CERUSO, MARIANGELA
CERUSO, MARIANGELA
Chimica 'Ugo Schiff' - DICUS
4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies
2016 Cornelio, Benedetta; Laronze Cochard, Marie; Ceruso, Mariangela; Ferraroni, Marta; Rance, Graham A.; Carta, Fabrizio; Khlobystov, Andrei N.; Fontana, Antonella; Supuran, CLAUDIU TRANDAFIR; Sapi, Janos
4-Functionalized 1,3-diarylpyrazoles bearing 6-aminosulfonylbenzothiazole moiety as potent inhibitors of carbonic anhydrase isoforms hCA I, II, IX and XII
2014 Sitaram, Null; Ceruso, Mariangela; Khloya, Poonam; Supuran, Claudiu T.; Sharma, Pawan K.
5-Arylisothiazol-3(2H)-one-1,(1)-(di)oxides: A new class of selective tumor-associated carbonic anhydrases (hCA IX and XII) inhibitors
2019 Cornelio, Benedetta; Laronze-Cochard, Marie; Miambo, Raimundo; De Grandis, Michela; Riccioni, Rossana; Borisova, Boryana; Dontchev, Dimitar; Machado, Carine; Ceruso, Mariangela; Fontana, Antonella; Supuran, Claudiu T; Sapi, Janos
7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII
2016 Nocentini, Alessio; Ceruso, Mariangela; Carta, Fabrizio; Supuran, Claudiu T.
A new class of quinazoline-sulfonamides acting as efficient inhibitors against the α-carbonic anhydrase from Trypanosoma cruzi
2015 Alafeefy AM; Ceruso M; Al-Jaber NA; Parkkila S; Vermelho AB; Supuran CT
A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
2016 Carradori, Simone; Secci, Daniela; De Monte, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P.; Codispoti, Rossella; De Cosmi, Federica; Guglielmi, Paolo; Supuran, Claudiu T.
Amido/ureidosubstituted benzenesulfonamides-isatin conjugates as low nanomolar/subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform XII
2016 Eldehna, Wagdy M; Fares, Mohamed; Ceruso, Mariangela; Ghabbour, Hazem A.; Abou-Seri, Sahar M.; Abdel-Aziz, Hatem A.; Abou El Ella, Dalal A.; Supuran, Claudiu T.
Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide derivatives bearing a sulfonamide moiety show single-digit nanomolar-to-subnanomolar inhibition constants against the tumor-associated human carbonic anhydrases IX and XII
2020 Hargunani P.; Tadge N.; Ceruso M.; Leitans J.; Kazaks A.; Tars K.; Gratteri P.; Supuran C.T.; Nocentini A.; Toraskar M.P.
Arylamino bisphosphonates: Potent and selective inhibitors of the tumor-associated carbonic anhydrase XII
2014 Tauro, Marilena; Loiodice, Fulvio; Ceruso, Mariangela; Supuran, Claudiu T.; Tortorella, Paolo
Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations
2016 Nocentini, Alessio; Ferraroni, Marta; Carta, Fabrizio; Ceruso, Mariangela; Gratteri, Paola; Lanzi, Cecilia; Masini, Emanuela; Supuran, Claudiu T
Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms
2015 Buemi, Maria Rosa; De Luca, Laura; Ferro, Stefania; Bruno, Elvira; Ceruso, Mariangela; Supuran, Claudiu T.; Pospíšilová, Klára; Brynda, Jiří; Řezáčová, Pavlína; Gitto, Rosaria
Carbonic anhydrase inhibitors: Design, synthesis, and biological evaluation of novel sulfonyl semicarbazide derivatives
2014 Pichake, Jayashree; Kharkar, Prashant S.; Ceruso, Mariangela; Supuran, Claudiu T; Toraskar, Mrunmayee P.
Carbonic anhydrase inhibitors: Synthesis, molecular docking, cytotoxic and inhibition of the human carbonic anhydrase isoforms I, II, IX, XII with novel benzenesulfonamides incorporating pyrrole, pyrrolopyrimidine and fused pyrrolopyrimidine moieties
2014 Ghorab, Mostafa M.; Alsaid, Mansour S.; Ceruso, Mariangela; Nissan, Yassin M.; Supuran, Claudiu T.
Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds
2014 Abdel-Aziz, Alaa A.-M.; El-Azab, Adel S.; Ceruso, Mariangela; Supuran, Claudiu T.
Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII
2015 Nocentini, Alessio; Carta, Fabrizio; Ceruso, Mariangela; Bartolucci, Gianluca; Supuran, Claudiu T.
Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
2014 De Monte, Celeste; Carradori, Simone; Secci, Daniela; D'Ascenzio, Melissa; Vullo, Daniela; Ceruso, Mariangela; Supuran, Claudiu T.
Design and synthesis of benzothiazole-6-sulfonamides acting as highly potent inhibitors of carbonic anhydrase isoforms I, II, IX and XII
2015 Ibrahim, Diaa A.; Lasheen, Deena S.; Zaky, Maysoun Y.; Ibrahim, Amany W.; Vullo, Daniela; Ceruso, Mariangela; Supuran, Claudiu T.; Abou El Ella, Dalal A.
Design and validation of FRESH, a drug discovery paradigm resting on robust chemical synthesis
2015 Shi, Qi; Kaiser, Thomas M.; Dentmon, Zackery W.; Ceruso, Mariangela; Vullo, Daniela; Supuran, Claudiu T.; Snyder, James P.
Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII
2014 D'Ascenzio, Melissa; Carradori, Simone; De Monte, Celeste; Secci, Daniela; Ceruso, Mariangela; Supuran, Claudiu T.
Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma
2016 Alafeefy, Ahmed M; Carta, Fabrizio; Ceruso, Mariangela; Al-Tamimi, Abdul-Malek S; Al-Kahtani, Abdulla A; Supuran, Claudiu T