GRIFAGNI, DEBORAH
GRIFAGNI, DEBORAH
Chimica 'Ugo Schiff' - DICUS
1H, 13C and 15N assignment of the human mitochondrial paramagnetic iron-sulfur protein CISD3
2022 Silva, José Malanho; Grifagni, Deborah; Cantini, Francesca; Piccioli, Mario
A Structural Investigation of the Interaction between a GC-376-Based Peptidomimetic PROTAC and Its Precursor with the Viral Main Protease of Coxsackievirus B3
2024 De Santis, Alessia; Grifagni, Deborah; Orsetti, Andrea; Lenci, Elena; Rosato, Antonio; D'Onofrio, Mariapina; Trabocchi, Andrea; Ciofi-Baffoni, Simone; Cantini, Francesca; Calderone, Vito
An antiviral agent triggering the proteolysis of the main protease from Coxsackievirus B3
2023 Alessia De Santis, Andrea Orsetti , Deborah Grifagni , Elena Lenci , Francesca Lucarelli , Francesca Cantini , Vito Calderone , Andrea Trabocchi , Mariapina D’Onofrio, Simone Ciofi-Baffoni
Application of the PROTAC-based approach to trigger proteolysis of the Coxsackievirus B3 main protease
2025 Alessia De Santis, Deborah Grifagni, Andrea Orsetti, Chiara La Guidara, Niccolò Moradei, Koi L. Merz, Elena Lenci, Antonio Rosato, Mariapina D’Onofrio, Andrea Trabocchi, Simone Ciofi-Baffoni, Francesca Cantini, Vito Calderone
Biochemical and cellular characterization of the CISD3 protein: molecular bases of cluster release and destabilizing effects of nitric oxide
2024 Grifagni, Deborah; Silva, José Malanho; Querci, Leonardo; Lepoivre, Michel; Vallières, Cindy; Louro, Ricardo O.; Banci, Lucia; Piccioli, Mario; Golinelli-Cohen, Marie-Pierre; Cantini, Francesca
CIAO3 protein forms a stable ternary complex with two key players of the human cytosolic iron–sulfur cluster assembly machinery
2020 Maione V.; Grifagni D.; Torricella F.; Cantini F.; Banci L.
Congresso Nazionale della Divisione di Chimica dei Sistemi Biologici
2025 Chiara La Guidara, Alessia De Santis, Niccolò Moradei, Deborah Grifagni, Francesca Cantini, Mariapina D'Onofrio, Alfonso Carotenuto, Simone Ciofi-Baffoni, Antonio Rosato
Development of a GC-376 Based Peptidomimetic PROTAC as a Degrader of 3-Chymotrypsin-like Protease of SARS-CoV-2
2024 Grifagni, Deborah; Lenci, Elena; De Santis, Alessia; Orsetti, Andrea; Barracchia, Carlo Giorgio; Tedesco, Filomena; Bellini Puglielli, Raffaele; Lucarelli, Francesca; Lauriola, Angela; Assfalg, Michael; Cantini, Francesca; Calderone, Vito; Guardavaccaro, Daniele; Trabocchi, Andrea; D’Onofrio, Mariapina; Ciofi-Baffoni, Simone
Exploration of PROTAC technology for the development of broad-spectrum antiviral drugs to trigger the proteolysis of the main viral protease
2025 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, MariapinaD’Onofrio, Simone Ciofi-Baffoni
Gold-Based Metal Drugs as Inhibitors of Coronavirus Proteins: The Inhibition of SARS-CoV-2 Main Protease by Auranofin and Its Analogs
2022 Massai, Lara; Grifagni, Deborah; De Santis, Alessia; Geri, Andrea; Cantini, Francesca; Calderone, Vito; Banci, Lucia; Messori, Luigi
Paramagnetic NMR to study iron sulfur proteins: 13C detected experiments illuminate the vicinity of the metal center
2023 Querci, Leonardo; Grifagni, Deborah; Trindade, Inês B; Malanho da Silva, Jose Pedro; Louro, Ricardo O; Cantini, Francesca; Piccioli, Mario
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis , Deborah Grifagni , Elena Lenci , Andrea Orsetti , Carlo Giorgio Barracchia , Filomena Tedesco , Raffaele Bellini Puglielli , Francesca Lucarelli , Chiara La Guidara , Angela Lauriola , Michael Assfalg , Francesca Cantini , Vito Calderone , Daniele Guardavaccaro , Andrea Trabocchi, Antonio Rosato, Mariapina D'Onofrio , Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco,Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2024 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni
PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease
2023 Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni
Relaxation-based NMR assignment: Spotlights on ligand binding sites in human CISD3
2023 Grifagni D.; Silva J.M.; Cantini F.; Piccioli M.; Banci L.
SARS-CoV-2 Mproinhibition by a zinc ion: structural features and hints for drug design
2021 Grifagni D.; Calderone V.; Giuntini S.; Cantini F.; Fragai M.; Banci L.
Shedding Light on the Electron Delocalization Pathway at the [Fe2S2]2+ Cluster of FDX2
2025 Querci, Leonardo; Fiorucci, Letizia; Grifagni, Deborah; Costantini, Paola; Ravera, Enrico; Ciofi-Baffoni, Simone; Piccioli, Mario
Targeting the Main Protease (Mpro, nsp5) by Growth of Fragment Scaffolds Exploiting Structure-Based Methodologies
2023 Altincekic, Nadide; Jores, Nathalie; Löhr, Frank; Richter, Christian; Ehrhardt, Claus; Blommers, Marcel J. J.; Berg, Hannes; Öztürk, Sare; Gande, Santosh L.; Linhard, Verena; Orts, Julien; Abi Saad, Marie Jose; Bütikofer, Matthias; Kaderli, Janina; Karlsson, B. Göran; Brath, Ulrika; Hedenström, Mattias; Gröbner, Gerhard; Sauer, Uwe H.; Perrakis, Anastassis; Langer, Julian; Banci, Lucia; Cantini, Francesca; Fragai, Marco; Grifagni, Deborah; Barthel, Tatjana; Wollenhaupt, Jan; Weiss, Manfred S.; Robertson, Angus; Bax, Adriaan; Sreeramulu, Sridhar; Schwalbe, Harald
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1H, 13C and 15N assignment of the human mitochondrial paramagnetic iron-sulfur protein CISD3 | 2022 | Silva, José Malanho; Grifagni, Deborah; Cantini, Francesca; Piccioli, Mario | |
| A Structural Investigation of the Interaction between a GC-376-Based Peptidomimetic PROTAC and Its Precursor with the Viral Main Protease of Coxsackievirus B3 | 2024 | De Santis, Alessia; Grifagni, Deborah; Orsetti, Andrea; Lenci, Elena; Rosato, Antonio; D'Onofrio, Mariapina; Trabocchi, Andrea; Ciofi-Baffoni, Simone; Cantini, Francesca; Calderone, Vito | |
| An antiviral agent triggering the proteolysis of the main protease from Coxsackievirus B3 | 2023 | Alessia De Santis, Andrea Orsetti , Deborah Grifagni , Elena Lenci , Francesca Lucarelli , Francesca Cantini , Vito Calderone , Andrea Trabocchi , Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| Application of the PROTAC-based approach to trigger proteolysis of the Coxsackievirus B3 main protease | 2025 | Alessia De Santis, Deborah Grifagni, Andrea Orsetti, Chiara La Guidara, Niccolò Moradei, Koi L. Merz, Elena Lenci, Antonio Rosato, Mariapina D’Onofrio, Andrea Trabocchi, Simone Ciofi-Baffoni, Francesca Cantini, Vito Calderone | |
| Biochemical and cellular characterization of the CISD3 protein: molecular bases of cluster release and destabilizing effects of nitric oxide | 2024 | Grifagni, Deborah; Silva, José Malanho; Querci, Leonardo; Lepoivre, Michel; Vallières, Cindy; Louro, Ricardo O.; Banci, Lucia; Piccioli, Mario; Golinelli-Cohen, Marie-Pierre; Cantini, Francesca | |
| CIAO3 protein forms a stable ternary complex with two key players of the human cytosolic iron–sulfur cluster assembly machinery | 2020 | Maione V.; Grifagni D.; Torricella F.; Cantini F.; Banci L. | |
| Congresso Nazionale della Divisione di Chimica dei Sistemi Biologici | 2025 | Chiara La Guidara, Alessia De Santis, Niccolò Moradei, Deborah Grifagni, Francesca Cantini, Mariapina D'Onofrio, Alfonso Carotenuto, Simone Ciofi-Baffoni, Antonio Rosato | |
| Development of a GC-376 Based Peptidomimetic PROTAC as a Degrader of 3-Chymotrypsin-like Protease of SARS-CoV-2 | 2024 | Grifagni, Deborah; Lenci, Elena; De Santis, Alessia; Orsetti, Andrea; Barracchia, Carlo Giorgio; Tedesco, Filomena; Bellini Puglielli, Raffaele; Lucarelli, Francesca; Lauriola, Angela; Assfalg, Michael; Cantini, Francesca; Calderone, Vito; Guardavaccaro, Daniele; Trabocchi, Andrea; D’Onofrio, Mariapina; Ciofi-Baffoni, Simone | |
| Exploration of PROTAC technology for the development of broad-spectrum antiviral drugs to trigger the proteolysis of the main viral protease | 2025 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, MariapinaD’Onofrio, Simone Ciofi-Baffoni | |
| Gold-Based Metal Drugs as Inhibitors of Coronavirus Proteins: The Inhibition of SARS-CoV-2 Main Protease by Auranofin and Its Analogs | 2022 | Massai, Lara; Grifagni, Deborah; De Santis, Alessia; Geri, Andrea; Cantini, Francesca; Calderone, Vito; Banci, Lucia; Messori, Luigi | |
| Paramagnetic NMR to study iron sulfur proteins: 13C detected experiments illuminate the vicinity of the metal center | 2023 | Querci, Leonardo; Grifagni, Deborah; Trindade, Inês B; Malanho da Silva, Jose Pedro; Louro, Ricardo O; Cantini, Francesca; Piccioli, Mario | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis , Deborah Grifagni , Elena Lenci , Andrea Orsetti , Carlo Giorgio Barracchia , Filomena Tedesco , Raffaele Bellini Puglielli , Francesca Lucarelli , Chiara La Guidara , Angela Lauriola , Michael Assfalg , Francesca Cantini , Vito Calderone , Daniele Guardavaccaro , Andrea Trabocchi, Antonio Rosato, Mariapina D'Onofrio , Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco,Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2024 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Chiara La Guidara, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Antonio Rosato, Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| PROTAC-based approach to develop broad-spectrum antiviral agents triggering the proteolysis of the major viral protease | 2023 | Alessia De Santis, Deborah Grifagni, Elena Lenci, Andrea Orsetti, Carlo Giorgio Barracchia, Filomena Tedesco, Raffaele Bellini Puglielli, Francesca Lucarelli, Angela Lauriola, Michael Assfalg, Francesca Cantini, Vito Calderone, Daniele Guardavaccaro, Andrea Trabocchi, Mariapina D’Onofrio, Simone Ciofi-Baffoni | |
| Relaxation-based NMR assignment: Spotlights on ligand binding sites in human CISD3 | 2023 | Grifagni D.; Silva J.M.; Cantini F.; Piccioli M.; Banci L. | |
| SARS-CoV-2 Mproinhibition by a zinc ion: structural features and hints for drug design | 2021 | Grifagni D.; Calderone V.; Giuntini S.; Cantini F.; Fragai M.; Banci L. | |
| Shedding Light on the Electron Delocalization Pathway at the [Fe2S2]2+ Cluster of FDX2 | 2025 | Querci, Leonardo; Fiorucci, Letizia; Grifagni, Deborah; Costantini, Paola; Ravera, Enrico; Ciofi-Baffoni, Simone; Piccioli, Mario | |
| Targeting the Main Protease (Mpro, nsp5) by Growth of Fragment Scaffolds Exploiting Structure-Based Methodologies | 2023 | Altincekic, Nadide; Jores, Nathalie; Löhr, Frank; Richter, Christian; Ehrhardt, Claus; Blommers, Marcel J. J.; Berg, Hannes; Öztürk, Sare; Gande, Santosh L.; Linhard, Verena; Orts, Julien; Abi Saad, Marie Jose; Bütikofer, Matthias; Kaderli, Janina; Karlsson, B. Göran; Brath, Ulrika; Hedenström, Mattias; Gröbner, Gerhard; Sauer, Uwe H.; Perrakis, Anastassis; Langer, Julian; Banci, Lucia; Cantini, Francesca; Fragai, Marco; Grifagni, Deborah; Barthel, Tatjana; Wollenhaupt, Jan; Weiss, Manfred S.; Robertson, Angus; Bax, Adriaan; Sreeramulu, Sridhar; Schwalbe, Harald |