Sfoglia per Autore
Auranofin, Et3PAuCl, and Et3PAuI Are Highly Cytotoxic on Colorectal Cancer Cells: A Chemical and Biological Study
2017 Marzo, Tiziano; Cirri, Damiano; Gabbiani, Chiara; Gamberi, Tania; Magherini, Francesca; Pratesi, Alessandro; Guerri, Annalisa; Biver, Tarita; Binacchi, Francesca; Stefanini, Matteo; Arcangeli, Annarosa; Messori, Luigi
DOTA-Derivatives of Octreotide Dicarba-Analogs with High Affinity for Somatostatin sst2,5 Receptors
2017 Pratesi, Alessandro; Ginanneschi, Mauro; Lumini, Marco; Papini, Anna M; Novellino, Ettore; Brancaccio, Diego; Carotenuto, Alfonso
Ruthenium arene complexes with triphenylphosphane ligands: cytotoxicity towards pancreatic cancer cells, interaction with model proteins, and effect of ethacrynic acid substitution
2017 Biancalana, Lorenzo; Pratesi, Alessandro; Chiellini, Federica; Zacchini, Stefano; Funaioli, Tiziana; Gabbiani, Chiara; Marchetti, Fabio
Synthesis of dicarba-cyclooctapeptide Somatostatin analogs by conventional and MW-assisted RCM: A study about the impact of the configuration at Cα of selected amino acids
2017 Pratesi, Alessandro; Stazzoni, Samuele; Lumini, Marco; Sabatino, Giuseppina; Carotenuto, Alfonso; Brancaccio, Diego; Novellino, Ettore; Chinol, Marco; Rovero, Paolo; Ginanneschi, Mauro; Papini, Anna Maria
Mass spectrometry and metallomics: A general protocol to assess stability of metallodrug-protein adducts in bottom-up MS experiments
2017 Michelucci, Elena; Pieraccini, Giuseppe; Moneti, Gloriano; Gabbiani, Chiara; Pratesi, Alessandro; Messori, Luigi
Antiproliferative effects of two gold(I)-N-heterocyclic carbene complexes in A2780 human ovarian cancer cells: A comparative proteomic study
2018 Magherini, Francesca; Fiaschi, Tania; Valocchia, Elisa; Becatti, Matteo; Pratesi, Alessandro; Marzo, Tiziano; Massai, Lara; Gabbiani, Chiara; Landini, Ida; Nobili, Stefania; Mini, Enrico; Messori, Luigi; Modesti, Alessandra; Gamberi, Tania*
The NAMI A-human ferritin system: A biophysical characterization
2018 Ciambellotti, Silvia; Pratesi, Alessandro; Severi, Mirko; Ferraro, Giarita; Alessio, Enzo; Merlino, Antonello*; Messori, Luigi
Reactions of Auranofin and Its Pseudohalide Derivatives with Serum Albumin Investigated through ESI-Q-TOF MS
2018 Alessandro Pratesi, Damiano Cirri, Lorenzo Ciofi, Luigi Messori
Chlorido and bromido oxaliplatin analogues as potential agents for CRC treatment: Solution behavior, protein binding and cytotoxicity evaluation
2018 Marzo, Tiziano; Pratesi, Alessandro; Cirri, Damiano; Pillozzi, Serena; Petroni, Giulia; Guerri, Annalisa; Arcangeli, Annarosa; Messori, Luigi; Gabbiani, Chiara
A Fluorescent Silver(I) Carbene Complex with Anticancer Properties: Synthesis, Characterization, and Biological Studies
2019 Maria Giulia Fabbrini, Damiano Cirri, Alessandro Pratesi, Lorenzo Ciofi, Tiziano Marzo, Annalisa Guerri, Silvia Nistri, Alfonso Dell'Accio, Tania Gamberi, Mirko Severi, Andrea Bencini, Luigi messori
Structural Characterization of a Gold/Serum Albumin Complex
2019 Pratesi, Alessandro; Cirri, Damiano; Fregona, Dolores; Ferraro, Giarita; Giorgio, Anna; Merlino, Antonello; Messori, Luigi
The cisplatin/serum albumin system: A reappraisal
2019 Massai, Lara; Pratesi, Alessandro; Gailer, Jurgen; Marzo, Tiziano; Messori, Luigi
The leading established metal-based drugs: a revisitation of their relevant physico-chemical data
2019 Damiano Cirri, Maria Giulia Fabbrini, Alessandro Pratesi, Lorenzo Ciofi, Lara Massai, Tiziano Marzo, Luigi Messori
Replacement of the Thiosugar of Auranofin with Iodide Enhances the Anticancer Potency in a Mouse Model of Ovarian Cancer
2019 Tiziano Marzo, Lara Massai, Alessandro Pratesi, Matteo Stefanini, Damiano Cirri, Francesca Magherini, Matteo Becatti, Ida Landini, Stefania Nobili, Enrico Mini, Olivia Crociani, Annarosa Arcangeli, Serena Pillozzi, Tania Gamberi, Luigi Messori
ESI MS studies highlight the selective interaction of Auranofin with protein free thiols
2020 Zoppi C.; Messori L.; Pratesi A.
Native mass spectrometry of human carbonic anhydrase I and its inhibitor complexes
2020 Zoppi C.; Nocentini A.; Supuran C.T.; Pratesi A.; Messori L.
Computationally enhanced X-ray diffraction analysis of a gold(III) complex interacting with the human telomeric DNA G-quadruplex. Unravelling non-unique ligand positioning
2022 Cirri, Damiano; Bazzicalupi, Carla; Ryde, Ulf; Bergmann, Justin; Binacchi, Francesca; Nocentini, Alessio; Pratesi, Alessandro; Gratteri, Paola; Messori, Luigi
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Auranofin, Et3PAuCl, and Et3PAuI Are Highly Cytotoxic on Colorectal Cancer Cells: A Chemical and Biological Study | 2017 | Marzo, Tiziano; Cirri, Damiano; Gabbiani, Chiara; Gamberi, Tania; Magherini, Francesca; Pratesi, Alessandro; Guerri, Annalisa; Biver, Tarita; Binacchi, Francesca; Stefanini, Matteo; Arcangeli, Annarosa; Messori, Luigi | |
DOTA-Derivatives of Octreotide Dicarba-Analogs with High Affinity for Somatostatin sst2,5 Receptors | 2017 | Pratesi, Alessandro; Ginanneschi, Mauro; Lumini, Marco; Papini, Anna M; Novellino, Ettore; Brancaccio, Diego; Carotenuto, Alfonso | |
Ruthenium arene complexes with triphenylphosphane ligands: cytotoxicity towards pancreatic cancer cells, interaction with model proteins, and effect of ethacrynic acid substitution | 2017 | Biancalana, Lorenzo; Pratesi, Alessandro; Chiellini, Federica; Zacchini, Stefano; Funaioli, Tiziana; Gabbiani, Chiara; Marchetti, Fabio | |
Synthesis of dicarba-cyclooctapeptide Somatostatin analogs by conventional and MW-assisted RCM: A study about the impact of the configuration at Cα of selected amino acids | 2017 | Pratesi, Alessandro; Stazzoni, Samuele; Lumini, Marco; Sabatino, Giuseppina; Carotenuto, Alfonso; Brancaccio, Diego; Novellino, Ettore; Chinol, Marco; Rovero, Paolo; Ginanneschi, Mauro; Papini, Anna Maria | |
Mass spectrometry and metallomics: A general protocol to assess stability of metallodrug-protein adducts in bottom-up MS experiments | 2017 | Michelucci, Elena; Pieraccini, Giuseppe; Moneti, Gloriano; Gabbiani, Chiara; Pratesi, Alessandro; Messori, Luigi | |
Antiproliferative effects of two gold(I)-N-heterocyclic carbene complexes in A2780 human ovarian cancer cells: A comparative proteomic study | 2018 | Magherini, Francesca; Fiaschi, Tania; Valocchia, Elisa; Becatti, Matteo; Pratesi, Alessandro; Marzo, Tiziano; Massai, Lara; Gabbiani, Chiara; Landini, Ida; Nobili, Stefania; Mini, Enrico; Messori, Luigi; Modesti, Alessandra; Gamberi, Tania* | |
The NAMI A-human ferritin system: A biophysical characterization | 2018 | Ciambellotti, Silvia; Pratesi, Alessandro; Severi, Mirko; Ferraro, Giarita; Alessio, Enzo; Merlino, Antonello*; Messori, Luigi | |
Reactions of Auranofin and Its Pseudohalide Derivatives with Serum Albumin Investigated through ESI-Q-TOF MS | 2018 | Alessandro Pratesi, Damiano Cirri, Lorenzo Ciofi, Luigi Messori | |
Chlorido and bromido oxaliplatin analogues as potential agents for CRC treatment: Solution behavior, protein binding and cytotoxicity evaluation | 2018 | Marzo, Tiziano; Pratesi, Alessandro; Cirri, Damiano; Pillozzi, Serena; Petroni, Giulia; Guerri, Annalisa; Arcangeli, Annarosa; Messori, Luigi; Gabbiani, Chiara | |
A Fluorescent Silver(I) Carbene Complex with Anticancer Properties: Synthesis, Characterization, and Biological Studies | 2019 | Maria Giulia Fabbrini, Damiano Cirri, Alessandro Pratesi, Lorenzo Ciofi, Tiziano Marzo, Annalisa Guerri, Silvia Nistri, Alfonso Dell'Accio, Tania Gamberi, Mirko Severi, Andrea Bencini, Luigi messori | |
Structural Characterization of a Gold/Serum Albumin Complex | 2019 | Pratesi, Alessandro; Cirri, Damiano; Fregona, Dolores; Ferraro, Giarita; Giorgio, Anna; Merlino, Antonello; Messori, Luigi | |
The cisplatin/serum albumin system: A reappraisal | 2019 | Massai, Lara; Pratesi, Alessandro; Gailer, Jurgen; Marzo, Tiziano; Messori, Luigi | |
The leading established metal-based drugs: a revisitation of their relevant physico-chemical data | 2019 | Damiano Cirri, Maria Giulia Fabbrini, Alessandro Pratesi, Lorenzo Ciofi, Lara Massai, Tiziano Marzo, Luigi Messori | |
Replacement of the Thiosugar of Auranofin with Iodide Enhances the Anticancer Potency in a Mouse Model of Ovarian Cancer | 2019 | Tiziano Marzo, Lara Massai, Alessandro Pratesi, Matteo Stefanini, Damiano Cirri, Francesca Magherini, Matteo Becatti, Ida Landini, Stefania Nobili, Enrico Mini, Olivia Crociani, Annarosa Arcangeli, Serena Pillozzi, Tania Gamberi, Luigi Messori | |
ESI MS studies highlight the selective interaction of Auranofin with protein free thiols | 2020 | Zoppi C.; Messori L.; Pratesi A. | |
Native mass spectrometry of human carbonic anhydrase I and its inhibitor complexes | 2020 | Zoppi C.; Nocentini A.; Supuran C.T.; Pratesi A.; Messori L. | |
Computationally enhanced X-ray diffraction analysis of a gold(III) complex interacting with the human telomeric DNA G-quadruplex. Unravelling non-unique ligand positioning | 2022 | Cirri, Damiano; Bazzicalupi, Carla; Ryde, Ulf; Bergmann, Justin; Binacchi, Francesca; Nocentini, Alessio; Pratesi, Alessandro; Gratteri, Paola; Messori, Luigi |
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