RENZI, GIOELE
RENZI, GIOELE
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity
2024 Hakan Aslan; Gioele Renzi; Andrea Angeli; Ilaria D'Agostino; Roberto Ronca; Maria Luisa Massardi; Camilla Tavani; Simone Carradori; Marta Ferraroni; Paolo Governa; Fabrizio Manetti; Fabrizio Carta; Claudiu T. Supuran
Design, Synthesis, and In Vitro Evaluation of Aromatic Sulfonamides as Human Carbonic Anhydrase I, II, IX, and XII Inhibitors and Their Antioxidant Activity
2025 Abha Mishra K.M.; Kumari N.; Carta F.; Renzi G.; Supuran C.T.; Sethi K.K.
Dual inhibition of carbonic anhydrases VA and VII by silychristin and isosilybin A from Silybum marianum: A potential antiobesity strategy
2025 Emanuele Liborio Citriniti; Roberta Rocca; Giosuè Costa; Gioele Renzi; Fabrizio Carta; Claudiu T. Supuran; Stefano Alcaro; Francesco Ortuso
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms
2024 Kilbile, JT; Sapkal, SB; Renzi, G; D'Agostino, I; Boudjelal, M; Tamboli, Y; Cutarella, L; Mori, M; Sgambellone, S; Villano, S; Marri, S; Lucarini, L; Carradori, S; Carta, F; Supuran, CT
Lasamide, a Potent Human Carbonic Anhydrase Inhibitor from the Market: Inhibition Profiling and Crystallographic Studies
2024 Baroni C.; D'Agostino I.; Renzi G.; Kilbile J.T.; Tamboli Y.; Ferraroni M.; Carradori S.; Capasso C.; Carta F.; Supuran C.T.
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors
2024 Kilbile J.T.; Sapkal S.B.; Renzi G.; D'Agostino I.; Cutarella L.; Mori M.; De Filippis B.; Islam I.; Massardi M.L.; Somenza E.; Ronca R.; Tamboli Y.; Carta F.; Supuran C.T.
Preliminary Investigations on Acyl Hydrazones Bearing Sulfonamides as Inhibitors of the Human Carbonic Anhydrase Isoforms I, II, IX, and XII
2025 Efe Doğukan Dincel; Ebru Didem Kuran; Abdulilah Ece; Faika Başoğlu-Ünal; Gioele Renzi; Gloria Badii; Fabrizio Carta; Claudiu T. Supuran; Nuray Ulusoy-Güzeldemirci
The carbonic anhydrase enzymes as new targets for the management of neglected tropical diseases
2024 Gioele Renzi; Federico Ladu; Fabrizio Carta; Claudiu T. Supuran
The Integrase: An Overview of a Key Player Enzyme in the Antiviral Scenario
2023 Gioele Renzi; Fabrizio Carta; Claudiu T. Supuran
Thia- and Seleno-Michael Reactions for the Synthesis of Carbonic Anhydrases Inhibitors
2024 Angeli A.; Occhini A.; Renzi G.; Capperucci A.; Ferraroni M.; Tanini D.; Supuran C.T.
X-ray crystallographic and kinetic studies of biguanide containing aryl sulfonamides as carbonic anhydrase inhibitors
2025 Chiara Baroni; Murat Bozdag; Gioele Renzi; Viviana De Luca; Clemente Capasso; Carla Bazzicalupi; Silvia Selleri; Marta Ferraroni; Fabrizio Carta; Claudiu T. Supuran
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity | 2024 | Hakan Aslan; Gioele Renzi; Andrea Angeli; Ilaria D'Agostino; Roberto Ronca; Maria Luisa Massardi; Camilla Tavani; Simone Carradori; Marta Ferraroni; Paolo Governa; Fabrizio Manetti; Fabrizio Carta; Claudiu T. Supuran | |
Design, Synthesis, and In Vitro Evaluation of Aromatic Sulfonamides as Human Carbonic Anhydrase I, II, IX, and XII Inhibitors and Their Antioxidant Activity | 2025 | Abha Mishra K.M.; Kumari N.; Carta F.; Renzi G.; Supuran C.T.; Sethi K.K. | |
Dual inhibition of carbonic anhydrases VA and VII by silychristin and isosilybin A from Silybum marianum: A potential antiobesity strategy | 2025 | Emanuele Liborio Citriniti; Roberta Rocca; Giosuè Costa; Gioele Renzi; Fabrizio Carta; Claudiu T. Supuran; Stefano Alcaro; Francesco Ortuso | |
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms | 2024 | Kilbile, JT; Sapkal, SB; Renzi, G; D'Agostino, I; Boudjelal, M; Tamboli, Y; Cutarella, L; Mori, M; Sgambellone, S; Villano, S; Marri, S; Lucarini, L; Carradori, S; Carta, F; Supuran, CT | |
Lasamide, a Potent Human Carbonic Anhydrase Inhibitor from the Market: Inhibition Profiling and Crystallographic Studies | 2024 | Baroni C.; D'Agostino I.; Renzi G.; Kilbile J.T.; Tamboli Y.; Ferraroni M.; Carradori S.; Capasso C.; Carta F.; Supuran C.T. | |
Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors | 2024 | Kilbile J.T.; Sapkal S.B.; Renzi G.; D'Agostino I.; Cutarella L.; Mori M.; De Filippis B.; Islam I.; Massardi M.L.; Somenza E.; Ronca R.; Tamboli Y.; Carta F.; Supuran C.T. | |
Preliminary Investigations on Acyl Hydrazones Bearing Sulfonamides as Inhibitors of the Human Carbonic Anhydrase Isoforms I, II, IX, and XII | 2025 | Efe Doğukan Dincel; Ebru Didem Kuran; Abdulilah Ece; Faika Başoğlu-Ünal; Gioele Renzi; Gloria Badii; Fabrizio Carta; Claudiu T. Supuran; Nuray Ulusoy-Güzeldemirci | |
The carbonic anhydrase enzymes as new targets for the management of neglected tropical diseases | 2024 | Gioele Renzi; Federico Ladu; Fabrizio Carta; Claudiu T. Supuran | |
The Integrase: An Overview of a Key Player Enzyme in the Antiviral Scenario | 2023 | Gioele Renzi; Fabrizio Carta; Claudiu T. Supuran | |
Thia- and Seleno-Michael Reactions for the Synthesis of Carbonic Anhydrases Inhibitors | 2024 | Angeli A.; Occhini A.; Renzi G.; Capperucci A.; Ferraroni M.; Tanini D.; Supuran C.T. | |
X-ray crystallographic and kinetic studies of biguanide containing aryl sulfonamides as carbonic anhydrase inhibitors | 2025 | Chiara Baroni; Murat Bozdag; Gioele Renzi; Viviana De Luca; Clemente Capasso; Carla Bazzicalupi; Silvia Selleri; Marta Ferraroni; Fabrizio Carta; Claudiu T. Supuran |