BOZDAG, MURAT
BOZDAG, MURAT
Chimica 'Ugo Schiff' - DICUS
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site
2020 Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V.
7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring.
2015 Vullo, Daniela*; Isik, Semra; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T.
A class of 4-Sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.
2014 M. Bozdag;M. Pinard;F. Carta;E. Masini;A. Scozzafava;R. McKenna;C. T. Supuran
A non-catalytic function of carbonic anhydrase IX contributes to the glycolytic phenotype and pH regulation in human breast cancer cells
2019 Mboge M.Y.; Chen Z.; Khokhar D.; Wolff A.; Ai L.; Heldermon C.D.; Bozdag M.; Carta F.; Supuran C.T.; Brown K.D.; McKenna R.; Frost C.J.; Frost S.C.
Azidothymidine "clicked" into 1,2,3-Triazoles: First Report on Carbonic Anhydrase-Telomerase Dual-Hybrid Inhibitors
2020 Berrino E.; Angeli A.; Zhdanov D.D.; Kiryukhina A.P.; Milaneschi A.; De Luca A.; Bozdag M.; Carradori S.; Selleri S.; Bartolucci G.; Peat T.S.; Ferraroni M.; Supuran C.T.; Carta F.
Benzamide-4-sulfonamides are effective human carbonic anhydrase I, II, VII, and IX inhibitors
2018 Abdoli M.; Bozdag M.; Angeli A.; Supuran C.T.
Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity
2015 Bozdag, Murat; Alafeefy, Ahmed M.; Vullo, Daniela; Carta, Fabrizio; Dedeoglu, Nurcan; Al-Tamimi, Abdul-Malek S.; Al-Jaber, Nabila A.; Scozzafava, Andrea; Supuran, Claudiu T
Benzylaminoethylureido-Tailed Benzenesulfonamides Show Potent Inhibitory Activity against Bacterial Carbonic Anhydrases
2020 Ali M.; Angeli A.; Bozdag M.; Carta F.; Capasso C.; Farooq U.; Supuran C.T.
Benzylaminoethyureido-Tailed Benzenesulfonamides: Design, Synthesis, Kinetic and X-ray Investigations on Human Carbonic Anhydrases
2020 Ali, Majid; Bozdag, Murat; Farooq, Umar; Angeli, Andrea; Carta, Fabrizio; Berto, Paola; Zanotti, Giuseppe; Supuran, Claudiu T
Carbonic anhydrase I, II, IV and IX inhibition with a series of 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives
2017 Bozdag, Murat; Bua, Silvia; Osman, Sameh M; AlOthman, Zeid; Supuran, Claudiu T
Carbonic anhydrase inhibitors based on sorafenib scaffold: Design, synthesis, crystallographic investigation and effects on primary breast cancer cells
2019 Bozdag, Murat; Ferraroni, Marta; Ward, Carol; Carta, Fabrizio; Bua, Silvia; Angeli, Andrea; Langdon, Simon P; Kunkler, Ian H; Al-Tamimi, Abdul-Malek S; Supuran, Claudiu T
Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: Solution and X-ray crystallographic studies
2014 Bozdag M.; Ferraroni M.; Nuti E.; Vullo D.; Rossello A.; Carta F.; Scozzafava A.; Supuran C.T.
Coumarins and other fused bicyclic heterocycles with selective tumor-associated carbonic anhydrase isoforms inhibitory activity
2017 Bozdag, Murat; Alafeefy, Ahmed Mahmoud; Altamimi, Abdul Malik; Vullo, Daniela; Carta, Fabrizio; Supuran, Claudiu T.
Cyclodextrin complexation highly enhances efficacy of arylsulfonylureido benzenesulfonamide carbonic anhydrase inhibitors as a topical antiglaucoma agents
2015 Bragagni, Marco; Bozdag, Murat; Carta, Fabrizio; Scozzafava, Andrea; Lanzi, Cecilia; Masini, Emanuela; Mura, Paola; Supuran, Claudiu T.
Dithiocarbamates effectively inhibit the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa
2017 Vullo, Daniela; Del Prete, Sonia; Nocentini, Alessio; Osman, Sameh M.; Alothman, Zeid; Capasso, Clemente; Bozdag, Murat; Carta, Fabrizio; Gratteri, Paola; Supuran, Claudiu T.
Dithiocarbamates with potent inhibitory activity against the Saccharomyces cerevisiae β-carbonic anhydrase
2016 Bozdag, Murat; Carta, Fabrizio; Vullo, Daniela*; Isik, Semra; AlOthman, Zeid; Osman, Sameh M.; Scozzafava, Andrea; Supuran, Claudiu T.
In vitro inhibition of Mycobacterium tuberculosis β-carbonic anhydrase 3 with Mono- and dithiocarbamates and evaluation of their toxicity using zebrafish developing embryos
2020 Aspatwar, Ashok; Hammaren, Milka; Parikka, Mataleena; Parkkila, Seppo; Carta, Fabrizio; Bozdag, Murat; Vullo, Daniela; Supuran, Claudiu T
Inhibition of carbonic anhydrases by a substrate analog: benzyl carbamate directly coordinates the catalytic zinc ion mimicking bicarbonate binding
2018 De Simone G.; Angeli A.; Bozdag M.; Supuran C.T.; Winum J.-Y.; Monti S.M.; Alterio V.
Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N'-aryl-N-hydroxy-ureas
2018 Berrino, Emanuela; Bozdag, Murat; Del Prete, Sonia; Alasmary, Fatmah A S; Alqahtani, Linah S; AlOthman, Zeid; Capasso, Clemente; Supuran, Claudiu T
Mono- and di-thiocarbamate inhibition studies of the δ-carbonic anhydrase TweCAδ from the marine diatom Thalassiosira weissflogii
2018 Bua, Silvia; Bozdag, Murat; Del Prete, Sonia; Carta, Fabrizio; Donald, William A; Capasso, Clemente; Supuran, Claudiu T