MARTELLI, CECILIA

MARTELLI, CECILIA  

Scienze farmaceutiche (attivo dal 01/08/1980 al 31/12/2012)  

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Risultati 1 - 20 di 40 (tempo di esecuzione: 0.034 secondi).
Titolo Data di pubblicazione Autore(i) File
2-PYRROLIDINONE MOIETY IS NOT CRITICAL FOR THE COGNITION ENHANCING ACTIVITY OF PIRACETAM-LIKE DRUGS 2003 S. SCAPECCHI; C. MARTELLI; C. GHELARDINI; L. GUANDALINI; E. MARTINI; F. GUALTIERI
Design and synthesis of multidrug resistance (MDR) inhibitors 2009 Cecilia Martelli; Francesca Orlandi; Silvia Dei; Elisabetta Teodori
Design, synthesis and nootropic activity of new analogues of sunifiram and sapunifiram, two potent cognition-enhancers. 2009 Martini, Elisabetta; Salvicchi, A.; Ghelardini, Carla; Manetti, Dina; Dei, Silvia; Guandalini, Luca; Martelli, Cecilia; Melchiorre, Michele; Cellai, Cristina; Scapecchi, Serena; Teodori, Elisabetta; Romanelli, MARIA NOVELLA
Design, synthesis and pharmacological evaluation of some frozen-analogues of DMPP 2003 L. Guandalini; M.N. Romanelli; S. Scapecchi; D. Manetti; C. Martelli; E. Martini; S. Dei; E. Teodori; F. Gualtieri; K. Varani; P.A.Borea
Design, synthesis and preliminary biological evaluation of zatebradine analogues as potential blockers of the hyperpolarization-activated current 2005 Romanelli, MARIA NOVELLA; Cerbai, Elisabetta; Dei, Silvia; Guandalini, Luca; Martelli, Cecilia; Martini, Elisabetta; Scapecchi, Serena; Teodori, Elisabetta; Mugelli, Alessandro
Diphenylcyclohexylamine derivatives as new potent multidrug resistance (MDR) modulators 2005 S. DEI; R. BUDRIESI; P. SUDWAN; M. FERRARONI; A. CHIARINI; A. GARNIER-SUILLEROT; D. MANETTI; C. MARTELLI; S. SCAPECCHI; E. TEODORI
Exploratory chemistry toward the identification of a new class of MDR reverters inspired by pervilleine and verapamil models 2005 Teodori, Elisabetta; Dei, Silvia; GARNIER SUILLEROT, A.; Gualtieri, Fulvio; Manetti, Dina; Martelli, Cecilia; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Sudwan, P.; Salerno, M.
Exploratory Chemistry toward the identification of new classes of MDR reverters 2005 Elisabetta Teodori; Silvia Dei; Arlette Garnier-Suillerot; Fulvio Gualtieri; Luca Guandalini; Dina Manetti; Cecilia Martelli; Maria Novella Romanelli; Serena Scapecchi
Highly chiral muscarinic ligands: synthesis and affinity of diastereomeric and enantiomeric isomers of 1-methyl-2-(2-methyl-1,3-oxathiolane-5-yl)pyrrolidine 3-sulfoxides and their methyl iodides 2003 Serena Scapecchi; Cecilia Martelli; Elisabetta Martini; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Luca Guandalini; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori
Highly chiral muscarinic ligands: the discovery of (2S,2'R,3'S,5'R)-1-methyl-2-(2-methyl-1,3-oxathiolan-5-yl)pyrrolidine 3-sulfoxide methyl iodide, a potent, functionally selective, M2 partial agonist. 2006 Scapecchi, Serena; Matucci, Rosanna; Bellucci, Cristina; Buccioni, M.; Dei, Silvia; Guandalini, Luca; Martelli, Cecilia; Manetti, Dina; Martini, Elisabetta; Marucci, G.; Nesi, Marta; Romanelli, MARIA NOVELLA; Teodori, Elisabetta; Gualtieri, Fulvio
Inhibition of P-glycoprotein-mediated Multidrug Resistance (MDR) by N,N-bis(cyclohexanol)amine aryl esters: further restriction of molecular flexibility maintains high potency and efficacy 2011 Martelli, Cecilia; Dei, Silvia; Lambert, C.; Manetti, Dina; Orlandi, Francesca; Romanelli, MARIA NOVELLA; Scapecchi, Serena; Salerno, M.; Teodori, Elisabetta
Inhibition of P-glycoprotein-mediated multidrug resistance (MDR) by N,N-bis(cyclohexanol)amine aryl esters: structure-activity relationships 2010 Teodori E.; Martelli C.; Dei S.; Frosini M.; Manetti D.; Neri A.; Orlandi F.; Romanelli M.N.; Scapecchi S.; Salerno M.; Sgaragli G.
Isomeric N,N-(dicyclohexane-4-ol)amine aryl esters: the discovery of a new class of highly potent and efficacious Pgp-dependent MDR inhibitors 2006 E. Teodori; C. Martelli; D. Manetti; S. Dei; M.N.Romanelli; S. Scapecchi; M. Salerno; A.Garnier-Suillerot; F. Gualtieri
ISOMERIC N,N-BIS(CYCLOHEXANOL)AMINE ARYL ESTERS: THE DISCOVERY OF A NEW CLASS OF HIGHLY POTENT P-GLYCOPROTEIN (PGP)-DEPENDENT MULTIDRUG RESISTANCE (MDR) INHIBITORS 2007 Teodori, Elisabetta; Martelli, Cecilia; Salerno, M.; Darghal, N.; Dei, Silvia; GARNIER SUILLEROT, A.; Gualtieri, Fulvio; Manetti, Dina; Scapecchi, Serena; Romanelli, MARIA NOVELLA
Isomeric N,N-dicyclohexane-4-ol-amine aryl esters: chemical and pharmacological development of highly potent and efficacious Pgp-dependent MDR inhibitors 2007 Cecilia Martelli; Elisabetta Teodori; Silvia Dei; Marcella Coronnello; Enrico Mini; Giampietro Sgaragli; Daniela Alderighi; Milena Salerno
Isomeric N,N-dicyclohexane-4-ol-amine aryl esters: the discovery of a new class of highly potent and efficacious Pgp-dependent MDR inhibitors 2007 Elisabetta Teodori; Cecilia Martelli; Milena Salerno; Nacira Darghal; Silvia Dei; Fulvio Gualtieri; Dina Manetti; Serena Scapecchi; Maria Novella Romanelli
Modulazione molecolare di antagonisti muscarinici. Sintesi e valutazione farmacologica preliminare di esteri amminoalchil piperazinici e piperidinici dell'acido 2,2-difenil-2-etiltioacetico 2004 S. Scapecchi; E. Martini; C. Bellucci; S. Dei; L. Guandalini; D. Manetti; C. Martelli; G. Marucci; R. Matucci
MOLECULAR MODULATION OF MUSCARINIC ANTAGONISTS. SYNTHESIS AND AFFINITY PROFILE OF 2,2-DIPHENYL-2-ETHYLTHIO-ACETIC ACID ESTERS DESIGNED TO PROBE THE BINDING SITE CAVITY 2004 S. SCAPECCHI; E. MARTINI; C. BELLUCCI; M. BUCCIONI; S. DEI; L. GUANDALINI; D. MANETTI; C. MARTELLI; G. MARUCCI; R. MATUCCI
Molecular modulation of muscarinic antagonists. Synthesis and pharmacological profile of 2,2-diphenyl-2-ethylthioacetic acid and 3,3-diphenyl-3-ethylthiopropionic acid derivatives characterized by a dipeptide spacer 2003 Serena Scapecchi; Piero Angeli; Cristina Bellucci; Silvia Dei; Fulvio Gualtieri; Cecilia Martelli; Gabriella Marucci; Rosanna Matucci; Maria Novella Romanelli; Elisabetta Teodori
MOLECULAR MODULATION OF MUSCARINIC ANTAGONISTS. SYNTHESIS AND PHARMACOLOGICAL PROFILE OF 2,2-DIPHENYL-2-ETHYLTHIOACETIC AND 3,3-DIPHENYL-3-ETHYLTHIOPROPIONIC ACID DERIVATIVES CHARACTERIZED BY A DIPEPTIDE SPACER 2004 S. SCAPECCHI; C. MARTELLI; P. ANGELI; C. BELLUCCI; M. BUCCIONI; S. DEI; F. GUALTIERI; G. MARUCCI; R. MATUCCI; M. ROMANELLI; E. TEODORI