CROCETTI, LETIZIA
CROCETTI, LETIZIA
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulators
2021 Crocetti, Letizia; Guerrini, Gabriella; Cantini, Niccolò; Vergelli, Claudia; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors
2021 Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria
1H-pyrrolo[2,3-b]pyridine: a new scaffold for human neutrophil elastase (HNE) inhibitors
2018 Letizia Crocetti, Maria Paola Giovannoni, Igor A. Schepetkinb, Mark T. Quinn, Andrei I. Khlebnikovc, Niccolò Cantini, Gabriella Guerrini, Antonella Iacovone, Elisabetta Teodori, Claudia Vergelli
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists.
2016 Vergelli, C; Schepetkin, I.A; Ciciani, G; Cilibrizzi, A; Crocetti, L; Giovannoni, M.P; Guerrini, G; Iacovone, A; Kirpotina, L.N; Khlebnikov, A.I; Ye, R.D; Quinn, M.T.
3,8-Disubstituted Pyrazolo[1,5-a]quinazoline as GABAA Receptor Modulators: Synthesis, Electrophysiological Assays, and Molecular Modelling Studies
2024 Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola
4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor Subtype
2023 Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola
A patenting perspective on human neutrophil elastase (HNE) inhibitors (2014-2018) and their therapeutic applications
2019 Crocetti L.; Quinn M.T.; Schepetkin I.A.; Giovannoni M.P.
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases.
2009 L. Crocetti;A. Maresca;C. Temperini;R. A. Hall;A. Scozzafava;F. A. Mühlschlegel;C. T. Supuran
An Overview of PDE4 Inhibitors in Clinical Trials: 2010 to Early 2022
2022 Crocetti, Letizia; Floresta, Giuseppe; Cilibrizzi, Agostino; Giovannoni, Maria Paola
Anti-Inflammatory Activity of Pyrazolo[1,5-a]quinazolines
2024 Crocetti, Letizia; Khlebnikov, Andrei I.; Guerrini, Gabriella; Schepetkin, Igor A.; Melani, Fabrizio; Giovannoni, Maria Paola; Quinn, Mark T.
Cinnoline derivatives as human neutrophil elastase inhibitors
2016 Giovannoni, Maria Paola; Crocetti, Letizia; Ciciani, Giovanna; Cilibrizzi, Agostino; Guerrini, Gabriella; Vergelli, Claudia
Design and synthesis of the first indole-based blockers of Panx-1 channel
2021 Crocetti, Letizia; Guerrini, Gabriella; Puglioli, Sara; Giovannoni, Maria Paola; Di Cesare Mannelli, Lorenzo; Lucarini, Elena; Ghelardini, Carla; Wang, Junjie; Dahl, Gerhard
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase
2011 L. Crocetti; M.P. Giovannoni; I.A. Schepetkin; M.T. Quinn; A.I. Khlebnikov; A. Cilibrizzi; V. Dal Piaz; A. Graziano; C. Vergelli
Design, Synthesis and Pharmacological Evaluation of New Quinoline-Based Panx-1 Channel Blockers
2023 Crocetti, Letizia; Giovannoni, Maria Paola; Guerrini, Gabriella; Lamanna, Silvia; Melani, Fabrizio; Bartolucci, Gian Luca; Pallecchi, Marco; Paoli, Paola; Lippi, Martina; Wang, Junjie; Dahl, Gerhard
Ebselen analogues with dual human neutrophil elastase (HNE) inhibitory and antiradical activity
2024 Crocetti, Letizia; Catarzi, Francesca; Giovannoni, Maria Paola; Vergelli, Claudia; Bartolucci, Gianluca; Pallecchi, Marco; Paoli, Paola; Rossi, Patrizia; Lippi, Martina; Schepetkin, Igor A.; Quinn, Mark T.; Guerrini, Gabriella
Editorial: Serine protease inhibitors and their therapeutic applications
2022 Crocetti, Letizia; Quinn, Mark T; Cilibrizzi, Agostino; Giovannoni, Maria Paola
Exploration of Nitrogen Heterocycle Scaffolds for the Development of Potent Human Neutrophil Elastase Inhibitors
2021 Cantini, Niccolò; Khlebnikov, Andrei I.; Crocetti, Letizia; Schepetkin, Igor A.; Floresta, Giuseppe; Guerrini, Gabriella; Vergelli, Claudia; Bartolucci, Gianluca; Quinn, Mark T.; Paola Giovannoni, Maria
Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: synthesis and evaluation of their phosphodiesterase 4 inhibitory activity
2010 P.Biagini; C.Biancalani; A.Graziano; N.Cesari; M.Giovannoni; A.Cilibrizzi; V.Dal Piaz; C.Vergelli; L.Crocetti; M.Delcanale; E.Armani; A.Rizzi; P.Puccini; P.Gallo; D.Spinabelli; P.Caruso
Further modifications of 1H-pyrrolo[2,3-b]pyridine derivatives as inhibitors of human neutrophil elastase
2019 Giovannoni M.P.; Cantini N.; Crocetti L.; Guerrini G.; Iacovone A.; Schepetkin I.A.; Vergelli C.; Khlebnikov A.I.; Quinn M.T.
Further studies on 2-arylacetamide pyridazin-3(2H)-ones: design, synthesis and evaluation of 4,6-disubstituted analogs as formyl peptide receptors (FPRs) agonists.
2013 M.P. Giovannoni; I.A. Schepetkin; A. Cilibrizzi; L. Crocetti; A.I. Khlebnikov; C. Dahlgren; A. Graziano; V. Dal Piaz; L.N. Kirpotina; S. Zerbinati; C. Vergelli; M.T. Quinn
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulators | 2021 | Crocetti, Letizia; Guerrini, Gabriella; Cantini, Niccolò; Vergelli, Claudia; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola | |
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors | 2021 | Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria | |
1H-pyrrolo[2,3-b]pyridine: a new scaffold for human neutrophil elastase (HNE) inhibitors | 2018 | Letizia Crocetti, Maria Paola Giovannoni, Igor A. Schepetkinb, Mark T. Quinn, Andrei I. Khlebnikovc, Niccolò Cantini, Gabriella Guerrini, Antonella Iacovone, Elisabetta Teodori, Claudia Vergelli | |
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists. | 2016 | Vergelli, C; Schepetkin, I.A; Ciciani, G; Cilibrizzi, A; Crocetti, L; Giovannoni, M.P; Guerrini, G; Iacovone, A; Kirpotina, L.N; Khlebnikov, A.I; Ye, R.D; Quinn, M.T. | |
3,8-Disubstituted Pyrazolo[1,5-a]quinazoline as GABAA Receptor Modulators: Synthesis, Electrophysiological Assays, and Molecular Modelling Studies | 2024 | Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola | |
4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor Subtype | 2023 | Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola | |
A patenting perspective on human neutrophil elastase (HNE) inhibitors (2014-2018) and their therapeutic applications | 2019 | Crocetti L.; Quinn M.T.; Schepetkin I.A.; Giovannoni M.P. | |
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases. | 2009 | L. Crocetti;A. Maresca;C. Temperini;R. A. Hall;A. Scozzafava;F. A. Mühlschlegel;C. T. Supuran | |
An Overview of PDE4 Inhibitors in Clinical Trials: 2010 to Early 2022 | 2022 | Crocetti, Letizia; Floresta, Giuseppe; Cilibrizzi, Agostino; Giovannoni, Maria Paola | |
Anti-Inflammatory Activity of Pyrazolo[1,5-a]quinazolines | 2024 | Crocetti, Letizia; Khlebnikov, Andrei I.; Guerrini, Gabriella; Schepetkin, Igor A.; Melani, Fabrizio; Giovannoni, Maria Paola; Quinn, Mark T. | |
Cinnoline derivatives as human neutrophil elastase inhibitors | 2016 | Giovannoni, Maria Paola; Crocetti, Letizia; Ciciani, Giovanna; Cilibrizzi, Agostino; Guerrini, Gabriella; Vergelli, Claudia | |
Design and synthesis of the first indole-based blockers of Panx-1 channel | 2021 | Crocetti, Letizia; Guerrini, Gabriella; Puglioli, Sara; Giovannoni, Maria Paola; Di Cesare Mannelli, Lorenzo; Lucarini, Elena; Ghelardini, Carla; Wang, Junjie; Dahl, Gerhard | |
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase | 2011 | L. Crocetti; M.P. Giovannoni; I.A. Schepetkin; M.T. Quinn; A.I. Khlebnikov; A. Cilibrizzi; V. Dal Piaz; A. Graziano; C. Vergelli | |
Design, Synthesis and Pharmacological Evaluation of New Quinoline-Based Panx-1 Channel Blockers | 2023 | Crocetti, Letizia; Giovannoni, Maria Paola; Guerrini, Gabriella; Lamanna, Silvia; Melani, Fabrizio; Bartolucci, Gian Luca; Pallecchi, Marco; Paoli, Paola; Lippi, Martina; Wang, Junjie; Dahl, Gerhard | |
Ebselen analogues with dual human neutrophil elastase (HNE) inhibitory and antiradical activity | 2024 | Crocetti, Letizia; Catarzi, Francesca; Giovannoni, Maria Paola; Vergelli, Claudia; Bartolucci, Gianluca; Pallecchi, Marco; Paoli, Paola; Rossi, Patrizia; Lippi, Martina; Schepetkin, Igor A.; Quinn, Mark T.; Guerrini, Gabriella | |
Editorial: Serine protease inhibitors and their therapeutic applications | 2022 | Crocetti, Letizia; Quinn, Mark T; Cilibrizzi, Agostino; Giovannoni, Maria Paola | |
Exploration of Nitrogen Heterocycle Scaffolds for the Development of Potent Human Neutrophil Elastase Inhibitors | 2021 | Cantini, Niccolò; Khlebnikov, Andrei I.; Crocetti, Letizia; Schepetkin, Igor A.; Floresta, Giuseppe; Guerrini, Gabriella; Vergelli, Claudia; Bartolucci, Gianluca; Quinn, Mark T.; Paola Giovannoni, Maria | |
Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: synthesis and evaluation of their phosphodiesterase 4 inhibitory activity | 2010 | P.Biagini; C.Biancalani; A.Graziano; N.Cesari; M.Giovannoni; A.Cilibrizzi; V.Dal Piaz; C.Vergelli; L.Crocetti; M.Delcanale; E.Armani; A.Rizzi; P.Puccini; P.Gallo; D.Spinabelli; P.Caruso | |
Further modifications of 1H-pyrrolo[2,3-b]pyridine derivatives as inhibitors of human neutrophil elastase | 2019 | Giovannoni M.P.; Cantini N.; Crocetti L.; Guerrini G.; Iacovone A.; Schepetkin I.A.; Vergelli C.; Khlebnikov A.I.; Quinn M.T. | |
Further studies on 2-arylacetamide pyridazin-3(2H)-ones: design, synthesis and evaluation of 4,6-disubstituted analogs as formyl peptide receptors (FPRs) agonists. | 2013 | M.P. Giovannoni; I.A. Schepetkin; A. Cilibrizzi; L. Crocetti; A.I. Khlebnikov; C. Dahlgren; A. Graziano; V. Dal Piaz; L.N. Kirpotina; S. Zerbinati; C. Vergelli; M.T. Quinn |