VULLO, DANIELA

VULLO, DANIELA  

Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)  

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1,2-Benzisothiazole Derivatives Bearing 4-, 5-, or 6-Alkyl/arylcarboxamide Moieties Inhibit Carbonic Anhydrase Isoform IX (CAIX) and Cell Proliferation under Hypoxic Conditions 2016 Coviello, Vito; Marchi, Beatrice; Sartini, Stefania; Quattrini, Luca; Marini, Anna Maria; Simorini, Francesca; Taliani, Sabrina; Salerno, Silvia; Orlandi, Paola; Fioravanti, Anna; Desidero, Teresa Di; Vullo, Daniela; Da Settimo, Federico; Supuran, Claudiu T; Bocci, Guido; La Motta, Concettina
3-phenyl-1H-indole-5-sulfonamides: structure-based drug design of a promising class of carbonic anhydrase inhibitors. 2010 O. Güzel;A. Innocenti;D. Vullo;A. Scozzafava;C. T. Supuran
3H-1,2-benzoxathiepine 2,2-dioxides: a new class of isoform-selective carbonic anhydrase inhibitors 2017 Pustenko, Aleksandrs; Stepanovs, Dmitrijs; Žalubovskis, Raivis; Vullo, Daniela; Kazaks, Andris; Leitans, Janis; Tars, Kaspars; Supuran, Claudiu T
4-Functionalized 1,3-diarylpyrazoles bearing benzenesulfonamide moiety as selective potent inhibitors of the tumor associated carbonic anhydrase isoforms IX and XII 2014 Khloya, Poonam; Celik, Gulsah; Sitaram, Null; Vullo, Daniela; Supuran, Claudiu T.; Sharma, Pawan K
5-Substituted-benzylsulfanyl-thiophene-2-sulfonamides with effective carbonic anhydrase inhibitory activity: Solution and crystallographic investigations 2017 Ivanova, Jekaterīna; Balode, Agnese; Žalubovskis, Raivis; Leitans, Janis; Kazaks, Andris; Vullo, Daniela; Tars, Kaspars; Supuran, Claudiu T.
7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. 2015 Vullo, Daniela*; Isik, Semra; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T.
A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors 2019 Costa G.; Carta F.; Ambrosio F.A.; Artese A.; Ortuso F.; Moraca F.; Rocca R.; Romeo I.; Lupia A.; Maruca A.; Bagetta D.; Catalano R.; Vullo D.; Alcaro S.; Supuran C.T.
A Divalent PAMAM-Based Matrix Metalloproteinase/Carbonic Anhydrase Inhibitor for the Treatment of Dry Eye Syndrome 2016 Richichi, B.; Baldoneschi, V.; Burgalassi, S.; Fragai, M.; Vullo, D.; Akdemir, A.; Dragoni, E.; Louka, A.; Mamusa, M.; Monti, D.; Berti, D.; Novellino, E.; Rosa, G. De; Supuran, C.T.; Nativi, C.
A highly catalytically active γ-carbonic anhydrase from the pathogenic anaerobe Porphyromonas gingivalis and its inhibition profile with anions and small molecules. 2013 S. D. Prete;D. Vullo;V. D. Luca;V. Carginale;A. Scozzafava;C. T. Supuran;C. Capasso
A new procedure for the cloning, expression and purification of the β-carbonic anhydrase from the pathogenic yeast Malassezia globosa, an anti-dandruff drug target 2016 Del Prete, Sonia; De Luca, Viviana; Vullo, Daniela; Osman, Sameh M.; Alothman, Zeid; Carginale, Vincenzo; Supuran, Claudiu T.; Capasso, Clemente
A new way of synthesizing heterocyclic primary sulfonamide probes for carbonic anhydrase 2023 Krivovicheva, Vasilisa; Bubyrev, Andrey; Kalinin, Stanislav; Dar'in, Dmitry; Gureev, Maxim; Vullo, Daniela; Krasavin, Mikhail; Korsakov, Mikhail; Supuran, Claudiu T.
A new β-carbonic anhydrase from Brucella suis, its cloning, characterization, and inhibition with sulfonamides and sulfamates, leading to impaired pathogen growth. 2011 P. Joseph;S. Ouahrani-Bettache;J. Montero;I. Nishimori;T. Minakuchi;D. Vullo;A. Scozzafava;J. Winum;S. Köhler;C. T. Supuran
A prodrug approach toward cancer-related carbonic anhydrase inhibition 2013 Carroux, Cindy J.; Rankin, Gregory M.; Moeker, Janina; Bornaghi, Laurent F.; Katneni, Kasiram; Morizzi, Julia; Charman, Susan A.; Vullo, Daniela; Supuran, Claudiu T; Poulsen, Sally-Ann
A Series of Thiadiazolyl-Benzenesulfonamides Incorporating an Aromatic Tail as Isoform-Selective, Potent Carbonic Anhydrase II/XII Inhibitors 2022 Banoglu, Erden; Ercanlı, Taner; Gür Maz, Tuğçe; Vullo, Daniela; Bonardi, Alessandro; Gratteri, Paola; Supuran, Claudiu T
A Spectroscopic Study of the Reaction of NAMI, a Novel Ruthenium(III) Antineoplastic Complex, with Bovine Serum Albumin. Eur. J. Biochem. 2000, 267 (4), 1206-13. 2000 L. MESSORI; ORIOLI P; VULLO D.; ALESSIO E; IENGO E
A substituted sulfonamide and its Co (II), Cu (II), and Zn (II) complexes as potential antifungal agents 2016 Diaz, Jorge R. A.; Fernández Baldo, Martín; Echeverría, Gustavo; Baldoni, Héctor; Vullo, Daniela; Soria, Delia B.; Supuran, Claudiu T.; Camí, Gerardo E
Acetaldehyde-derived modifications on cytosolic human carbonic anhydrases. 2011 F. Bootorabi;J. Jänis;V. P. Hytönen;J. Valjakka;M. Kuuslahti;D. Vullo;O. Niemelä;C. T. Supuran;S. Parkkila
Activation Profile Analysis of CruCA4, an α-Carbonic Anhydrase Involved in Skeleton Formation of the Mediterranean Red Coral, Corallium rubrum 2017 Del Prete, Sonia; Vullo, Daniela; Zoccola, Didier; Tambutté, Sylvie; Supuran, Claudiu T; Capasso, Clemente
Active components of essential oils as anti-obesity potential drugs investigated by in silico techniques 2016 Costa, Giosuè; Gidaro, Maria Concetta; Vullo, Daniela; Supuran, Claudiu T.; Alcaro, Stefano
An anion and small molecule inhibition study of the β-carbonic anhydrase from Staphylococcus aureus 2021 Urbanski, Linda J; Vullo, Daniela; Parkkila, Seppo; Supuran, Claudiu T