Sfoglia per Autore
MODELING AND STRUCTURE-BASED APPROACHES IN THE DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF LIGANDS TARGETING THE METALLOENZYMES CARBONIC ANHYDRASES
2018 Alessio Nocentini
Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms
2018 Nocentini, Alessio; Bonardi, Alessandro; Gratteri, Paola; Cerra, Bruno; Gioiello, Antimo*; Supuran, Claudiu T.
Discovery of β-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy
2018 Nocentini, Alessio; Ceruso, Mariangela; Bua, Silvia; Lomelino, Carrie L.; Andring, Jacob T.; McKenna, Robert; Lanzi, Cecilia; Sgambellone, Silvia; Pecori, Riccardo; Matucci, Rosanna; Filippi, Luca; Gratteri, Paola; Carta, Fabrizio; Masini, Emanuela; Selleri, Silvia*; Supuran, Claudiu T.
Benzoxaborole compounds for therapeutic uses: a patent review (2010- 2018)
2018 Nocentini, Alessio; Supuran, Claudiu T; Winum, Jean-Yves
2-Benzylpiperazine: a new scaffold for potent human Carbonic Anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents.
2018 Niccolò Chiaramonte, Silvia Bua, Marta Ferraroni, Alessio Nocentini, Alessandro Bonardi, Gian Luca Bartolucci, Maria Concetta Durante, Laura Lucarini, Donata Chiapponi, Silvia Dei, Dina Manetti, Elisabetta Teodori, Paola Gratteri, Emanuela Masini, Claudiu T. Supuran, Maria Novella Romanelli
4-Hydroxy-3-nitro-5-ureido-benzenesulfonamides selectively target the tumor-associated carbonic anhydrase isoforms IX and XII showing hypoxia-enhanced anti-proliferative profiles.
2018 Nocentini A, Trallori E, Singh S, Lomelino CL, Bartolucci G, Di Cesare Mannelli L, Ghelardini C, McKenna R, Gratteri P, Supuran CT
Synthesis, biological evaluation and computational studies of novel iminothiazolidinone benzenesulfonamides as potent carbonic anhydrase II and IX inhibitors
2018 Mahmood, Shams-ul; Saeed, Aamer*; Bua, Sivia; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T.
Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform
2018 Ibrahim, Hany S.*; Allam, Heba Abdelrasheed; Mahmoud, Walaa R.; Bonardi, Alessandro; Nocentini, Alessio; Gratteri, Paola; Ibrahim, Eslam S.; Abdel-Aziz, Hatem A.; Supuran, Claudiu T.
Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails
2018 Awadallah, Fadi M.; Bua, Silvia; Mahmoud, Walaa R.; Nada, Hossam H.; Nocentini, Alessio; Supuran, Claudiu T.*
Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies
2018 Nocentini, Alessio; Carta, Fabrizio; Tanc, Muhammet; Selleri, Silvia; Supuran, Claudiu T.; Bazzicalupi, Carla*; Gratteri, Paola
Use of Innovative (Micro)Extraction Techniques to Characterise Harpagophytum procumbens Root and its Commercial Food Supplements
2018 Diuzheva, Alina; Carradori, Simone; Andruch, Vasil; Locatelli, Marcello; Luca, Elisa De; Tiecco, Matteo; Germani, Raimondo; Menghini, Luigi; Nocentini, Alessio; Gratteri, Paola; Campestre, Cristina
Novel hydrazido benzenesulfonamides-isatin conjugates: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies
2018 Mahmoud F. Abo-Ashour; Wagdy M. Eldehna; Alessio Nocentini; Hany S. Ibrahim; Silvia Bua; Sahar M. Abou-Seri; Claudiu T. Supuran
Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer
2018 Eldehna, Wagdy M; Nocentini, Alessio; Al-Rashood, Sara T; Hassan, Ghada S; Alkahtani, Hamad M; Almehizia, Abdulrahman A; Reda, Ahmed M; Abdel-Aziz, Hatem A; Supuran, Claudiu T
Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy
2018 Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Salvadori, Severo; Onnis, Valentina; Supuran, Claudiu T
Carbonic anhydrase inhibition with a series of novel benzenesulfonamide-triazole conjugates
2018 El-Gazzar, Marwa G; Nafie, Nessma H; Nocentini, Alessio; Ghorab, Mostafa M; Heiba, Helmi I; Supuran, Claudiu T
Evaluation of 99mTc-sulfonamide and sulfocoumarin derivatives for imaging carbonic anhydrase IX expression
2018 Nakai, Misaki; Pan, Jihne; Lin, Kuo-Shyan; Thompson, John R; Nocentini, Alessio; Supuran, Claudiu T; Nakabayashi, Yasuo; Storr, Tim
Synthesis of novel isoindoline-1,3-dione-based oximes and benzenesulfonamide hydrazones as selective inhibitors of the tumor-associated carbonic anhydrase IX
2018 Abdel-Aziz, Alaa A-M; El-Azab, Adel S; Abu El-Enin, Mohamed A; Almehizia, Abdulrahman A; Supuran, Claudiu T; Nocentini, Alessio
Carbonic anhydrase inhibitors as antitumor/antimetastatic agents: a patent review (2008-2018)
2018 Nocentini, Alessio; Supuran, Claudiu T
Natural Polyphenols Selectively Inhibit β-Carbonic Anhydrase from the Dandruff-Producing Fungus Malassezia globosa: Activity and Modeling Studies
2018 Nocentini, Alessio; Bua, Silvia; Del Prete, Sonia; Heravi, Yeganeh Entezari; Saboury, Ali A; Karioti, Anastasia; Bilia, Anna Rita; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T
Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors
2018 Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Onnis, Valentina; Supuran, Claudiu T
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| MODELING AND STRUCTURE-BASED APPROACHES IN THE DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF LIGANDS TARGETING THE METALLOENZYMES CARBONIC ANHYDRASES | 2018 | Alessio Nocentini | |
| Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms | 2018 | Nocentini, Alessio; Bonardi, Alessandro; Gratteri, Paola; Cerra, Bruno; Gioiello, Antimo*; Supuran, Claudiu T. | |
| Discovery of β-Adrenergic Receptors Blocker-Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy | 2018 | Nocentini, Alessio; Ceruso, Mariangela; Bua, Silvia; Lomelino, Carrie L.; Andring, Jacob T.; McKenna, Robert; Lanzi, Cecilia; Sgambellone, Silvia; Pecori, Riccardo; Matucci, Rosanna; Filippi, Luca; Gratteri, Paola; Carta, Fabrizio; Masini, Emanuela; Selleri, Silvia*; Supuran, Claudiu T. | |
| Benzoxaborole compounds for therapeutic uses: a patent review (2010- 2018) | 2018 | Nocentini, Alessio; Supuran, Claudiu T; Winum, Jean-Yves | |
| 2-Benzylpiperazine: a new scaffold for potent human Carbonic Anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents. | 2018 | Niccolò Chiaramonte, Silvia Bua, Marta Ferraroni, Alessio Nocentini, Alessandro Bonardi, Gian Luca Bartolucci, Maria Concetta Durante, Laura Lucarini, Donata Chiapponi, Silvia Dei, Dina Manetti, Elisabetta Teodori, Paola Gratteri, Emanuela Masini, Claudiu T. Supuran, Maria Novella Romanelli | |
| 4-Hydroxy-3-nitro-5-ureido-benzenesulfonamides selectively target the tumor-associated carbonic anhydrase isoforms IX and XII showing hypoxia-enhanced anti-proliferative profiles. | 2018 | Nocentini A, Trallori E, Singh S, Lomelino CL, Bartolucci G, Di Cesare Mannelli L, Ghelardini C, McKenna R, Gratteri P, Supuran CT | |
| Synthesis, biological evaluation and computational studies of novel iminothiazolidinone benzenesulfonamides as potent carbonic anhydrase II and IX inhibitors | 2018 | Mahmood, Shams-ul; Saeed, Aamer*; Bua, Sivia; Nocentini, Alessio; Gratteri, Paola; Supuran, Claudiu T. | |
| Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform | 2018 | Ibrahim, Hany S.*; Allam, Heba Abdelrasheed; Mahmoud, Walaa R.; Bonardi, Alessandro; Nocentini, Alessio; Gratteri, Paola; Ibrahim, Eslam S.; Abdel-Aziz, Hatem A.; Supuran, Claudiu T. | |
| Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails | 2018 | Awadallah, Fadi M.; Bua, Silvia; Mahmoud, Walaa R.; Nada, Hossam H.; Nocentini, Alessio; Supuran, Claudiu T.* | |
| Deciphering the Mechanism of Human Carbonic Anhydrases Inhibition with Sulfocoumarins: Computational and Experimental Studies | 2018 | Nocentini, Alessio; Carta, Fabrizio; Tanc, Muhammet; Selleri, Silvia; Supuran, Claudiu T.; Bazzicalupi, Carla*; Gratteri, Paola | |
| Use of Innovative (Micro)Extraction Techniques to Characterise Harpagophytum procumbens Root and its Commercial Food Supplements | 2018 | Diuzheva, Alina; Carradori, Simone; Andruch, Vasil; Locatelli, Marcello; Luca, Elisa De; Tiecco, Matteo; Germani, Raimondo; Menghini, Luigi; Nocentini, Alessio; Gratteri, Paola; Campestre, Cristina | |
| Novel hydrazido benzenesulfonamides-isatin conjugates: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies | 2018 | Mahmoud F. Abo-Ashour; Wagdy M. Eldehna; Alessio Nocentini; Hany S. Ibrahim; Silvia Bua; Sahar M. Abou-Seri; Claudiu T. Supuran | |
| Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer | 2018 | Eldehna, Wagdy M; Nocentini, Alessio; Al-Rashood, Sara T; Hassan, Ghada S; Alkahtani, Hamad M; Almehizia, Abdulrahman A; Reda, Ahmed M; Abdel-Aziz, Hatem A; Supuran, Claudiu T | |
| Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy | 2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Salvadori, Severo; Onnis, Valentina; Supuran, Claudiu T | |
| Carbonic anhydrase inhibition with a series of novel benzenesulfonamide-triazole conjugates | 2018 | El-Gazzar, Marwa G; Nafie, Nessma H; Nocentini, Alessio; Ghorab, Mostafa M; Heiba, Helmi I; Supuran, Claudiu T | |
| Evaluation of 99mTc-sulfonamide and sulfocoumarin derivatives for imaging carbonic anhydrase IX expression | 2018 | Nakai, Misaki; Pan, Jihne; Lin, Kuo-Shyan; Thompson, John R; Nocentini, Alessio; Supuran, Claudiu T; Nakabayashi, Yasuo; Storr, Tim | |
| Synthesis of novel isoindoline-1,3-dione-based oximes and benzenesulfonamide hydrazones as selective inhibitors of the tumor-associated carbonic anhydrase IX | 2018 | Abdel-Aziz, Alaa A-M; El-Azab, Adel S; Abu El-Enin, Mohamed A; Almehizia, Abdulrahman A; Supuran, Claudiu T; Nocentini, Alessio | |
| Carbonic anhydrase inhibitors as antitumor/antimetastatic agents: a patent review (2008-2018) | 2018 | Nocentini, Alessio; Supuran, Claudiu T | |
| Natural Polyphenols Selectively Inhibit β-Carbonic Anhydrase from the Dandruff-Producing Fungus Malassezia globosa: Activity and Modeling Studies | 2018 | Nocentini, Alessio; Bua, Silvia; Del Prete, Sonia; Heravi, Yeganeh Entezari; Saboury, Ali A; Karioti, Anastasia; Bilia, Anna Rita; Capasso, Clemente; Gratteri, Paola; Supuran, Claudiu T | |
| Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors | 2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Onnis, Valentina; Supuran, Claudiu T |
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