Two novel casuarine-6-alpha-D-glucoside analogues, as well as the parent compound, were synthesized and tested as inhibitors towards Chironomus riparius, mammalian pig kidney and Escherichia coli trehalases. Their potent and selective activity is promising for the development of new insecticides.

Casuarine-6-O-alpha-D-glucoside and its analogues are tight binding inhibitors of insect and bacterial trehalases / F. CARDONA; A. GOTI; C. PARMEGGIANI; P. PARENTI; M. FORCELLA; P. FUSI; L. CIPOLLA; S. M. ROBERTS; G. J. DAVIES; T. M. GLOSTER. - In: CHEMICAL COMMUNICATIONS. - ISSN 1359-7345. - STAMPA. - 46:(2010), pp. 2629-2631. [10.1039/b926600c]

Casuarine-6-O-alpha-D-glucoside and its analogues are tight binding inhibitors of insect and bacterial trehalases

CARDONA, FRANCESCA;GOTI, ANDREA;PARMEGGIANI, CAMILLA;
2010

Abstract

Two novel casuarine-6-alpha-D-glucoside analogues, as well as the parent compound, were synthesized and tested as inhibitors towards Chironomus riparius, mammalian pig kidney and Escherichia coli trehalases. Their potent and selective activity is promising for the development of new insecticides.
2010
46
2629
2631
F. CARDONA; A. GOTI; C. PARMEGGIANI; P. PARENTI; M. FORCELLA; P. FUSI; L. CIPOLLA; S. M. ROBERTS; G. J. DAVIES; T. M. GLOSTER
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Utilizza questo identificatore per citare o creare un link a questa risorsa: https://hdl.handle.net/2158/393789
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