.; Esposito D.; Nocentini A.; Berrino E.; Bua S.; Polentarutti M.; Supuran C.T.; Monti S.M.; De Simone G.
An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
2021 Mansoldo F.R.P.; Berrino E.; Guglielmi P.; Carradori S.; Carta F.; Secci D.; Supuran C.T.; Vermelho A.B.
Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages
2021 Berrino E.; Carradori S.; Angeli A.; Carta F.; Supuran C.T.; Guglielmi P.; Coletti C.; Paciotti R.; Schweikl H.; Maestrelli F.; Cerbai E.; Gallorini M.
Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors
2021 Plyasova A.A.; Berrino E.; Khan I.I.; Veselovsky A.V.; Pokrovsky V.S.; Angeli A.; Ferraroni M.; Supuran C.T.; Pokrovskaya M.V.; Alexandrova S.S.; Gladilina Y.A.; Sokolov N.N.; Hilal A.; Carta F.; Zhdanov D.D.
Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies
2021 Baglini, Emma; Ravichandran, Rahul; Berrino, Emanuela; Salerno, Silvia; Barresi, Elisabetta; Marini, Anna Maria; Viviano, Monica; Castellano, Sabrina; Da Settimo, Federico; Supuran, Claudiu T; Cosconati, Sandro; Taliani, Sabrina
Amine-and amino acid-based compounds as carbonic anhydrase activators
2021 Angeli A.; Berrino E.; Carradori S.; Supuran C.T.; Cirri M.; Carta F.; Costantino G.
Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution
2021 Emanuela Berrino; Bastien Michelet; Agnes Martin-Mingot; Fabrizio Carta; Claudiu Supuran; Sebastien Thibaudeau
Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
2022 Pontecorvi V.; Mori M.; Picarazzi F.; Zara S.; Carradori S.; Cataldi A.; Angeli A.; Berrino E.; Chimenti P.; Ciogli A.; Secci D.; Guglielmi P.; Supuran C.T.
Uncovering Novel Capsaicin Inhibitory Activity towards Human Carbonic Anhydrase Isoforms IX and XII by Combining In Silico and In Vitro Studies
2023 Gualtieri G.; Maruca A.; Rocca R.; Carta F.; Berrino E.; Salatino A.; Brescia C.; Torcasio R.; Crispo M.; Trapasso F.; Alcaro S.; Supuran C.T.; Costa G.
Design and synthesis of 6-arylpyridine-tethered sulfonamides as novel selective inhibitors of carbonic anhydrase IX with promising antitumor features toward the human colorectal cancer
2023 Eldehna, Wagdy M.; Mohammed, Eslam E.; Al-Ansary, Ghada H.; Berrino, Emanuela; Elbadawi, Mostafa M.; Ibrahim, Tamer M.; Jaballah, Maiy Y.; Al-Rashood, Sara T.; Binjubair, Faizah A.; Celik, Meltem; Nocentini, Alessio; Elbarbry, Fawzy A.; Sahin, Fikrettin; Abdel-Aziz, Hatem A.; Supuran, Claudiu T.; Fares, Mohamed
Escinosome thermosensitive gel optimizes efficacy of CAI-CORM in a rat model of rheumatoid arthritis
2023 Vanti, Giulia; Micheli, Laura; Berrino, Emanuela; Mannelli, Lorenzo Di Cesare; Bogani, Irene; Carta, Fabrizio; Bergonzi, Maria Camilla; Supuran, Claudiu T; Ghelardini, Carla; Bilia, Anna Rita
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors | 2020 | Berrino E.; Angeli A.; Zhdanov D.D.; Kiryukhina A.P.; Milaneschi A.; De Luca A.; Bozdag M.; Carradori S.; Selleri S.; Bartolucci G.; Peat T.S.; Ferraroni M.; Supuran C.T.; Carta F. | |
| N-aryl-N′-ureido-O-sulfamates as potent and selective inhibitors of hCA VB over hCA VA: Deciphering the binding mode of new potential agents in mitochondrial dysfunctions | 2020 | Poli G.; Bozdag M.; Berrino E.; Angeli A.; Tuccinardi T.; Carta F.; Supuran C.T. | |
| New thiopyrimidine-benzenesulfonamide conjugates as selective carbonic anhydrase II inhibitors: synthesis, in vitro biological evaluation, and molecular docking studies | 2020 | Abdel-Mohsen, Heba T; El Kerdawy, Ahmed M; Omar, Mohamed A; Berrino, Emanuela; Abdelsamie, Ahmed S; El Diwani, Hoda I; Supuran, Claudiu T | |
| Zeta-carbonic anhydrases show CS2 hydrolase activity: A new metabolic carbon acquisition pathway in diatoms? | 2021 | Alterio V.; Langella E.; Buonanno M.; Esposito D.; Nocentini A.; Berrino E.; Bua S.; Polentarutti M.; Supuran C.T.; Monti S.M.; De Simone G. | |
| An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods | 2021 | Mansoldo F.R.P.; Berrino E.; Guglielmi P.; Carradori S.; Carta F.; Secci D.; Supuran C.T.; Vermelho A.B. | |
| Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages | 2021 | Berrino E.; Carradori S.; Angeli A.; Carta F.; Supuran C.T.; Guglielmi P.; Coletti C.; Paciotti R.; Schweikl H.; Maestrelli F.; Cerbai E.; Gallorini M. | |
| Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase-Carbonic Anhydrase Dual-Hybrid Inhibitors | 2021 | Plyasova A.A.; Berrino E.; Khan I.I.; Veselovsky A.V.; Pokrovsky V.S.; Angeli A.; Ferraroni M.; Supuran C.T.; Pokrovskaya M.V.; Alexandrova S.S.; Gladilina Y.A.; Sokolov N.N.; Hilal A.; Carta F.; Zhdanov D.D. | |
| Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies | 2021 | Baglini, Emma; Ravichandran, Rahul; Berrino, Emanuela; Salerno, Silvia; Barresi, Elisabetta; Marini, Anna Maria; Viviano, Monica; Castellano, Sabrina; Da Settimo, Federico; Supuran, Claudiu T; Cosconati, Sandro; Taliani, Sabrina | |
| Amine-and amino acid-based compounds as carbonic anhydrase activators | 2021 | Angeli A.; Berrino E.; Carradori S.; Supuran C.T.; Cirri M.; Carta F.; Costantino G. | |
| Modulating the Efficacy of Carbonic Anhydrase Inhibitors through Fluorine Substitution | 2021 | Emanuela Berrino; Bastien Michelet; Agnes Martin-Mingot; Fabrizio Carta; Claudiu Supuran; Sebastien Thibaudeau | |
| Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies | 2022 | Pontecorvi V.; Mori M.; Picarazzi F.; Zara S.; Carradori S.; Cataldi A.; Angeli A.; Berrino E.; Chimenti P.; Ciogli A.; Secci D.; Guglielmi P.; Supuran C.T. | |
| Uncovering Novel Capsaicin Inhibitory Activity towards Human Carbonic Anhydrase Isoforms IX and XII by Combining In Silico and In Vitro Studies | 2023 | Gualtieri G.; Maruca A.; Rocca R.; Carta F.; Berrino E.; Salatino A.; Brescia C.; Torcasio R.; Crispo M.; Trapasso F.; Alcaro S.; Supuran C.T.; Costa G. | |
| Design and synthesis of 6-arylpyridine-tethered sulfonamides as novel selective inhibitors of carbonic anhydrase IX with promising antitumor features toward the human colorectal cancer | 2023 | Eldehna, Wagdy M.; Mohammed, Eslam E.; Al-Ansary, Ghada H.; Berrino, Emanuela; Elbadawi, Mostafa M.; Ibrahim, Tamer M.; Jaballah, Maiy Y.; Al-Rashood, Sara T.; Binjubair, Faizah A.; Celik, Meltem; Nocentini, Alessio; Elbarbry, Fawzy A.; Sahin, Fikrettin; Abdel-Aziz, Hatem A.; Supuran, Claudiu T.; Fares, Mohamed | |
| Escinosome thermosensitive gel optimizes efficacy of CAI-CORM in a rat model of rheumatoid arthritis | 2023 | Vanti, Giulia; Micheli, Laura; Berrino, Emanuela; Mannelli, Lorenzo Di Cesare; Bogani, Irene; Carta, Fabrizio; Bergonzi, Maria Camilla; Supuran, Claudiu T; Ghelardini, Carla; Bilia, Anna Rita | |
| A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran |
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