AMMARA, ANDREA
AMMARA, ANDREA
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
A new framework for novel analogues of pazopanib as potent and selective human carbonic anhydrase inhibitors: Design, repurposing rational, synthesis, crystallographic, in vivo and in vitro biological assessments
2024 Hefny S.M.; El-Moselhy T.F.; El-Din N.; Ammara A.; Angeli A.; Ferraroni M.; El-Dessouki A.M.; Shaldam M.A.; Yahya G.; Al-Karmalawy A.A.; Supuran C.T.; Tawfik H.O.
Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors
2023 Elsayed, Zainab M; Almahli, Hadia; Nocentini, Alessio; Ammara, Andrea; Supuran, Claudiu T; Eldehna, Wagdy M; Abou-Seri, Sahar M
Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma
2024 Tawfik, Haytham O.; Saleh, Mohamed M.; Ammara, Andrea; Khaleel, Eman F.; Badi, Rehab; Khater, Yomna T. T.; Rasheed, Rabab A.; Attia, Ahmed A.; Hefny, Salma M.; Elkaeed, Eslam B.; Nocentini, Alessio; Supuran, Claudiu T.; Eldehna, Wagdy M.; Shaldam, Moataz A.
Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases
2024 Nocentini A.; Costa A.; Bonardi A.; Ammara A.; Giovannuzzi S.; Petreni A.; Bartolucci G.; Rani B.; Leri M.; Bucciantini M.; Fernandez-Bolanos J.G.; Lopez O.; Passani M.B.; Provensi G.; Gratteri P.; Supuran C.T.
Repurposing Drug Metabolites into Dual β-Adrenergic Receptor-Carbonic Anhydrase Modulators as Potential Tools for Ocular Disorders
2025 Ammara, Andrea; Carone, Alessandra; Lucarini, Laura; Sgambellone, Silvia; Marri, Silvia; Villano, Serafina; Matucci, Rosanna; Luga, Gerta; Fittipaldi, Chiara; Pecori, Riccardo; Pieraccini, Giuseppe; Di Serio, Claudia; García-Llorca, Andrea; Eysteinsson, Thor; Kalinin, Stanislav; Viita, Julius Aleksi Olavi; Urtti, Arto; Carta, Fabrizio; Selleri, Silvia; Supuran, Claudiu T
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A new framework for novel analogues of pazopanib as potent and selective human carbonic anhydrase inhibitors: Design, repurposing rational, synthesis, crystallographic, in vivo and in vitro biological assessments | 2024 | Hefny S.M.; El-Moselhy T.F.; El-Din N.; Ammara A.; Angeli A.; Ferraroni M.; El-Dessouki A.M.; Shaldam M.A.; Yahya G.; Al-Karmalawy A.A.; Supuran C.T.; Tawfik H.O. | |
| Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors | 2023 | Elsayed, Zainab M; Almahli, Hadia; Nocentini, Alessio; Ammara, Andrea; Supuran, Claudiu T; Eldehna, Wagdy M; Abou-Seri, Sahar M | |
| Discovery of Novel Pyridazine-Tethered Sulfonamides as Carbonic Anhydrase II Inhibitors for the Management of Glaucoma | 2024 | Tawfik, Haytham O.; Saleh, Mohamed M.; Ammara, Andrea; Khaleel, Eman F.; Badi, Rehab; Khater, Yomna T. T.; Rasheed, Rabab A.; Attia, Ahmed A.; Hefny, Salma M.; Elkaeed, Eslam B.; Nocentini, Alessio; Supuran, Claudiu T.; Eldehna, Wagdy M.; Shaldam, Moataz A. | |
| Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases | 2024 | Nocentini A.; Costa A.; Bonardi A.; Ammara A.; Giovannuzzi S.; Petreni A.; Bartolucci G.; Rani B.; Leri M.; Bucciantini M.; Fernandez-Bolanos J.G.; Lopez O.; Passani M.B.; Provensi G.; Gratteri P.; Supuran C.T. | |
| Repurposing Drug Metabolites into Dual β-Adrenergic Receptor-Carbonic Anhydrase Modulators as Potential Tools for Ocular Disorders | 2025 | Ammara, Andrea; Carone, Alessandra; Lucarini, Laura; Sgambellone, Silvia; Marri, Silvia; Villano, Serafina; Matucci, Rosanna; Luga, Gerta; Fittipaldi, Chiara; Pecori, Riccardo; Pieraccini, Giuseppe; Di Serio, Claudia; García-Llorca, Andrea; Eysteinsson, Thor; Kalinin, Stanislav; Viita, Julius Aleksi Olavi; Urtti, Arto; Carta, Fabrizio; Selleri, Silvia; Supuran, Claudiu T |