FILACCHIONI, GUIDO

FILACCHIONI, GUIDO  

Scienze farmaceutiche (attivo dal 01/08/1980 al 31/12/2012)  

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Titolo Data di pubblicazione Autore(i) File
. PYRROLNITRIN ANALOGS. XII. SYNTHESIS AND BIOLOGICAL ACTIVITY OF SOME PYRAZOLE CARBOXYLIC ACIDS. 1986 G. PALAZZINO; F. MELANI; L. CECCHI; G. FILACCHIONI
1,2,4-Triazolo[1,5-a]quinoxaline as a versatile tool for the design of selective human A3 adenosine receptor antagonists: synthesis, biological evaluation and molecular modeling studies of 2-(hetero)aryl- and 2-carboxy-substituted derivatives. 2005 D. CATARZI; V. COLOTTA; F. VARANO; O. LENZI; G. FILACCHIONI; L. TRINCAVELLI; C. MARTINI; C. MONOPOLI; S. MORO
1,2,4-Triazolo[4,3-a]quinoxalin-1-one: a versatile tool for the synthesis of potent and selective adenosine receptor antagonists. 2000 V. COLOTTA; D. CATARZI; F. VARANO; L.CECCHI; G.FILACCHIONI; C. MARTINI; L. TRINCAVELLI; A. LUCACCHINI
1,3-DIARYLPYRAZOLO[4,5-C]- AND -[5,4-C]QUINOLIN-4-ONES. 4. SYNTHESIS AND SPECIFIC INHIBITION OF BENZODIAZEPINE RECEPTOR BINDING. 1987 G. PALAZZINO; L. CECCHI; F. MELANI; V. COLOTTA; G. FILACCHIONI; C. MARTINI; A. LUCACCHINI
1-(3-Aminophenyl)-3-methyl[1]benzopyrano[2,3-c]pyrazol-4-one: a new selective A2 adenosine receptor antagonist. 1992 V.Colotta; L.Cecchi; D.Catarzi; F.Melani; G.Filacchioni; C.Martini; P.Tacchi; A.Lucacchini
1-Substituted pyrazolo[1,5-c]quinazolines as novel Gly/NMDA receptor antagonists: synthesis, biological evaluation and molecular modeling study 2005 F.VARANO; D. CATARZI; V. COLOTTA; F. R. CALABRI; O. LENZI; G. FILACCHIONI; A. GALLI; C. COSTAGLI; F. DEFLORIAN; S. MORO
2-Aryl-8-chloro-1,2,4-triazolo[1,5-a]quinoxalin-4-amines as highly potent A1 and A3 adenosine receptor antagonists 2005 D.CATARZI; V.COLOTTA; F. VARANO; F.R.CALABRI; O.LENZI; G. FILACCHIONI; L.TRINCAVELLI; C. MARTINI; A.TRALLI; C.MONTOPOLI; S.MORO
2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a New Scaffold to obtain Potent and Selective Human A3 Adenosine Receptor Antagonists: New Insights into the Receptor-Antagonist Recognition† 2009 O. Lenzi; V. Colotta; D. Catarzi; F. Varano; D. Poli; G. Filacchioni; K. Varani; F. Vincenzi; P. A. Borea; S. Paoletta; E. Morizzo; S. Moro.
4,5-Dihydro-1,2,4-triazolo[1,5-a]quinoxalin-4-ones. Excitatory amino acid antagonists with combined glycine/NMDA and AMPA receptor affinity 1999 D. CATARZI; V. COLOTTA; F. VARANO; L. CECCHI; G. FILACCHIONI; A. GALLI; C. COSTAGLI
4-Amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as New Potent and Selective Human A3 Adenosine Receptor Antagonists. Synthesis, Pharmacological Evaluation and Ligand-Receptor Modeling Studies. 2006 O. LENZI; V. COLOTTA; D. CATARZI; F.VARANO; G. FILACCHIONI; C. MARTINI; L. TRINCAVELLI; OSELE CIAMPI; KATIA VARANI; FEDERICO MARIGHETTI; ERIKA MORIZZO; STEFANO MORO
4-Amino-2-chloro-1,3,5-triazine: a new metabolite of atrazine by a soil bacterium. 1980 M.Giardina; M. Giardi; G.Filacchioni
4-Amino-6-benzylamino-1,2-dihydro-2-phenyl-1,2,4-triazolo[4,3-a] quinoxalin-1-one: a new A2A adenosine receptor antagonist with high selectivity versus A1 receptors. 1999 V. COLOTTA; D. CATARZI; F. VARANO; L. CECCHI; G. FILACCHIONI; C. MARTINI; L. TRINCAVELLI; A. LUCACCHINI
7-Chloro-4,5-dihydro-8-(1,2,4-triazol-4-yl)-4-oxo-1,2,4-triazolo[1,5-a]quinoxaline-2-carboxylates as novel highly selective AMPA receptor antagonists. 2000 D.CATARZI; V.COLOTTA; F.VARANO; L.CECCHI; G.FILACCHIONI; A.GALLI; C. COSTAGLI; V.CARLA'
[1]Benzopyrano-pyrazole-3-ones. Correct and generalized synthetic metod 1987 V. Colotta; L. Cecchi; G. Filacchioni; F. Melani; G. Palazzino.
[1]Benzopyrano-pyrazole-4-ones. Synthesis, binding studies and structure-activity relationships 1987 V. Colotta; L. Cecchi; ; G. Filacchioni; F. Melani; G. Palazzino; C. Martini; A. Lucacchini.
Antiblastic agents. XXXVI. Anthramycin and analogous compounds. 1. Synthesis of 10,11-dihydro-5H-pyrrolo-[2,1-s][1,4]-benzodiazepine. 1969 M.Artico; G.De Martino; G.Filacchioni; R.Giuliano
Antiblastic substances. LII. Tylophorine analogs. 1. Synthesis and cytostotic and cytotoxic activity of 4-(3,4-dimethoxyphenyl)piperidine. 1973 V.Nacci; G.Stefancich; R.Giuliano; G.Filacchioni
Atrazine metabolism by Nocardia: elucidation of initial pathway and synthesis of potential metabolites. 1982 M.Giardina; M. Giardi; G. Filacchioni
Benzodiazepine binding activity of some tricyclic heteroarometic systems to define the hydrogen bonding strength of the proton donors of the receptor site. 1996 V. COLOTTA; D. CATARZI; F. VARANO; F. MELANI; G.FILACCHIONI; L. CECCHI; A. GALLI; C. COSTAGLI
Chemical and biological degradation of primary metabolites of atrazine by a Nocardia strain. 1985 M. GIARDI; M.GIARDINA; G.FILACCHIONI