LUCARINI, ELENA
LUCARINI, ELENA
Neuroscienze, Area del Farmaco e Salute del Bambino (NEUROFARBA)
(E)-3-Furan-2-yl- N- p-tolyl-acrylamide and its Derivative DM489 Decrease Neuropathic Pain in Mice Predominantly by α7 Nicotinic Acetylcholine Receptor Potentiation
2020 Arias H.R.; Ghelardini C.; Lucarini E.; Tae H.-S.; Yousuf A.; Marcovich I.; Manetti D.; Romanelli M.N.; Elgoyhen A.B.; Adams D.J.; Di Cesare Mannelli L.
Acute visceral pain relief mediated by A(3)AR agonists in rats: involvement of N-type voltage-gated calcium channels
2020 Lucarini, E; Coppi, E; Micheli, L; Parisio, C; Vona, A; Cherchi, F; Pugliese, AM; Pedata, F; Failli, P; Palomino, S; Wahl, J; Largent-Milnes, TM; Vanderah, TW; Tosh, DK; Jacobson, KA; Salvemini, D; Ghelardini, C; Mannelli, LD
Adenosine A3 receptor activation inhibits pro-nociceptive N-type Ca2+ currents and cell excitability in dorsal root ganglion neurons
2019 Coppi, Elisabetta; Cherchi, Federica; Fusco, Irene; Failli, Paola; Vona, Alessia; Dettori, Ilaria; Gaviano, Lisa; Lucarini, Elena; Jacobson, Kenneth A; Tosh, Dilip K; Salvemini, Daniela; Ghelardini, Carla; Pedata, Felicita; Di Cesare Mannelli, Lorenzo; Pugliese, Anna Maria
Anti-inflammatory Effects of Novel P2X4 Receptor Antagonists, NC-2600 and NP-1815-PX, in a Murine Model of Colitis
2022 D'Antongiovanni, Vanessa; Pellegrini, Carolina; Benvenuti, Laura; Fornai, Matteo; Di Salvo, Clelia; Natale, Gianfranco; Ryskalin, Larisa; Bertani, Lorenzo; Lucarini, Elena; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Nemeth, Zoltan H; Haskó, György; Antonioli, Luca
Antioxidant-Conjugated 1,2,4-Triazolo[4,3-a]pyrazin-3-one Derivatives: Highly Potent and Selective Human A2A Adenosine Receptor Antagonists Possessing Protective Efficacy in Neuropathic Pain
2019 Falsini M.; Catarzi D.; Varano F.; Ceni C.; Dal Ben D.; Marucci G.; Buccioni M.; Volpini R.; Di Cesare Mannelli L.; Lucarini E.; Ghelardini C.; Bartolucci G.; Menicatti M.; Colotta V.
Beneficial Effect of H2S-Releasing Molecules in an In Vitro Model of Sarcopenia: Relevance of Glucoraphanin
2022 Micheli, Laura; Mitidieri, Emma; Turnaturi, Carlotta; Vanacore, Domenico; Ciampi, Clara; Lucarini, Elena; Cirino, Giuseppe; Ghelardini, Carla; Sorrentino, Raffaella; Di Cesare Mannelli, Lorenzo; d'Emmanuele di Villa Bianca, Roberta
Beneficial Effects of Eruca sativa Defatted Seed Meal on Visceral Pain and Intestinal Damage Resulting from Colitis in Rats
2022 Lucarini E.; Micheli L.; Pagnotta E.; Matteo R.; Parisio C.; Toti A.; Ferrara V.; Ciampi C.; Martelli A.; Testai L.; Calderone V.; Savino M.; Russo M.; Pecchioni N.; Ghelardini C.; Di Cesare Mannelli L.
Bioisosteric Development of Multitarget Nonsteroidal Anti-Inflammatory Drug-Carbonic Anhydrases Inhibitor Hybrids for the Management of Rheumatoid Arthritis
2020 Bua S.; Lucarini L.; Micheli L.; Menicatti M.; Bartolucci G.; Selleri S.; Di Cesare Mannelli L.; Ghelardini C.; Masini E.; Carta F.; Gratteri P.; Nocentini A.; Supuran C.T.
Carbonic Anhydrase IV Selective Inhibitors Counteract the Development of Colitis-Associated Visceral Pain in Rats
2021 Lucarini E., Nocentini A., Bonardi A., Chiaramonte N., Parisio C., Micheli L., Toti A., Ferrara V., Carrino D., Pacini A., Romanelli M.N., Supuran C.T., Ghelardini C., Di Cesare Mannelli L.
Chalcogenides-incorporating carbonic anhydrase inhibitors concomitantly reverted oxaliplatin-induced neuropathy and enhanced antiproliferative action
2021 Tanini D.; Carradori S.; Capperucci A.; Lupori L.; Zara S.; Ferraroni M.; Ghelardini C.; Mannelli L.D.C.; Micheli L.; Lucarini E.; Carta F.; Angeli A.; Supuran C.T.
Deepening the Mechanisms of Visceral Pain Persistence: An Evaluation of the Gut-Spinal Cord Relationship
2020 Lucarini E.; Parisio C.; Branca J.J.V.; Segnani C.; Ippolito C.; Pellegrini C.; Antonioli L.; Fornai M.; Micheli L.; Pacini A.; Bernardini N.; Blandizzi C.; Ghelardini C.; Di Cesare Mannelli L.
Design and Synthesis of Novel Thiazolo[5,4-d]pyrimidine Derivatives with High Affinity for Both the Adenosine A1 and A2A Receptors, and Efficacy in Animal Models of Depression
2021 Varano, Flavia; Catarzi, Daniela; Vigiani, Erica; Dal Ben, Diego; Buccioni, Michela; Marucci, Gabriella; Di Cesare Mannelli, Lorenzo; Lucarini, Elena; Ghelardini, Carla; Volpini, Rosaria; Colotta, Vittoria
Design and synthesis of the first indole-based blockers of Panx-1 channel
2021 Crocetti, Letizia; Guerrini, Gabriella; Puglioli, Sara; Giovannoni, Maria Paola; Di Cesare Mannelli, Lorenzo; Lucarini, Elena; Ghelardini, Carla; Wang, Junjie; Dahl, Gerhard
Design, synthesis and X-ray crystallography of selenides bearing benzenesulfonamide moiety with neuropathic pain modulating effects.
2018 Angeli A, di Cesare Mannelli L, Lucarini E, Peat TS, Ghelardini C, Supuran CT
Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: From Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands
2022 Gado F.; Ferrisi R.; Polini B.; Mohamed K.A.; Ricardi C.; Lucarini E.; Carpi S.; Domenichini F.; Stevenson L.A.; Rapposelli S.; Saccomanni G.; Nieri P.; Ortore G.; Pertwee R.G.; Ghelardini C.; Di Cesare Mannelli L.; Chiellini G.; Laprairie R.B.; Manera C.
Effect of glucoraphanin and sulforaphane against chemotherapy-induced neuropathic pain: Kv7 potassium channels modulation by H2 S release in vivo.
2018 Lucarini E, Micheli L, Trallori E, Citi V, Martelli A, Testai L, De Nicola G, Iori R, Calderone V, Ghelardini C, Di Cesare Mannelli L
Effect of NIR laser therapy by MLS-MiS source against neuropathic pain in rats: in vivo and ex vivo analysis.
2019 Micheli L, Cialdai F, Pacini A, Branca JJV, Morbidelli L, Ciccone V, Lucarini E, Ghelardini C, Monici M, Di Cesare Mannelli L
Effects of natural and synthetic isothiocyanate-based H2S-releasers against chemotherapy-induced neuropathic pain: Role of Kv7 potassium channels
2017 Di Cesare Mannelli, L; Lucarini, E; Micheli, L; Mosca, I; Ambrosino, P; Soldovieri, Mv; Martelli, A; Testai, L; Taglialatela, M; Calderone, V; Ghelardini, C.
Effects of the combination of β-hydroxy-β-methyl butyrate and R(+) lipoic acid in a cellular model of sarcopenia
2020 Di Cesare Mannelli L.; Micheli L.; Lucarini E.; Parisio C.; Toti A.; Tenci B.; Zanardelli M.; Branca J.J.V.; Pacini A.; Ghelardini C.
Effects of Ultramicronized N-Palmitoylethanolamine Supplementation on Tramadol and Oxycodone Analgesia and Tolerance Prevention
2022 Micheli L.; Lucarini E.; Toti A.; Ferrara V.; Ciampi C.; Parisio C.; Bartolucci G.; Di Cesare Mannelli L.; Ghelardini C.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
(E)-3-Furan-2-yl- N- p-tolyl-acrylamide and its Derivative DM489 Decrease Neuropathic Pain in Mice Predominantly by α7 Nicotinic Acetylcholine Receptor Potentiation | 2020 | Arias H.R.; Ghelardini C.; Lucarini E.; Tae H.-S.; Yousuf A.; Marcovich I.; Manetti D.; Romanelli M.N.; Elgoyhen A.B.; Adams D.J.; Di Cesare Mannelli L. | |
Acute visceral pain relief mediated by A(3)AR agonists in rats: involvement of N-type voltage-gated calcium channels | 2020 | Lucarini, E; Coppi, E; Micheli, L; Parisio, C; Vona, A; Cherchi, F; Pugliese, AM; Pedata, F; Failli, P; Palomino, S; Wahl, J; Largent-Milnes, TM; Vanderah, TW; Tosh, DK; Jacobson, KA; Salvemini, D; Ghelardini, C; Mannelli, LD | |
Adenosine A3 receptor activation inhibits pro-nociceptive N-type Ca2+ currents and cell excitability in dorsal root ganglion neurons | 2019 | Coppi, Elisabetta; Cherchi, Federica; Fusco, Irene; Failli, Paola; Vona, Alessia; Dettori, Ilaria; Gaviano, Lisa; Lucarini, Elena; Jacobson, Kenneth A; Tosh, Dilip K; Salvemini, Daniela; Ghelardini, Carla; Pedata, Felicita; Di Cesare Mannelli, Lorenzo; Pugliese, Anna Maria | |
Anti-inflammatory Effects of Novel P2X4 Receptor Antagonists, NC-2600 and NP-1815-PX, in a Murine Model of Colitis | 2022 | D'Antongiovanni, Vanessa; Pellegrini, Carolina; Benvenuti, Laura; Fornai, Matteo; Di Salvo, Clelia; Natale, Gianfranco; Ryskalin, Larisa; Bertani, Lorenzo; Lucarini, Elena; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Nemeth, Zoltan H; Haskó, György; Antonioli, Luca | |
Antioxidant-Conjugated 1,2,4-Triazolo[4,3-a]pyrazin-3-one Derivatives: Highly Potent and Selective Human A2A Adenosine Receptor Antagonists Possessing Protective Efficacy in Neuropathic Pain | 2019 | Falsini M.; Catarzi D.; Varano F.; Ceni C.; Dal Ben D.; Marucci G.; Buccioni M.; Volpini R.; Di Cesare Mannelli L.; Lucarini E.; Ghelardini C.; Bartolucci G.; Menicatti M.; Colotta V. | |
Beneficial Effect of H2S-Releasing Molecules in an In Vitro Model of Sarcopenia: Relevance of Glucoraphanin | 2022 | Micheli, Laura; Mitidieri, Emma; Turnaturi, Carlotta; Vanacore, Domenico; Ciampi, Clara; Lucarini, Elena; Cirino, Giuseppe; Ghelardini, Carla; Sorrentino, Raffaella; Di Cesare Mannelli, Lorenzo; d'Emmanuele di Villa Bianca, Roberta | |
Beneficial Effects of Eruca sativa Defatted Seed Meal on Visceral Pain and Intestinal Damage Resulting from Colitis in Rats | 2022 | Lucarini E.; Micheli L.; Pagnotta E.; Matteo R.; Parisio C.; Toti A.; Ferrara V.; Ciampi C.; Martelli A.; Testai L.; Calderone V.; Savino M.; Russo M.; Pecchioni N.; Ghelardini C.; Di Cesare Mannelli L. | |
Bioisosteric Development of Multitarget Nonsteroidal Anti-Inflammatory Drug-Carbonic Anhydrases Inhibitor Hybrids for the Management of Rheumatoid Arthritis | 2020 | Bua S.; Lucarini L.; Micheli L.; Menicatti M.; Bartolucci G.; Selleri S.; Di Cesare Mannelli L.; Ghelardini C.; Masini E.; Carta F.; Gratteri P.; Nocentini A.; Supuran C.T. | |
Carbonic Anhydrase IV Selective Inhibitors Counteract the Development of Colitis-Associated Visceral Pain in Rats | 2021 | Lucarini E., Nocentini A., Bonardi A., Chiaramonte N., Parisio C., Micheli L., Toti A., Ferrara V., Carrino D., Pacini A., Romanelli M.N., Supuran C.T., Ghelardini C., Di Cesare Mannelli L. | |
Chalcogenides-incorporating carbonic anhydrase inhibitors concomitantly reverted oxaliplatin-induced neuropathy and enhanced antiproliferative action | 2021 | Tanini D.; Carradori S.; Capperucci A.; Lupori L.; Zara S.; Ferraroni M.; Ghelardini C.; Mannelli L.D.C.; Micheli L.; Lucarini E.; Carta F.; Angeli A.; Supuran C.T. | |
Deepening the Mechanisms of Visceral Pain Persistence: An Evaluation of the Gut-Spinal Cord Relationship | 2020 | Lucarini E.; Parisio C.; Branca J.J.V.; Segnani C.; Ippolito C.; Pellegrini C.; Antonioli L.; Fornai M.; Micheli L.; Pacini A.; Bernardini N.; Blandizzi C.; Ghelardini C.; Di Cesare Mannelli L. | |
Design and Synthesis of Novel Thiazolo[5,4-d]pyrimidine Derivatives with High Affinity for Both the Adenosine A1 and A2A Receptors, and Efficacy in Animal Models of Depression | 2021 | Varano, Flavia; Catarzi, Daniela; Vigiani, Erica; Dal Ben, Diego; Buccioni, Michela; Marucci, Gabriella; Di Cesare Mannelli, Lorenzo; Lucarini, Elena; Ghelardini, Carla; Volpini, Rosaria; Colotta, Vittoria | |
Design and synthesis of the first indole-based blockers of Panx-1 channel | 2021 | Crocetti, Letizia; Guerrini, Gabriella; Puglioli, Sara; Giovannoni, Maria Paola; Di Cesare Mannelli, Lorenzo; Lucarini, Elena; Ghelardini, Carla; Wang, Junjie; Dahl, Gerhard | |
Design, synthesis and X-ray crystallography of selenides bearing benzenesulfonamide moiety with neuropathic pain modulating effects. | 2018 | Angeli A, di Cesare Mannelli L, Lucarini E, Peat TS, Ghelardini C, Supuran CT | |
Design, Synthesis, and Biological Activity of New CB2 Receptor Ligands: From Orthosteric and Allosteric Modulators to Dualsteric/Bitopic Ligands | 2022 | Gado F.; Ferrisi R.; Polini B.; Mohamed K.A.; Ricardi C.; Lucarini E.; Carpi S.; Domenichini F.; Stevenson L.A.; Rapposelli S.; Saccomanni G.; Nieri P.; Ortore G.; Pertwee R.G.; Ghelardini C.; Di Cesare Mannelli L.; Chiellini G.; Laprairie R.B.; Manera C. | |
Effect of glucoraphanin and sulforaphane against chemotherapy-induced neuropathic pain: Kv7 potassium channels modulation by H2 S release in vivo. | 2018 | Lucarini E, Micheli L, Trallori E, Citi V, Martelli A, Testai L, De Nicola G, Iori R, Calderone V, Ghelardini C, Di Cesare Mannelli L | |
Effect of NIR laser therapy by MLS-MiS source against neuropathic pain in rats: in vivo and ex vivo analysis. | 2019 | Micheli L, Cialdai F, Pacini A, Branca JJV, Morbidelli L, Ciccone V, Lucarini E, Ghelardini C, Monici M, Di Cesare Mannelli L | |
Effects of natural and synthetic isothiocyanate-based H2S-releasers against chemotherapy-induced neuropathic pain: Role of Kv7 potassium channels | 2017 | Di Cesare Mannelli, L; Lucarini, E; Micheli, L; Mosca, I; Ambrosino, P; Soldovieri, Mv; Martelli, A; Testai, L; Taglialatela, M; Calderone, V; Ghelardini, C. | |
Effects of the combination of β-hydroxy-β-methyl butyrate and R(+) lipoic acid in a cellular model of sarcopenia | 2020 | Di Cesare Mannelli L.; Micheli L.; Lucarini E.; Parisio C.; Toti A.; Tenci B.; Zanardelli M.; Branca J.J.V.; Pacini A.; Ghelardini C. | |
Effects of Ultramicronized N-Palmitoylethanolamine Supplementation on Tramadol and Oxycodone Analgesia and Tolerance Prevention | 2022 | Micheli L.; Lucarini E.; Toti A.; Ferrara V.; Ciampi C.; Parisio C.; Bartolucci G.; Di Cesare Mannelli L.; Ghelardini C. |