VERGELLI, CLAUDIA
VERGELLI, CLAUDIA
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulators
2021 Crocetti, Letizia; Guerrini, Gabriella; Cantini, Niccolò; Vergelli, Claudia; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors
2021 Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria
1H-pyrrolo[2,3-b]pyridine: a new scaffold for human neutrophil elastase (HNE) inhibitors
2018 Letizia Crocetti, Maria Paola Giovannoni, Igor A. Schepetkinb, Mark T. Quinn, Andrei I. Khlebnikovc, Niccolò Cantini, Gabriella Guerrini, Antonella Iacovone, Elisabetta Teodori, Claudia Vergelli
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists.
2016 Vergelli, C; Schepetkin, I.A; Ciciani, G; Cilibrizzi, A; Crocetti, L; Giovannoni, M.P; Guerrini, G; Iacovone, A; Kirpotina, L.N; Khlebnikov, A.I; Ye, R.D; Quinn, M.T.
4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor Subtype
2023 Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola
4-AMINO-3(2H)-PYRIDAZINONES BEARING ARYLPIPERAZINYLALKYL GROUPS AND RELATED COMPOUNDS: SYNTHESIS AND ANTINOCICEPTIVE ACTIVITY
2003 V. DAL PIAZ; M. GIOVANNONI; C. VERGELLI; M. SCHEIDELER; G. PETRONE; P. ZARATIN
4-Amino-5-substituted-3(2H)-pyridazinones as orally active antinociceptive agents: synthesis and studies on the mechanism of action
2007 M.GIOVANNONI; N.CESARI; C.VERGELLI; A.GRAZIANO; C.BIANCALANI; P.BIAGINI; C.GHELARDINI; E.VIVOLI; V.DAL PIAZ
4-amino-5-vinyl-3(2H)-pyridazinones and analogues as potent antinociceptive agents: synthesis, SARs, and preliminary studies on the mechanism of action
2007 C.VERGELLI; M.GIOVANNONI; S.PIERETTI; A.DI GIANNUARIO; V. DAL PIAZ; P.BIAGINI; C.BIANCALANI; A.GRAZIANO; N.CESARI
4-amino-5-vinyl-3(2H)-pyridazinones and related compounds: synthesis and evaluation of antinociceptive activity
2002 V. DAL PIAZ; PIERETTI S.; VERGELLI C.; CASTELLANA M.C.; GIOVANNONI M.P.
6-Methyl-2,4-disubstituted pyridazin-3(2H)-ones: a novel class of small-molecule agonists for formyl peptide receptors.
2009 A. CILIBRIZZI; M.T.QUINN; L.N. KIRPOTINA; I.A.SCHEPETKIN; J.HOLDERNESS; R.D.YE; M.J. RABIET; C.BIANCALANI; N. CESARI; A. GRAZIANO; C.VERGELLI; S.PIERETTI; V.DAL PIAZ; M.P.GIOVANNONI.
[(3-chlorophenyl)piperazinylpropyl]pyridazinones and analogues as potent antinociceptive agents
2003 GIOVANNONI M.P.; VERGELLI C.; GHELARDINI C.; GALEOTTI N.; BARTOLINI A.; V. DAL PIAZ
AIRWAY RELAXANT AND ANTI-INFLAMMATORY PROPERTIES OF A PDE 4 INHIBITOR WITH LOW AFFINITY FOR THE HIGH-AFFINITY ROLIPRAM BINDING SITE
2002 C. MARTIN; R. GOGGEL; V. DAL PIAZ; C. VERGELLI; M. GIOVANNONI; M. ERNST; S. UHLIG
Alpha-2-agonist as analgesic agents
2009 M. Giovannoni; C. Ghelardini; C. Vergelli; V. Dal Piaz
Arylpiperazinylalkylpyridazinones and analogues as potent and orally active antinociceptive agents: synthesis and studies on mechanism of action
2006 N.CESARI; C.BIANCALANI; C.VERGELLI; V. DAL PIAZ; A.GRAZIANO; P.BIAGINI; C.GHELARDINI; N.GALEOTTI; M.GIOVANNONI
Cinnoline derivatives as human neutrophil elastase inhibitors
2016 Giovannoni, Maria Paola; Crocetti, Letizia; Ciciani, Giovanna; Cilibrizzi, Agostino; Guerrini, Gabriella; Vergelli, Claudia
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase
2011 L. Crocetti; M.P. Giovannoni; I.A. Schepetkin; M.T. Quinn; A.I. Khlebnikov; A. Cilibrizzi; V. Dal Piaz; A. Graziano; C. Vergelli
Ebselen analogues with dual human neutrophil elastase (HNE) inhibitory and antiradical activity
2024 Crocetti, Letizia; Catarzi, Francesca; Giovannoni, Maria Paola; Vergelli, Claudia; Bartolucci, Gianluca; Pallecchi, Marco; Paoli, Paola; Rossi, Patrizia; Lippi, Martina; Schepetkin, Igor A.; Quinn, Mark T.; Guerrini, Gabriella
Effects of the neutrophil elastase inhibitor EL-17 in rat adjuvant-induced arthritis.
2016 Di Cesare Mannelli, L; Micheli, L; Cinci, L; Maresca, M; Vergelli, C; Pacini, A; Quinn, M.T.; Giovannoni, M. P.; Ghelardini, C.
Exploration of Nitrogen Heterocycle Scaffolds for the Development of Potent Human Neutrophil Elastase Inhibitors
2021 Cantini, Niccolò; Khlebnikov, Andrei I.; Crocetti, Letizia; Schepetkin, Igor A.; Floresta, Giuseppe; Guerrini, Gabriella; Vergelli, Claudia; Bartolucci, Gianluca; Quinn, Mark T.; Paola Giovannoni, Maria
Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: synthesis and evaluation of their phosphodiesterase 4 inhibitory activity
2010 P.Biagini; C.Biancalani; A.Graziano; N.Cesari; M.Giovannoni; A.Cilibrizzi; V.Dal Piaz; C.Vergelli; L.Crocetti; M.Delcanale; E.Armani; A.Rizzi; P.Puccini; P.Gallo; D.Spinabelli; P.Caruso
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulators | 2021 | Crocetti, Letizia; Guerrini, Gabriella; Cantini, Niccolò; Vergelli, Claudia; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola | |
| 1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors | 2021 | Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria | |
| 1H-pyrrolo[2,3-b]pyridine: a new scaffold for human neutrophil elastase (HNE) inhibitors | 2018 | Letizia Crocetti, Maria Paola Giovannoni, Igor A. Schepetkinb, Mark T. Quinn, Andrei I. Khlebnikovc, Niccolò Cantini, Gabriella Guerrini, Antonella Iacovone, Elisabetta Teodori, Claudia Vergelli | |
| 2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists. | 2016 | Vergelli, C; Schepetkin, I.A; Ciciani, G; Cilibrizzi, A; Crocetti, L; Giovannoni, M.P; Guerrini, G; Iacovone, A; Kirpotina, L.N; Khlebnikov, A.I; Ye, R.D; Quinn, M.T. | |
| 4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor Subtype | 2023 | Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola | |
| 4-AMINO-3(2H)-PYRIDAZINONES BEARING ARYLPIPERAZINYLALKYL GROUPS AND RELATED COMPOUNDS: SYNTHESIS AND ANTINOCICEPTIVE ACTIVITY | 2003 | V. DAL PIAZ; M. GIOVANNONI; C. VERGELLI; M. SCHEIDELER; G. PETRONE; P. ZARATIN | |
| 4-Amino-5-substituted-3(2H)-pyridazinones as orally active antinociceptive agents: synthesis and studies on the mechanism of action | 2007 | M.GIOVANNONI; N.CESARI; C.VERGELLI; A.GRAZIANO; C.BIANCALANI; P.BIAGINI; C.GHELARDINI; E.VIVOLI; V.DAL PIAZ | |
| 4-amino-5-vinyl-3(2H)-pyridazinones and analogues as potent antinociceptive agents: synthesis, SARs, and preliminary studies on the mechanism of action | 2007 | C.VERGELLI; M.GIOVANNONI; S.PIERETTI; A.DI GIANNUARIO; V. DAL PIAZ; P.BIAGINI; C.BIANCALANI; A.GRAZIANO; N.CESARI | |
| 4-amino-5-vinyl-3(2H)-pyridazinones and related compounds: synthesis and evaluation of antinociceptive activity | 2002 | V. DAL PIAZ; PIERETTI S.; VERGELLI C.; CASTELLANA M.C.; GIOVANNONI M.P. | |
| 6-Methyl-2,4-disubstituted pyridazin-3(2H)-ones: a novel class of small-molecule agonists for formyl peptide receptors. | 2009 | A. CILIBRIZZI; M.T.QUINN; L.N. KIRPOTINA; I.A.SCHEPETKIN; J.HOLDERNESS; R.D.YE; M.J. RABIET; C.BIANCALANI; N. CESARI; A. GRAZIANO; C.VERGELLI; S.PIERETTI; V.DAL PIAZ; M.P.GIOVANNONI. | |
| [(3-chlorophenyl)piperazinylpropyl]pyridazinones and analogues as potent antinociceptive agents | 2003 | GIOVANNONI M.P.; VERGELLI C.; GHELARDINI C.; GALEOTTI N.; BARTOLINI A.; V. DAL PIAZ | |
| AIRWAY RELAXANT AND ANTI-INFLAMMATORY PROPERTIES OF A PDE 4 INHIBITOR WITH LOW AFFINITY FOR THE HIGH-AFFINITY ROLIPRAM BINDING SITE | 2002 | C. MARTIN; R. GOGGEL; V. DAL PIAZ; C. VERGELLI; M. GIOVANNONI; M. ERNST; S. UHLIG | |
| Alpha-2-agonist as analgesic agents | 2009 | M. Giovannoni; C. Ghelardini; C. Vergelli; V. Dal Piaz | |
| Arylpiperazinylalkylpyridazinones and analogues as potent and orally active antinociceptive agents: synthesis and studies on mechanism of action | 2006 | N.CESARI; C.BIANCALANI; C.VERGELLI; V. DAL PIAZ; A.GRAZIANO; P.BIAGINI; C.GHELARDINI; N.GALEOTTI; M.GIOVANNONI | |
| Cinnoline derivatives as human neutrophil elastase inhibitors | 2016 | Giovannoni, Maria Paola; Crocetti, Letizia; Ciciani, Giovanna; Cilibrizzi, Agostino; Guerrini, Gabriella; Vergelli, Claudia | |
| Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastase | 2011 | L. Crocetti; M.P. Giovannoni; I.A. Schepetkin; M.T. Quinn; A.I. Khlebnikov; A. Cilibrizzi; V. Dal Piaz; A. Graziano; C. Vergelli | |
| Ebselen analogues with dual human neutrophil elastase (HNE) inhibitory and antiradical activity | 2024 | Crocetti, Letizia; Catarzi, Francesca; Giovannoni, Maria Paola; Vergelli, Claudia; Bartolucci, Gianluca; Pallecchi, Marco; Paoli, Paola; Rossi, Patrizia; Lippi, Martina; Schepetkin, Igor A.; Quinn, Mark T.; Guerrini, Gabriella | |
| Effects of the neutrophil elastase inhibitor EL-17 in rat adjuvant-induced arthritis. | 2016 | Di Cesare Mannelli, L; Micheli, L; Cinci, L; Maresca, M; Vergelli, C; Pacini, A; Quinn, M.T.; Giovannoni, M. P.; Ghelardini, C. | |
| Exploration of Nitrogen Heterocycle Scaffolds for the Development of Potent Human Neutrophil Elastase Inhibitors | 2021 | Cantini, Niccolò; Khlebnikov, Andrei I.; Crocetti, Letizia; Schepetkin, Igor A.; Floresta, Giuseppe; Guerrini, Gabriella; Vergelli, Claudia; Bartolucci, Gianluca; Quinn, Mark T.; Paola Giovannoni, Maria | |
| Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: synthesis and evaluation of their phosphodiesterase 4 inhibitory activity | 2010 | P.Biagini; C.Biancalani; A.Graziano; N.Cesari; M.Giovannoni; A.Cilibrizzi; V.Dal Piaz; C.Vergelli; L.Crocetti; M.Delcanale; E.Armani; A.Rizzi; P.Puccini; P.Gallo; D.Spinabelli; P.Caruso |