TANC, MUHAMMET

TANC, MUHAMMET  

Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)  

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Titolo Data di pubblicazione Autore(i) File
3-Hydroxy-1H-quinazoline-2,4-dione as a New Scaffold to Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII 2017 Falsini, Matteo; Squarcialupi, Lucia; Catarzi, Daniela; Varano, Flavia; Betti, Marco; Di Cesare Mannelli, Lorenzo; Tenci, Barbara; Ghelardini, Carla; Tanc, Muhammet; Angeli, Andrea; Supuran, Claudiu T.; Colotta, Vittoria
3-Hydroxy-1H-quinazoline-2,4-dione derivatives as new potent and selective inhibitors of the tumor-associated carbonic anhydrase IX and XII. 2015 Squarcialupi, L.; Falsini, M.; Catarzi, D.; Varano, F.; Betti, M.; Di Cesare Mannelli, L.; Zanardelli, M.; Ghelardini, C.; Tanc, M.; Supuran, C.T.; Colotta, V.
5-Aryl-1H-pyrazole-3-carboxylic acids as selective inhibitors of human carbonic anhydrases IX and XII 2015 Cvijetić, Ilija N; Tanç, Muhammet; Juranić, Ivan O.; Verbić, Tatjana Ž.; Supuran, Claudiu T.; Drakulić, Branko J.
5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: Solution and X-ray crystallographic studies 2013 Leitans, Janis; Sprudza, Agnese; Tanc, Muhammet; Vozny, Igor; Zalubovskis, Raivis; Tars, Kaspars; Supuran, Claudiu T.
6-Substituted 1,2-benzoxathiine-2,2-dioxides are isoform-selective inhibitors of human carbonic anhydrases IX, XII and VA. 2015 M. Tanc;F. Carta;A. Scozzafava;C. T. Supuran
6-substituted sulfocoumarins are selective carbonic anhdydrase IX and XII Inhibitors with significant cytotoxicity against colorectal cancer cells 2015 Grandane, Aiga; Tanc, Muhammet; Di Cesare Mannelli, Lorenzo; Carta, Fabrizio; Ghelardini, Carla; Žalubovskis, Raivis; Supuran, Claudiu T.
6-Triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrases IX and XII 2014 Grandane, Aiga; Tanc, Muhammet; Zalubovskis, Raivis; Supuran, Claudiu T.
9,10-Dibromo-N-aryl-9,10-dihydro-9,10-[3,4]epipyrroloanthracene-12,14-diones: Synthesis and Investigation of Their Effects on Carbonic Anhydrase Isozymes I, II, IX, and XII 2016 Göksu, Haydar; Topal, Meryem; Keskin, Ali; Gültekin, Mehmet S.; Çelik, Murat; Gülçin, Ilhami; Tanc, Muhammet; Supuran, Claudiu T.
A class of carbonic anhydrase I – selective activators 2016 Licsandru, Erol; Tanc, Muhammet; Kocsis, Istvan; Barboiu, Mihail; Supuran, Claudiu T.
Carbonic anhydrase inhibition and cytotoxicity studies of Mannich base derivatives of thymol 2016 Inci Gul, Halise; Yamali, Cem; Tugce Yasa, Asiye; Unluer, Elif; Sakagami, Hiroshi; Tanc, Muhammet; Supuran, Claudiu T.
Carbonic anhydrase inhibitors: Synthesis and inhibition of the cytosolic mammalian carbonic anhydrase isoforms I, II and VII with benzene sulfonamides incorporating 4,5,6,7-tetrachlorophthalimide moiety 2013 Sethi, Kalyan K; Verma, Saurabh M.; Tanç, Muhammet; Carta, Fabrizio; Supuran, Claudiu T.
Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, IX and XII with benzene sulfonamides incorporating 4- and 3-nitrophthalimide moieties 2014 Sethi, Kalyan K; Verma, Saurabh M.; Tanç, Muhammet; Purper, Gaultier; Calafato, Gaetan; Carta, Fabrizio; Supuran, Claudiu T.
Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety 2013 Sethi, Kalyan K; Vullo, Daniella; Verma, Saurabh M.; Tanç, Muhammet; Carta, Fabrizio; Supuran, Claudiu T.
CO2-capture by engineered mammalian carbonic anhydrases 2019 Nocentini A.; Tanc M.
Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies 2018 Nocentini, Alessio; Carta, Fabrizio; Tanc, Muhammet; Selleri, Silvia; Supuran, Claudiu T.; Bazzicalupi, Carla*; Gratteri, Paola
Dominant behaviours in the expression of human carbonic anhydrase hCA i activity 2014 Abdelrahim, M. Yahia M.; Tanc, Muhammet; Winum, Jean-Yves; Supuran, Claudiu T; Barboiu, Mihail
Effective Access to Multivalent Inhibitors of Carbonic Anhydrases Promoted by Peptide Bioconjugation 2017 Kanfar, Nasreddine; Tanc, Muhammet; Dumy, Pascal; Supuran, Claudiu T; Ulrich, Sébastien; Winum, Jean-Yves
Exploring carbonic anhydrase inhibition with multimeric coumarins displayed on a fullerene scaffold 2015 Abellán-Flos, Marta; Tanç, Muhammet; Supuran, Claudiu T.; Vincent, Stéphane P.
Fluorinated pyrrolidines and piperidines incorporating tertiary benzenesulfonamide moieties are selective carbonic anhydrase II inhibitors 2015 Le Darz, Alexandre; Mingot, Agnès; Bouazza, Fodil; Castelli, Ugo; Karam, Omar; Tanc, Muhammet; Supuran, Claudiu T.; Thibaudeau, Sébastien
Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds 2017 Krasavin, Mikhail; Korsakov, Mikhail; Zvonaryova, Zhanna; Semyonychev, Evgenii; Tuccinardi, Tiziano; Kalinin, Stanislav; Tanç, Muhammet; Supuran, Claudiu T