PAOLETTI, NICCOLÒ
PAOLETTI, NICCOLÒ
Computational approaches in drug discovery: strategies to address polypharmacology and the synthesis/optimization of lead compounds
2025 Niccolò Paoletti, Paola Gratteri, Claudiu T. Supuran, Alessandro Bonardi,
Design and synthesis of isoxazole-functionalized benzene sulphonamides as novel inhibitors of Mycobacterium tuberculosis β-carbonic anhydrases
2025 Bandela, Rani; Singampalli, Anuradha; Maddipatla, Sarvan; Kumar, Pardeep; Bellapukonda, Sri Mounika; Ramavath, Rajendhar; Mahajan, Lina S.; Nanduri, Srinivas; Vemula, Divya; Dalal, Aman; kalia, Nitin Pal; Bhandari, Vasundhra; Gratteri, Paola; Paoletti, Niccolò; Bonardi, Alessandro; Supuran, Claudiu T.; Yaddanapudi, Venkata Madhavi
Discovery of Novel Hydroxyimine-Tethered Benzenesulfonamides as Potential Human Carbonic Anhydrase IX/XII Inhibitors
2023 Peerzada, Mudasir Nabi; Vullo, Daniela; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Supuran, Claudiu T; Azam, Amir
Exploration of 3-aryl pyrazole-tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors
2023 Ommi, Ojaswitha; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Bhalerao, Harshada Anil; Sau, Shashikanta; Nanduri, Srinivas; Mohammed, Arifuddin; Kalia, Nitin Pal; Sonti, Rajesh; Supuran, Claudiu T; Yaddanapudi, Venkata Madhavi
Exploration of New Pyrazole–Hydrazone–Benzenesulfonamide Conjugates as Potent Mycobacterial Carbonic Anhydrase Inhibitors: Design, Synthesis, and Biological Evaluation
2025 Kumar, Pardeep; Singampalli, Anuradha; Bandela, Rani; Bellapukonda, Sri Mounika; Korra, Laxma Naik; Kodi, Ramakrishna; Ghosh, Subhendu; Dalal, Aman; Agnivesh, Puja Kumari; Devi, Ankita; Nanduri, Srinivas; Kalia, Nitin Pal; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Supuran, Claudiu T.; Yaddanapudi, Venkata Madhavi
Exploring aliphatic sulfonamides as multiclass inhibitors of the carbonic anhydrases from the pathogen bacterium Vibrio cholerae
2025 Paoletti, Niccolò; Giovannuzzi, Simone; Bonardi, Alessandro; De Luca, Viviana; Capasso, Clemente; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T.
Novel 3-Sulfonamide Dual-Tail Pyrrol-2-one Bridged Molecules as Potent Human Carbonic Anhydrase Isoform Inhibitors: Design, Synthesis, Molecular Modeling Investigation, and Anticancer Activity in MeWo, SK-BR-3, and MG-63 Cell Lines
2025 Al-Matarneh, Cristina M.; Simionescu, Natalia; Nicolescu, Alina; Silion, Mihaela; Angeli, Andrea; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Pinteala, Mariana; Supuran, Claudiu T.
Production, crystallographic studies, and functional profiling of γ-carbonic anhydrase from the probiotic Limosilactobacillus reuteri: In vitro and cell-based insights
2026 Bonardi, Alessandro; Carradori, Simone; Paoletti, Niccolò; Angeli, Andrea; Ferraroni, Marta; Iacovozzi, Damiano; Gallorini, Marialucia; D'Agostino, Ilaria; De Luca, Viviana; Gratteri, Paola; Cataldi, Amelia; Supuran, Claudiu T.; Capasso, Clemente
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Computational approaches in drug discovery: strategies to address polypharmacology and the synthesis/optimization of lead compounds | 2025 | Niccolò Paoletti, Paola Gratteri, Claudiu T. Supuran, Alessandro Bonardi, | |
| Design and synthesis of isoxazole-functionalized benzene sulphonamides as novel inhibitors of Mycobacterium tuberculosis β-carbonic anhydrases | 2025 | Bandela, Rani; Singampalli, Anuradha; Maddipatla, Sarvan; Kumar, Pardeep; Bellapukonda, Sri Mounika; Ramavath, Rajendhar; Mahajan, Lina S.; Nanduri, Srinivas; Vemula, Divya; Dalal, Aman; kalia, Nitin Pal; Bhandari, Vasundhra; Gratteri, Paola; Paoletti, Niccolò; Bonardi, Alessandro; Supuran, Claudiu T.; Yaddanapudi, Venkata Madhavi | |
| Discovery of Novel Hydroxyimine-Tethered Benzenesulfonamides as Potential Human Carbonic Anhydrase IX/XII Inhibitors | 2023 | Peerzada, Mudasir Nabi; Vullo, Daniela; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Supuran, Claudiu T; Azam, Amir | |
| Exploration of 3-aryl pyrazole-tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors | 2023 | Ommi, Ojaswitha; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Bhalerao, Harshada Anil; Sau, Shashikanta; Nanduri, Srinivas; Mohammed, Arifuddin; Kalia, Nitin Pal; Sonti, Rajesh; Supuran, Claudiu T; Yaddanapudi, Venkata Madhavi | |
| Exploration of New Pyrazole–Hydrazone–Benzenesulfonamide Conjugates as Potent Mycobacterial Carbonic Anhydrase Inhibitors: Design, Synthesis, and Biological Evaluation | 2025 | Kumar, Pardeep; Singampalli, Anuradha; Bandela, Rani; Bellapukonda, Sri Mounika; Korra, Laxma Naik; Kodi, Ramakrishna; Ghosh, Subhendu; Dalal, Aman; Agnivesh, Puja Kumari; Devi, Ankita; Nanduri, Srinivas; Kalia, Nitin Pal; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Supuran, Claudiu T.; Yaddanapudi, Venkata Madhavi | |
| Exploring aliphatic sulfonamides as multiclass inhibitors of the carbonic anhydrases from the pathogen bacterium Vibrio cholerae | 2025 | Paoletti, Niccolò; Giovannuzzi, Simone; Bonardi, Alessandro; De Luca, Viviana; Capasso, Clemente; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T. | |
| Novel 3-Sulfonamide Dual-Tail Pyrrol-2-one Bridged Molecules as Potent Human Carbonic Anhydrase Isoform Inhibitors: Design, Synthesis, Molecular Modeling Investigation, and Anticancer Activity in MeWo, SK-BR-3, and MG-63 Cell Lines | 2025 | Al-Matarneh, Cristina M.; Simionescu, Natalia; Nicolescu, Alina; Silion, Mihaela; Angeli, Andrea; Paoletti, Niccolò; Bonardi, Alessandro; Gratteri, Paola; Pinteala, Mariana; Supuran, Claudiu T. | |
| Production, crystallographic studies, and functional profiling of γ-carbonic anhydrase from the probiotic Limosilactobacillus reuteri: In vitro and cell-based insights | 2026 | Bonardi, Alessandro; Carradori, Simone; Paoletti, Niccolò; Angeli, Andrea; Ferraroni, Marta; Iacovozzi, Damiano; Gallorini, Marialucia; D'Agostino, Ilaria; De Luca, Viviana; Gratteri, Paola; Cataldi, Amelia; Supuran, Claudiu T.; Capasso, Clemente |