Sfoglia per Autore
The functions and structure of ABC transporters: implications for the design of new inhibitors of Pgp and MRP1 to control multidrug resistance (MDR)
2006 E. TEODORI; S. DEI; C. MARTELLI; S. SCAPECCHI; F. GUALTIERI
Highly chiral muscarinic ligands: the discovery of (2S,2'R,3'S,5'R)-1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine 3-sulfoxide methyl iodide, a potent, functionally selective, M2 partial agonist.
2006 Scapecchi, Serena; Matucci, Rosanna; Bellucci, Cristina; Buccioni, M.; Dei, Silvia; Guandalini, Luca; Martelli, Cecilia; Manetti, Dina; Martini, Elisabetta; Marucci, G.; Nesi, Marta; Romanelli, MARIA NOVELLA; Teodori, Elisabetta; Gualtieri, Fulvio
Structure-activity relationships on N,N-dialkylaminoaryl esters, a new class of potent Pgp dependent multidrug resistance (MDR) inhibitors
2007 Silvia Dei; Cecilia Martelli; Elisabetta Teodori; Milena Salerno; Fulvio Gualtieri
synthesis, chiral HPLC separation and pharmacological characterization of muscarinic furan derivatives
2007 Scapecchi, S.; Matucci, R.; Bellucci, C.; Buccioni, M.; Cirilli, R.; Dei, S.; Ferretti, R.; Guandalini, L.; Martelli, C.; Manetti, D.; Martini, E.; Marucci, G.; Nesi, M.; Mnromanelli, M.N.Romanelli; Teodori, E.; Angeli, P.
Isomeric N,N-dicyclohexane-4-ol-amine aryl esters: the discovery of a new class of highly potent and efficacious Pgp-dependent MDR inhibitors
2007 Elisabetta Teodori; Cecilia Martelli; Milena Salerno; Nacira Darghal; Silvia Dei; Fulvio Gualtieri; Dina Manetti; Serena Scapecchi; Maria Novella Romanelli
Isomeric N,N-dicyclohexane-4-ol-amine aryl esters: chemical and pharmacological development of highly potent and efficacious Pgp-dependent MDR inhibitors
2007 Cecilia Martelli; Elisabetta Teodori; Silvia Dei; Marcella Coronnello; Enrico Mini; Giampietro Sgaragli; Daniela Alderighi; Milena Salerno
ISOMERIC N,N-BIS(CYCLOHEXANOL)AMINE ARYL ESTERS: THE DISCOVERY OF A NEW CLASS OF HIGHLY POTENT P-GLYCOPROTEIN (PGP)-DEPENDENT MULTIDRUG RESISTANCE (MDR) INHIBITORS
2007 Teodori, Elisabetta; Martelli, Cecilia; Salerno, M.; Darghal, N.; Dei, Silvia; GARNIER SUILLEROT, A.; Gualtieri, Fulvio; Manetti, Dina; Scapecchi, Serena; Romanelli, MARIA NOVELLA
N,N-bis(alkanol)amine aryl esters and N,N-bis(cyclohexanol)amine aryl esters: Idantification of a new class of Pgp-dependent multidrug resistance (MDR) reverters andowed with potencies in the nanomolar range
2008 Silvia Dei; Cecilia Martelli; Elisabetta Teodori; Dina Manetti; Marcella Coronnello; Milena Salerno; Giampietro Sgaragli; Fulvio Gualtieri
Multidrug resistance (MDR) modulators: Verapamil offsprings and heterocyclic derivatives
2008 E. Teodori; S. Dei; C. Martelli; S. Scapecchi; F. Gualtieri
SAR studies in a series of N,N-bis(arylaLKANOL)AMINE ARYL ESTERS AS p-GLYCOPROTEIN (Pgp) dependent multidrug resistance (MDR) inhibitors
2009 Elisabetta Teodori; Cecilia Martelli; Milena Salerno; Silvia Dei; Fulvio Gualtieri; Dina Manetti; Francesca Orlandi; Serena Scapecchi; Maria Novella Romanelli
Design and synthesis of multidrug resistance (MDR) inhibitors
2009 Cecilia Martelli; Francesca Orlandi; Silvia Dei; Elisabetta Teodori
Design, synthesis and nootropic activity of new analogues of sunifiram and sapunifiram, two potent cognition-enhancers.
2009 Martini, Elisabetta; Salvicchi, A.; Ghelardini, Carla; Manetti, Dina; Dei, Silvia; Guandalini, Luca; Martelli, Cecilia; Melchiorre, Michele; Cellai, Cristina; Scapecchi, Serena; Teodori, Elisabetta; Romanelli, MARIA NOVELLA
N,N-bis(cyclohexanol)amine aryl esters: a new class of highly potent Pgp-dependent multidrug resistance (MDR) inhibitors
2009 Martelli, Cecilia; Alderighi, Daniela; Coronnello, MARCELLA MARIA; Dei, Silvia; Frosini, Maria; Bozec, Benedicte Le; Manetti, Dina; Neri, Annalisa; Romanelli, MARIA NOVELLA; Salerno, Milena; Scapecchi, Serena; Mini, Enrico; Sgaragli, Giampietro; Teodori, Elisabetta
Inhibition of P-glycoprotein-mediated multidrug resistance (MDR) by N,N-bis(cyclohexanol)amine aryl esters: structure-activity relationships
2010 Teodori E.; Martelli C.; Dei S.; Frosini M.; Manetti D.; Neri A.; Orlandi F.; Romanelli M.N.; Scapecchi S.; Salerno M.; Sgaragli G.
N,N-bis(cyclohexanol)amine aryl esters: the discovery of a new class of highly potent inhibitors of transporter-dependent multidrug resistance (MDR)
2010 Teodori, Elisabetta; Dei, Silvia; Martelli, Cecilia; Scapecchi, Serena
Structure-activity relationships studies in a series of N,N-bis(alkanol)amine aryl esters as P-glycoprotein (Pgp) dependent multidrug resistance (MDR) inhibitors
2010 Martelli, Cecilia; Coronnello, MARCELLA MARIA; Dei, Silvia; Manetti, Dina; Orlandi, Francesca; Scapecchi, Serena; Romanelli, MARIA NOVELLA; Salerno, M.; Mini, Enrico; Teodori, Elisabetta
Synthesis, Affinity Profile and Functional Activity of Potent Chiral Muscarinic Antagonists with a Pyrrolidinylfuran Structure
2010 S. Scapecchi; M. Nesi; R. Matucci; C. Bellucci; M. Buccioni; S. Dei; L. Guandalini; D. Manetti; C. Martelli; E. Martini; G. Marucci; F. Orlandi; M. N. Romanelli; E. Teodori; R. Cirilli
The Novel Potent Multidrug Resistance Inhibitors N,N-bis(cyclohexanol)amine Aryl Esters Are Devoid of Vascular Effects
2011 S. Saponara; B. Gorelli; V. Tzankova; C. Martelli; E. Teodori; G. Sgaragli; F. Fusi
Inhibition of P-glycoprotein-mediated Multidrug Resistance (MDR) by N,N-bis(cyclohexanol)amine aryl esters: further restriction of molecular flexibility maintains high potency and efficacy
2011 Martelli, Cecilia; Dei, Silvia; Lambert, C.; Manetti, Dina; Orlandi, Francesca; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Salerno, M.; Teodori, Elisabetta
New structure–activity relationship studies in a series of N,N-bis(cyclohexanol)amine aryl esters as potent reversers of P-glycoprotein-mediated multidrug resistance (MDR)
2013 F. Orlandi; M. Coronnello; C. Bellucci; S. Dei; L. Guandalini; D. Manetti; C. Martelli; M. N. Romanelli; S. Scapecchi; M. Salerno; H. Menif; I. Bello; E. Mini; E. Teodori
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
The functions and structure of ABC transporters: implications for the design of new inhibitors of Pgp and MRP1 to control multidrug resistance (MDR) | 2006 | E. TEODORI; S. DEI; C. MARTELLI; S. SCAPECCHI; F. GUALTIERI | |
Highly chiral muscarinic ligands: the discovery of (2S,2'R,3'S,5'R)-1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine 3-sulfoxide methyl iodide, a potent, functionally selective, M2 partial agonist. | 2006 | Scapecchi, Serena; Matucci, Rosanna; Bellucci, Cristina; Buccioni, M.; Dei, Silvia; Guandalini, Luca; Martelli, Cecilia; Manetti, Dina; Martini, Elisabetta; Marucci, G.; Nesi, Marta; Romanelli, MARIA NOVELLA; Teodori, Elisabetta; Gualtieri, Fulvio | |
Structure-activity relationships on N,N-dialkylaminoaryl esters, a new class of potent Pgp dependent multidrug resistance (MDR) inhibitors | 2007 | Silvia Dei; Cecilia Martelli; Elisabetta Teodori; Milena Salerno; Fulvio Gualtieri | |
synthesis, chiral HPLC separation and pharmacological characterization of muscarinic furan derivatives | 2007 | Scapecchi, S.; Matucci, R.; Bellucci, C.; Buccioni, M.; Cirilli, R.; Dei, S.; Ferretti, R.; Guandalini, L.; Martelli, C.; Manetti, D.; Martini, E.; Marucci, G.; Nesi, M.; Mnromanelli, M.N.Romanelli; Teodori, E.; Angeli, P. | |
Isomeric N,N-dicyclohexane-4-ol-amine aryl esters: the discovery of a new class of highly potent and efficacious Pgp-dependent MDR inhibitors | 2007 | Elisabetta Teodori; Cecilia Martelli; Milena Salerno; Nacira Darghal; Silvia Dei; Fulvio Gualtieri; Dina Manetti; Serena Scapecchi; Maria Novella Romanelli | |
Isomeric N,N-dicyclohexane-4-ol-amine aryl esters: chemical and pharmacological development of highly potent and efficacious Pgp-dependent MDR inhibitors | 2007 | Cecilia Martelli; Elisabetta Teodori; Silvia Dei; Marcella Coronnello; Enrico Mini; Giampietro Sgaragli; Daniela Alderighi; Milena Salerno | |
ISOMERIC N,N-BIS(CYCLOHEXANOL)AMINE ARYL ESTERS: THE DISCOVERY OF A NEW CLASS OF HIGHLY POTENT P-GLYCOPROTEIN (PGP)-DEPENDENT MULTIDRUG RESISTANCE (MDR) INHIBITORS | 2007 | Teodori, Elisabetta; Martelli, Cecilia; Salerno, M.; Darghal, N.; Dei, Silvia; GARNIER SUILLEROT, A.; Gualtieri, Fulvio; Manetti, Dina; Scapecchi, Serena; Romanelli, MARIA NOVELLA | |
N,N-bis(alkanol)amine aryl esters and N,N-bis(cyclohexanol)amine aryl esters: Idantification of a new class of Pgp-dependent multidrug resistance (MDR) reverters andowed with potencies in the nanomolar range | 2008 | Silvia Dei; Cecilia Martelli; Elisabetta Teodori; Dina Manetti; Marcella Coronnello; Milena Salerno; Giampietro Sgaragli; Fulvio Gualtieri | |
Multidrug resistance (MDR) modulators: Verapamil offsprings and heterocyclic derivatives | 2008 | E. Teodori; S. Dei; C. Martelli; S. Scapecchi; F. Gualtieri | |
SAR studies in a series of N,N-bis(arylaLKANOL)AMINE ARYL ESTERS AS p-GLYCOPROTEIN (Pgp) dependent multidrug resistance (MDR) inhibitors | 2009 | Elisabetta Teodori; Cecilia Martelli; Milena Salerno; Silvia Dei; Fulvio Gualtieri; Dina Manetti; Francesca Orlandi; Serena Scapecchi; Maria Novella Romanelli | |
Design and synthesis of multidrug resistance (MDR) inhibitors | 2009 | Cecilia Martelli; Francesca Orlandi; Silvia Dei; Elisabetta Teodori | |
Design, synthesis and nootropic activity of new analogues of sunifiram and sapunifiram, two potent cognition-enhancers. | 2009 | Martini, Elisabetta; Salvicchi, A.; Ghelardini, Carla; Manetti, Dina; Dei, Silvia; Guandalini, Luca; Martelli, Cecilia; Melchiorre, Michele; Cellai, Cristina; Scapecchi, Serena; Teodori, Elisabetta; Romanelli, MARIA NOVELLA | |
N,N-bis(cyclohexanol)amine aryl esters: a new class of highly potent Pgp-dependent multidrug resistance (MDR) inhibitors | 2009 | Martelli, Cecilia; Alderighi, Daniela; Coronnello, MARCELLA MARIA; Dei, Silvia; Frosini, Maria; Bozec, Benedicte Le; Manetti, Dina; Neri, Annalisa; Romanelli, MARIA NOVELLA; Salerno, Milena; Scapecchi, Serena; Mini, Enrico; Sgaragli, Giampietro; Teodori, Elisabetta | |
Inhibition of P-glycoprotein-mediated multidrug resistance (MDR) by N,N-bis(cyclohexanol)amine aryl esters: structure-activity relationships | 2010 | Teodori E.; Martelli C.; Dei S.; Frosini M.; Manetti D.; Neri A.; Orlandi F.; Romanelli M.N.; Scapecchi S.; Salerno M.; Sgaragli G. | |
N,N-bis(cyclohexanol)amine aryl esters: the discovery of a new class of highly potent inhibitors of transporter-dependent multidrug resistance (MDR) | 2010 | Teodori, Elisabetta; Dei, Silvia; Martelli, Cecilia; Scapecchi, Serena | |
Structure-activity relationships studies in a series of N,N-bis(alkanol)amine aryl esters as P-glycoprotein (Pgp) dependent multidrug resistance (MDR) inhibitors | 2010 | Martelli, Cecilia; Coronnello, MARCELLA MARIA; Dei, Silvia; Manetti, Dina; Orlandi, Francesca; Scapecchi, Serena; Romanelli, MARIA NOVELLA; Salerno, M.; Mini, Enrico; Teodori, Elisabetta | |
Synthesis, Affinity Profile and Functional Activity of Potent Chiral Muscarinic Antagonists with a Pyrrolidinylfuran Structure | 2010 | S. Scapecchi; M. Nesi; R. Matucci; C. Bellucci; M. Buccioni; S. Dei; L. Guandalini; D. Manetti; C. Martelli; E. Martini; G. Marucci; F. Orlandi; M. N. Romanelli; E. Teodori; R. Cirilli | |
The Novel Potent Multidrug Resistance Inhibitors N,N-bis(cyclohexanol)amine Aryl Esters Are Devoid of Vascular Effects | 2011 | S. Saponara; B. Gorelli; V. Tzankova; C. Martelli; E. Teodori; G. Sgaragli; F. Fusi | |
Inhibition of P-glycoprotein-mediated Multidrug Resistance (MDR) by N,N-bis(cyclohexanol)amine aryl esters: further restriction of molecular flexibility maintains high potency and efficacy | 2011 | Martelli, Cecilia; Dei, Silvia; Lambert, C.; Manetti, Dina; Orlandi, Francesca; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Salerno, M.; Teodori, Elisabetta | |
New structure–activity relationship studies in a series of N,N-bis(cyclohexanol)amine aryl esters as potent reversers of P-glycoprotein-mediated multidrug resistance (MDR) | 2013 | F. Orlandi; M. Coronnello; C. Bellucci; S. Dei; L. Guandalini; D. Manetti; C. Martelli; M. N. Romanelli; S. Scapecchi; M. Salerno; H. Menif; I. Bello; E. Mini; E. Teodori |
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