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NOTA: è possibile cercare una corrispondenza esatta usando i doppi apici, ad es: "evoluzione della specie". Qualora si cerchi un identificativo, è consigliabile cercarlo in due modi differenti: tra apici con caratteri speciali es: "978-94-6366-274" oppure senza caratteri speciali solo come sequenza numerica: es 978946366274.
Mono- and three-tailed sugar and iminosugar decorated benzenesulfonamide carbonic anhydrase inhibitors
2023 Maria Giulia Davighi, Camilla Matassini, Andrea Goti, Marta Ferraroni, Andrea Angeli, Claudiu T. Supuran, Francesca Cardona
First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome
2023 Andrea Angeli; Marta Ferraroni; Carlotta Granchi; Filippo Minutolo; Xiaozhuo Chen; Pratik Shriwas; Emilio Russo; Antonio Leo; Silvia Selleri; Fabrizio Carta; Claudiu T. Supuran
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran
4-Cyanamido-substituted benzenesulfonamides act as dual carbonic anhydrase and cathepsin inhibitors
2023 Abdoli, Morteza; Krasniqi, Vesa; Bonardi, Alessandro; Gütschow, Michael; Supuran, Claudiu T; Žalubovskis, Raivis
6-Aminocoumarin oxime-ether/sulfonamides as selective hCA IX and XII inhibitors: Synthesis, evaluation, and molecular dynamics studies
2023 Ghouse, Shaik Mahammad; Sinha, Kareena; Bonardi, Alessandro; Pawar, Gaurav; Malasala, Satyaveni; Danaboina, Srikanth; Mohammed, Arifuddin; Yaddanapudi, Venkata M; Supuran, Claudiu T; Nanduri, Srinivas
Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties
2023 Tekeli, Tuba; Akocak, Suleyman; Petreni, Andrea; Lolak, Nebih; Çete, Servet; Supuran, Claudiu T
Expression Dynamics of CA IX Epitope in Cancer Cells under Intermittent Hypoxia Correlates with Extracellular pH Drop and Cell Killing by Ureido-Sulfonamide CA IX Inhibitors
2023 Sufian, Md Abu; Zamanova, Sabina; Shabana, Ahmed M; Kemp, Brianna; Mondal, Utpal K; Supuran, Claudiu T; Ilies, Marc A
Inhibition Studies on Carbonic Anhydrase Isoforms I, II, IX, and XII with a Series of Sulfaguanidines
2023 Abdoli, Morteza; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T; Žalubovskis, Raivis
Synthesis, biological evaluation and theoretical studies of (E)-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitors
2023 Ramzan, Farhat; Nabi, Syed Ayaz; Lone, Mehak Saba; Bonardi, Alessandro; Hamid, Aabid; Bano, Sameena; Sharma, Kalicharan; Shafi, Syed; Samim, Mohammed; Javed, Kalim; Supuran, Claudiu T
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis
2023 Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Mono- and three-tailed sugar and iminosugar decorated benzenesulfonamide carbonic anhydrase inhibitors | 2023 | Maria Giulia Davighi, Camilla Matassini, Andrea Goti, Marta Ferraroni, Andrea Angeli, Claudiu T. Supuran, Francesca Cardona | |
First-in-Class Dual Targeting Compounds for the Management of Seizures in Glucose Transporter Type 1 Deficiency Syndrome | 2023 | Andrea Angeli; Marta Ferraroni; Carlotta Granchi; Filippo Minutolo; Xiaozhuo Chen; Pratik Shriwas; Emilio Russo; Antonio Leo; Silvia Selleri; Fabrizio Carta; Claudiu T. Supuran | |
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran | |
4-Cyanamido-substituted benzenesulfonamides act as dual carbonic anhydrase and cathepsin inhibitors | 2023 | Abdoli, Morteza; Krasniqi, Vesa; Bonardi, Alessandro; Gütschow, Michael; Supuran, Claudiu T; Žalubovskis, Raivis | |
6-Aminocoumarin oxime-ether/sulfonamides as selective hCA IX and XII inhibitors: Synthesis, evaluation, and molecular dynamics studies | 2023 | Ghouse, Shaik Mahammad; Sinha, Kareena; Bonardi, Alessandro; Pawar, Gaurav; Malasala, Satyaveni; Danaboina, Srikanth; Mohammed, Arifuddin; Yaddanapudi, Venkata M; Supuran, Claudiu T; Nanduri, Srinivas | |
Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties | 2023 | Tekeli, Tuba; Akocak, Suleyman; Petreni, Andrea; Lolak, Nebih; Çete, Servet; Supuran, Claudiu T | |
Expression Dynamics of CA IX Epitope in Cancer Cells under Intermittent Hypoxia Correlates with Extracellular pH Drop and Cell Killing by Ureido-Sulfonamide CA IX Inhibitors | 2023 | Sufian, Md Abu; Zamanova, Sabina; Shabana, Ahmed M; Kemp, Brianna; Mondal, Utpal K; Supuran, Claudiu T; Ilies, Marc A | |
Inhibition Studies on Carbonic Anhydrase Isoforms I, II, IX, and XII with a Series of Sulfaguanidines | 2023 | Abdoli, Morteza; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T; Žalubovskis, Raivis | |
Synthesis, biological evaluation and theoretical studies of (E)-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitors | 2023 | Ramzan, Farhat; Nabi, Syed Ayaz; Lone, Mehak Saba; Bonardi, Alessandro; Hamid, Aabid; Bano, Sameena; Sharma, Kalicharan; Shafi, Syed; Samim, Mohammed; Javed, Kalim; Supuran, Claudiu T | |
Novel Insights on CAI-CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis | 2023 | Berrino, Emanuela; Micheli, Laura; Carradori, Simone; di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T |
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Opzioni
Scopri
Tipologia
- 1 - Contributo su rivista 1916
- 1 - Contributo su rivista::1a - Articolo su rivista 1916
Data di pubblicazione
- 2020 - 2024 479
- 2010 - 2019 957
- 2000 - 2009 429
- 1992 - 1999 51
Editore
- Academic Press Inc. 1
- American Chemical Society:1155 Sixteenth Street Northwest:Washington, DC 20036:(800)227-5558, EMAIL: service@acs.org, INTERNET: http://www.pubs.acs.org, Fax: (614)447-3671 1
- Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598 Editore precedente:Prof Ugo Croatto Luogo pubbl. Padova Ultimo luogo pubblicazione: Lausanne. 1
- John Libby Eurotext Ltd:127 avenue de la Republique, F 92120 Montrouge France:011 33 1 46730660, EMAIL: marketing@jle.com, INTERNET: http://www.john-libbey-eurotext.fr, Fax: 011 33 1 40840999 1
- TAYLOR & FRANCIS LTD 1
Rivista
- JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY 402
- BIOORGANIC & MEDICINAL CHEMISTRY 197
- BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 180
- JOURNAL OF MEDICINAL CHEMISTRY 132
- EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 93
- BIOORGANIC CHEMISTRY 84
- BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS 37
- EXPERT OPINION ON THERAPEUTIC PATENTS 37
- MOLECULES 35
- JOURNAL OF ENZYME INHIBITION 34
Keyword
- Humans 636
- Carbonic Anhydrase Inhibitors 631
- Carbonic Anhydrases 552
- Carbonic anhydrase 407
- Sulfonamides 403
- Structure-Activity Relationship 397
- Drug Discovery3003 Pharmaceutical Science 292
- Molecular Structure 266
- Isoenzymes 254
- Animals 216
Lingua
- eng 1428
- enm 1
- ita 1
Accesso al fulltext
- no fulltext 1630
- open 156
- reserved 121
- partially open 9