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NOTA: è possibile cercare una corrispondenza esatta usando i doppi apici, ad es: "evoluzione della specie". Qualora si cerchi un identificativo, è consigliabile cercarlo in due modi differenti: tra apici con caratteri speciali es: "978-94-6366-274" oppure senza caratteri speciali solo come sequenza numerica: es 978946366274.
Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors
2024 De Luca, Viviana; Angeli, Andrea; Nocentini, Alessio; Gratteri, Paola; Pratesi, Silvia; Tanini, Damiano; Carginale, Vincenzo; Capperucci, Antonella; Supuran, Claudiu T.; Capasso, Clemente
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains
2024 Bua, Silvia; Bonardi, Alessandro; Mük, Georgiana Ramona; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T.
Boron-containing carbonic anhydrases inhibitors
2024 Giovannuzzi, Simone; Nikitjuka, Anna; Pereira Resende, Bruna Rafaela; Smietana, Michael; Nocentini, Alessio; Supuran, Claudiu T.; Winum, Jean-Yves
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy
2024 Angeli A.; Chelli I.; Lucarini L.; Sgambellone S.; Marri S.; Villano S.; Ferraroni M.; De Luca V.; Capasso C.; Carta F.; Supuran C.T.
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction
2024 Giovannuzzi, Simone; Chavarria, Daniel; Provensi, Gustavo; Leri, Manuela; Bucciantini, Monica; Carradori, Simone; Bonardi, Alessandro; Gratteri, Paola; Borges, Fernanda; Nocentini, Alessio; Supuran, Claudiu T.
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids
2024 Morteza Abdoli; Alessandro Bonardi; Paola Gratteri; Claudiu T Supuran; Raivis Žalubovskis
Sulfonamide-incorporated bis(α-aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic studies
2024 Marjan Sobati; Morteza Abdoli; Andrea Angeli; Alessandro Bonardi; Marta Ferraroni; Claudiu T Supuran; Raivis Žalubovskis
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors | 2024 | De Luca, Viviana; Angeli, Andrea; Nocentini, Alessio; Gratteri, Paola; Pratesi, Silvia; Tanini, Damiano; Carginale, Vincenzo; Capperucci, Antonella; Supuran, Claudiu T.; Capasso, Clemente | |
Benzothiadiazinone-1,1-Dioxide Carbonic Anhydrase Inhibitors Suppress the Growth of Drug-Resistant Mycobacterium tuberculosis Strains | 2024 | Bua, Silvia; Bonardi, Alessandro; Mük, Georgiana Ramona; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T. | |
Boron-containing carbonic anhydrases inhibitors | 2024 | Giovannuzzi, Simone; Nikitjuka, Anna; Pereira Resende, Bruna Rafaela; Smietana, Michael; Nocentini, Alessio; Supuran, Claudiu T.; Winum, Jean-Yves | |
Novel Carbonic Anhydrase Inhibitors with Dual-Tail Core Sulfonamide Show Potent and Lasting Effects for Glaucoma Therapy | 2024 | Angeli A.; Chelli I.; Lucarini L.; Sgambellone S.; Marri S.; Villano S.; Ferraroni M.; De Luca V.; Capasso C.; Carta F.; Supuran C.T. | |
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction | 2024 | Giovannuzzi, Simone; Chavarria, Daniel; Provensi, Gustavo; Leri, Manuela; Bucciantini, Monica; Carradori, Simone; Bonardi, Alessandro; Gratteri, Paola; Borges, Fernanda; Nocentini, Alessio; Supuran, Claudiu T. | |
Synthesis, carbonic anhydrase inhibition studies and modelling investigations of phthalimide-hydantoin hybrids | 2024 | Morteza Abdoli; Alessandro Bonardi; Paola Gratteri; Claudiu T Supuran; Raivis Žalubovskis | |
Sulfonamide-incorporated bis(α-aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic studies | 2024 | Marjan Sobati; Morteza Abdoli; Andrea Angeli; Alessandro Bonardi; Marta Ferraroni; Claudiu T Supuran; Raivis Žalubovskis |
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Opzioni
Scopri
Tipologia
- 1 - Contributo su rivista 1917
- 1 - Contributo su rivista::1a - Articolo su rivista 1917
Data di pubblicazione
- 2020 - 2024 480
- 2010 - 2019 957
- 2000 - 2009 429
- 1992 - 1999 51
Editore
- Academic Press Inc. 1
- American Chemical Society:1155 Sixteenth Street Northwest:Washington, DC 20036:(800)227-5558, EMAIL: service@acs.org, INTERNET: http://www.pubs.acs.org, Fax: (614)447-3671 1
- Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598 Editore precedente:Prof Ugo Croatto Luogo pubbl. Padova Ultimo luogo pubblicazione: Lausanne. 1
- John Libby Eurotext Ltd:127 avenue de la Republique, F 92120 Montrouge France:011 33 1 46730660, EMAIL: marketing@jle.com, INTERNET: http://www.john-libbey-eurotext.fr, Fax: 011 33 1 40840999 1
- TAYLOR & FRANCIS LTD 1
Rivista
- JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY 402
- BIOORGANIC & MEDICINAL CHEMISTRY 197
- BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 180
- JOURNAL OF MEDICINAL CHEMISTRY 133
- EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 93
- BIOORGANIC CHEMISTRY 84
- BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS 37
- EXPERT OPINION ON THERAPEUTIC PATENTS 37
- MOLECULES 35
- JOURNAL OF ENZYME INHIBITION 34
Keyword
- Humans 636
- Carbonic Anhydrase Inhibitors 631
- Carbonic Anhydrases 552
- Carbonic anhydrase 407
- Sulfonamides 403
- Structure-Activity Relationship 397
- Drug Discovery3003 Pharmaceutical Science 292
- Molecular Structure 266
- Isoenzymes 254
- Animals 216
Lingua
- eng 1429
- enm 1
- ita 1
Accesso al fulltext
- no fulltext 1634
- open 154
- reserved 120
- partially open 9