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Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase
2016 Bozdag, Murat; Carta, Fabrizio; Vullo, Daniela*; Isik, Semra; AlOthman, Zeid; Osman, Sameh M.; Scozzafava, Andrea; Supuran, Claudiu T.
Polyamines and α-carbonic anhydrases
2016 Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio
1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads
2017 Ferraroni, Marta; Lucarini, Laura; Masini, Emanuela; Korsakov, Mikhail; Scozzafava, Andrea; Supuran, Claudiu T.*; Krasavin, Mikhail
Carbonic anhydrase activation enhances object recognition memory in mice through phosphorylation of the extracellular signal-regulated kinase in the cortex and the hippocampus.
2017 Lucas Canto de Souza, Gustavo Provensi, Daniela Vullo, Fabrizio Carta, Andrea Scozzafava, Alessia Costa, Scheila D. Schmidt; Maria Beatrice Passani, Claudiu T. Supuran, Patrizio Blandina
The crystal structures of native hydroquinone 1,2-dioxygenase from Sphingomonas sp. TTNP3 and of substrate and inhibitor complexes
2017 Ferraroni, Marta; Da Vela, Stefano; Kolvenbach, Boris A.; Corvini, Philippe F.X.; Scozzafava, Andrea
Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens
2017 Vullo, Daniela; Kumar, R. Siva Sai; Scozzafava, Andrea; Ferry, James G; Supuran, Claudiu T.
Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis
2017 Bua, Silvia; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Ghelardini, Carla; Bartolucci, Gianluca; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio
Dioxygen, an unexpected carbonic anhydrase ligand
2018 Ferraroni, Marta*; Gaspari, Roberto; Scozzafava, Andrea; Cavalli, Andrea; Supuran, Claudiu T.
Sulfonamide carbonic anhydrase inhibitors: Zinc coordination and tail effects influence inhibitory efficacy and selectivity for different isoforms
2018 Ferraroni, Marta; Cornelio, Benedetta; Sapi, Janos; Supuran, Claudiu T.; Scozzafava, Andrea
Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis
2018 Akgul, Ozlem; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Angeli, Andrea; Ghelardini, Carla; Bartolucci, Gianluca; Altamimi, Abdulmalik Saleh Alfawaz; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase | 2016 | Bozdag, Murat; Carta, Fabrizio; Vullo, Daniela*; Isik, Semra; AlOthman, Zeid; Osman, Sameh M.; Scozzafava, Andrea; Supuran, Claudiu T. | |
Polyamines and α-carbonic anhydrases | 2016 | Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio | |
1,3-Oxazole-based selective picomolar inhibitors of cytosolic human carbonic anhydrase II alleviate ocular hypertension in rabbits: Potency is supported by X-ray crystallography of two leads | 2017 | Ferraroni, Marta; Lucarini, Laura; Masini, Emanuela; Korsakov, Mikhail; Scozzafava, Andrea; Supuran, Claudiu T.*; Krasavin, Mikhail | |
Carbonic anhydrase activation enhances object recognition memory in mice through phosphorylation of the extracellular signal-regulated kinase in the cortex and the hippocampus. | 2017 | Lucas Canto de Souza, Gustavo Provensi, Daniela Vullo, Fabrizio Carta, Andrea Scozzafava, Alessia Costa, Scheila D. Schmidt; Maria Beatrice Passani, Claudiu T. Supuran, Patrizio Blandina | |
The crystal structures of native hydroquinone 1,2-dioxygenase from Sphingomonas sp. TTNP3 and of substrate and inhibitor complexes | 2017 | Ferraroni, Marta; Da Vela, Stefano; Kolvenbach, Boris A.; Corvini, Philippe F.X.; Scozzafava, Andrea | |
Sulphonamide inhibition studies of the β-carbonic anhydrase from the bacterial pathogen Clostridium perfringens | 2017 | Vullo, Daniela; Kumar, R. Siva Sai; Scozzafava, Andrea; Ferry, James G; Supuran, Claudiu T. | |
Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis | 2017 | Bua, Silvia; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Ghelardini, Carla; Bartolucci, Gianluca; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio | |
Dioxygen, an unexpected carbonic anhydrase ligand | 2018 | Ferraroni, Marta*; Gaspari, Roberto; Scozzafava, Andrea; Cavalli, Andrea; Supuran, Claudiu T. | |
Sulfonamide carbonic anhydrase inhibitors: Zinc coordination and tail effects influence inhibitory efficacy and selectivity for different isoforms | 2018 | Ferraroni, Marta; Cornelio, Benedetta; Sapi, Janos; Supuran, Claudiu T.; Scozzafava, Andrea | |
Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis | 2018 | Akgul, Ozlem; Di Cesare Mannelli, Lorenzo; Vullo, Daniela; Angeli, Andrea; Ghelardini, Carla; Bartolucci, Gianluca; Altamimi, Abdulmalik Saleh Alfawaz; Scozzafava, Andrea; Supuran, Claudiu T; Carta, Fabrizio |
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Opzioni
Scopri
Tipologia
- 1 - Contributo su rivista 601
- 1 - Contributo su rivista::1a - Articolo su rivista 601
Data di pubblicazione
- 2010 - 2020 178
- 2000 - 2009 301
- 1990 - 1999 68
- 1980 - 1989 23
- 1972 - 1979 31
Editore
- Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598 3
- American Society for Biochemistry and Molecular Biology:9650 Rockville Pike:Bethesda, MD 20814:(301)530-7145, EMAIL: asbmb@asbmb.faseb.org, INTERNET: http://www.faseb.org/asbmb, Fax: (301)571-1824 2
- Amer Chemical Soc 1
- American Chemical Society:1155 Sixteenth Street Northwest:Washington, DC 20036:(800)227-5558, EMAIL: service@acs.org, INTERNET: http://www.pubs.acs.org, Fax: (614)447-3671 1
- Blackwell Munksgaard:PO Box 2148, Periodicals Department, DK-1016 Copenhagen K Denmark:011 45 33 755913, EMAIL: agentservices@oxon.blackwellpublishing.com, INTERNET: http://www.blackwellmunksgaard.com, Fax: 011 45 77 333377 1
- Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598 Editore precedente:Prof Ugo Croatto Luogo pubbl. Padova Ultimo luogo pubblicazione: Lausanne. 1
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Rivista
- BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 114
- BIOORGANIC & MEDICINAL CHEMISTRY 52
- JOURNAL OF MEDICINAL CHEMISTRY 51
- JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY 47
- BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS 35
- JOURNAL OF ENZYME INHIBITION 33
- INORGANICA CHIMICA ACTA 18
- BIOORGANIC & MEDICINAL CHEMISTRY 17
- INORGANIC CHEMISTRY 16
- METAL-BASED DRUGS 13
Keyword
- Humans 225
- Carbonic Anhydrase Inhibitors 207
- Carbonic Anhydrases 180
- Sulfonamides 148
- Structure-Activity Relationship 140
- Isoenzymes 128
- Animals 102
- Molecular 75
- Molecular Structure 75
- Models 74
Lingua
- eng 254
- ita 1
Accesso al fulltext
- no fulltext 538
- reserved 44
- open 19