DE SANTIS, ALESSIA
DE SANTIS, ALESSIA
Chimica 'Ugo Schiff' - DICUS
A Structural Investigation of the Interaction between a GC-376-Based Peptidomimetic PROTAC and Its Precursor with the Viral Main Protease of Coxsackievirus B3
2024 De Santis, Alessia; Grifagni, Deborah; Orsetti, Andrea; Lenci, Elena; Rosato, Antonio; D'Onofrio, Mariapina; Trabocchi, Andrea; Ciofi-Baffoni, Simone; Cantini, Francesca; Calderone, Vito
An antiviral agent triggering the proteolysis of the main protease from Coxsackievirus B3
2023 Alessia De Santis, Andrea Orsetti , Deborah Grifagni , Elena Lenci , Francesca Lucarelli , Francesca Cantini , Vito Calderone , Andrea Trabocchi , Mariapina D’Onofrio, Simone Ciofi-Baffoni
Application of the PROTAC-based approach to trigger proteolysis of the Coxsackievirus B3 main protease
2025 Alessia De Santis, Deborah Grifagni, Andrea Orsetti, Chiara La Guidara, Niccolò Moradei, Koi L. Merz, Elena Lenci, Antonio Rosato, Mariapina D’Onofrio, Andrea Trabocchi, Simone Ciofi-Baffoni, Francesca Cantini, Vito Calderone
Congresso Nazionale della Divisione di Chimica dei Sistemi Biologici
2025 Chiara La Guidara, Alessia De Santis, Niccolò Moradei, Deborah Grifagni, Francesca Cantini, Mariapina D'Onofrio, Alfonso Carotenuto, Simone Ciofi-Baffoni, Antonio Rosato
Development of a GC-376 Based Peptidomimetic PROTAC as a Degrader of 3-Chymotrypsin-like Protease of SARS-CoV-2
2024 Grifagni, Deborah; Lenci, Elena; De Santis, Alessia; Orsetti, Andrea; Barracchia, Carlo Giorgio; Tedesco, Filomena; Bellini Puglielli, Raffaele; Lucarelli, Francesca; Lauriola, Angela; Assfalg, Michael; Cantini, Francesca; Calderone, Vito; Guardavaccaro, Daniele; Trabocchi, Andrea; D’Onofrio, Mariapina; Ciofi-Baffoni, Simone
Exploration of PROTAC technology for the development of broad-spectrum antiviral drugs to trigger the proteolysis of the main viral protease
2025 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, MariapinaD’Onofrio, Simone Ciofi-Baffoni
From Inhibition to Protein-Targeted Degradation: Structural Insights into SARS-CoV-2 and CVB3 Proteins for Antiviral Drug Development
2025 Alessia De Santis
Gold-Based Metal Drugs as Inhibitors of Coronavirus Proteins: The Inhibition of SARS-CoV-2 Main Protease by Auranofin and Its Analogs
2022 Massai, Lara; Grifagni, Deborah; De Santis, Alessia; Geri, Andrea; Cantini, Francesca; Calderone, Vito; Banci, Lucia; Messori, Luigi
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis , Deborah Grifagni , Elena Lenci , Andrea Orsetti , Carlo Giorgio Barracchia , Filomena Tedesco , Raffaele Bellini Puglielli , Francesca Lucarelli , Chiara La Guidara , Angela Lauriola , Michael Assfalg , Francesca Cantini , Vito Calderone , Daniele Guardavaccaro , Andrea Trabocchi, Antonio Rosato, Mariapina D'Onofrio , Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco,Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2023 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A Structural Investigation of the Interaction between a GC-376-Based Peptidomimetic PROTAC and Its Precursor with the Viral Main Protease of Coxsackievirus B3 | 2024 | De Santis, Alessia; Grifagni, Deborah; Orsetti, Andrea; Lenci, Elena; Rosato, Antonio; D'Onofrio, Mariapina; Trabocchi, Andrea; Ciofi-Baffoni, Simone; Cantini, Francesca; Calderone, Vito | |
| An antiviral agent triggering the proteolysis of the main protease from Coxsackievirus B3 | 2023 | Alessia De Santis, Andrea Orsetti , Deborah Grifagni , Elena Lenci , Francesca Lucarelli , Francesca Cantini , Vito Calderone , Andrea Trabocchi , Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| Application of the PROTAC-based approach to trigger proteolysis of the Coxsackievirus B3 main protease | 2025 | Alessia De Santis, Deborah Grifagni, Andrea Orsetti, Chiara La Guidara, Niccolò Moradei, Koi L. Merz, Elena Lenci, Antonio Rosato, Mariapina D’Onofrio, Andrea Trabocchi, Simone Ciofi-Baffoni, Francesca Cantini, Vito Calderone | |
| Congresso Nazionale della Divisione di Chimica dei Sistemi Biologici | 2025 | Chiara La Guidara, Alessia De Santis, Niccolò Moradei, Deborah Grifagni, Francesca Cantini, Mariapina D'Onofrio, Alfonso Carotenuto, Simone Ciofi-Baffoni, Antonio Rosato | |
| Development of a GC-376 Based Peptidomimetic PROTAC as a Degrader of 3-Chymotrypsin-like Protease of SARS-CoV-2 | 2024 | Grifagni, Deborah; Lenci, Elena; De Santis, Alessia; Orsetti, Andrea; Barracchia, Carlo Giorgio; Tedesco, Filomena; Bellini Puglielli, Raffaele; Lucarelli, Francesca; Lauriola, Angela; Assfalg, Michael; Cantini, Francesca; Calderone, Vito; Guardavaccaro, Daniele; Trabocchi, Andrea; D’Onofrio, Mariapina; Ciofi-Baffoni, Simone | |
| Exploration of PROTAC technology for the development of broad-spectrum antiviral drugs to trigger the proteolysis of the main viral protease | 2025 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, MariapinaD’Onofrio, Simone Ciofi-Baffoni | |
| From Inhibition to Protein-Targeted Degradation: Structural Insights into SARS-CoV-2 and CVB3 Proteins for Antiviral Drug Development | 2025 | Alessia De Santis | |
| Gold-Based Metal Drugs as Inhibitors of Coronavirus Proteins: The Inhibition of SARS-CoV-2 Main Protease by Auranofin and Its Analogs | 2022 | Massai, Lara; Grifagni, Deborah; De Santis, Alessia; Geri, Andrea; Cantini, Francesca; Calderone, Vito; Banci, Lucia; Messori, Luigi | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis , Deborah Grifagni , Elena Lenci , Andrea Orsetti , Carlo Giorgio Barracchia , Filomena Tedesco , Raffaele Bellini Puglielli , Francesca Lucarelli , Chiara La Guidara , Angela Lauriola , Michael Assfalg , Francesca Cantini , Vito Calderone , Daniele Guardavaccaro , Andrea Trabocchi, Antonio Rosato, Mariapina D'Onofrio , Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco,Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2023 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni |