GUERRINI, GABRIELLA
GUERRINI, GABRIELLA
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulators
2021 Crocetti, Letizia; Guerrini, Gabriella; Cantini, Niccolò; Vergelli, Claudia; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors
2021 Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria
1H-pyrrolo[2,3-b]pyridine: a new scaffold for human neutrophil elastase (HNE) inhibitors
2018 Letizia Crocetti, Maria Paola Giovannoni, Igor A. Schepetkinb, Mark T. Quinn, Andrei I. Khlebnikovc, Niccolò Cantini, Gabriella Guerrini, Antonella Iacovone, Elisabetta Teodori, Claudia Vergelli
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists.
2016 Vergelli, C; Schepetkin, I.A; Ciciani, G; Cilibrizzi, A; Crocetti, L; Giovannoni, M.P; Guerrini, G; Iacovone, A; Kirpotina, L.N; Khlebnikov, A.I; Ye, R.D; Quinn, M.T.
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective Peripheral Benzodiazepine Receptor ligands
2001 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; B. COSTA; C. MARTINI
3,8-Disubstituted Pyrazolo[1,5-a]quinazoline as GABAA Receptor Modulators: Synthesis, Electrophysiological Assays, and Molecular Modelling Studies
2024 Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola
4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor Subtype
2023 Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola
8H-PYRAZOLO[5',1':2,3]PYRIMIDO[5,4-D][1,2]DIAZEPINE. A NEW TRICYCLIC SYSTEM.
1993 F. BRUNI; B. COSIMELLI; A. COSTANZO; G. GUERRINI; S. SELLERI
A combined crystallographic and computational study on dexketoprofen trometamol dihydrate salt
2020 Rossi P.; Paoli P.; Milazzo S.; Chelazzi L.; Giovannoni M.P.; Guerrini G.; Ienco A.; Valleri M.; Conti L.
A new class of pyrazolo[5,1-c][1,2,4]triazines as γ-aminobutyric type A (GABAA) receptor subtype ligand: synthesis and pharmacological evaluation
2018 Gabriella Guerrini, Giovanna Ciciani, Simona Daniele, Claudia Martini, Camilla Costagli, Chiara Guarino, Silvia Selleri
A New Entry to Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine Derivatives
1990 F.BRUNI; S. CHIMICHI; B.COSIMELLI; A.COSTANZO; G.GUERRINI; S.SELLERI
A novel selective GABA-A alpha1 receptor agonist displaying sedative and anxiolytic-like properties in rodents.
2005 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. GRATTERI; F. BESNARD; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; M. MONTALI; J. FOHLIN
Anti-Inflammatory Activity of Pyrazolo[1,5-a]quinazolines
2024 Crocetti, Letizia; Khlebnikov, Andrei I.; Guerrini, Gabriella; Schepetkin, Igor A.; Melani, Fabrizio; Giovannoni, Maria Paola; Quinn, Mark T.
Antiproliferative and antimicrobial activities of pyrazolo[5,1-c][1,2,4]benzotriazines 5-oxides and their 5-deoxyderivatives.
1999 F. BRUNI; S. SELLERI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. LA COLLA; R. DONATO; C. SACCO; C. MUSIU; C. MILIA; S. LONGU; C. MINNEI
BENZODIAZEPINE RECEPTOR (BZR) LIGANDS.5. NEW 3-ALKYLOXYCARBONYL-, 3-CYCLOALKYLOXYCARBONYL-,3-ARYLOXYCARBONYLDERIVATIVES OF PYRAZOLO [5,1-C][1,2,4]BENZOTRIAZINE 5-OXIDES: A STUDY ON THE 3-ESTER FUNCTION MODIFICATION
1999 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG; A. IPPONI; A. LUCACCHINI
Benzodiazepine receptor ligands. 4.Synthesis, and pharmacological evaluation of 3-hetroaryl-8-chloro pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides.
1999 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; S. SELLERI; B. COSTA; C. MARTINI; A. LUCACCHINI; P. MALMBERG AIELLO; A. IPPONI
Benzodiazepine receptor ligands. 6. New 3-(2-,3- or 4-substituted benzyloxycarbonyl) derivatives of 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide receptor affinity and In vivo testing C. Martini, P. Malmberg Aiello
2001 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; C. COSTAGLI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG AIELLO
BENZODIAZEPINE RECEPTOR LIGANDS. 7. SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF NEW 3-ESTERS OF THE 8-CHLOROPYRAZOLO[5,1-C][1,2,4]BENZOTRIAZINE 5-OXIDE. 3-(2- THIENYLMETHOXYCARBONYL) DERIVATIVE: AN ANXIOSELECTIVE AGENT IN RODENTS.
2002 F. BRUNI; P. MALMBERG; A. COSTANZO; G. CICIANI; G. GUERRINI; S. SELLERI; C. COSTAGLI; C. MARTINI; B. COSTA; F. BESNARD
Benzodiazepine receptor ligands. 8. Synthesis and pharamcological evaluation of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide 3- and 8-disubstituted: high affinity ligands endowed with inverse-agonist pharmacological efficacy.
2006 G. GUERRINI; A. COSTANZO; G. CICIANI; F. BRUNI; S. SELLERI; C. COSTAGLI; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; F. BESNARD
BENZODIAZEPINE RECEPTOR LIGANDS. PART II. SYNTHESIS AND BIOLOGICAL EVALUATION OF PYRAZOLO[5,1-C][1,2,4]BENZOTRIAZINES 4-OXIDE.
1998 F. BRUNI; A. COSTANZO; G. CICIANI; G. GUERRINI; S. SELLERI; C. MARTINI; A. LUCACCHINI; B. COSTA; S. CAPPELLETTI
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulators | 2021 | Crocetti, Letizia; Guerrini, Gabriella; Cantini, Niccolò; Vergelli, Claudia; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola | |
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors | 2021 | Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria | |
1H-pyrrolo[2,3-b]pyridine: a new scaffold for human neutrophil elastase (HNE) inhibitors | 2018 | Letizia Crocetti, Maria Paola Giovannoni, Igor A. Schepetkinb, Mark T. Quinn, Andrei I. Khlebnikovc, Niccolò Cantini, Gabriella Guerrini, Antonella Iacovone, Elisabetta Teodori, Claudia Vergelli | |
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists. | 2016 | Vergelli, C; Schepetkin, I.A; Ciciani, G; Cilibrizzi, A; Crocetti, L; Giovannoni, M.P; Guerrini, G; Iacovone, A; Kirpotina, L.N; Khlebnikov, A.I; Ye, R.D; Quinn, M.T. | |
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective Peripheral Benzodiazepine Receptor ligands | 2001 | S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; B. COSTA; C. MARTINI | |
3,8-Disubstituted Pyrazolo[1,5-a]quinazoline as GABAA Receptor Modulators: Synthesis, Electrophysiological Assays, and Molecular Modelling Studies | 2024 | Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola | |
4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor Subtype | 2023 | Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola | |
8H-PYRAZOLO[5',1':2,3]PYRIMIDO[5,4-D][1,2]DIAZEPINE. A NEW TRICYCLIC SYSTEM. | 1993 | F. BRUNI; B. COSIMELLI; A. COSTANZO; G. GUERRINI; S. SELLERI | |
A combined crystallographic and computational study on dexketoprofen trometamol dihydrate salt | 2020 | Rossi P.; Paoli P.; Milazzo S.; Chelazzi L.; Giovannoni M.P.; Guerrini G.; Ienco A.; Valleri M.; Conti L. | |
A new class of pyrazolo[5,1-c][1,2,4]triazines as γ-aminobutyric type A (GABAA) receptor subtype ligand: synthesis and pharmacological evaluation | 2018 | Gabriella Guerrini, Giovanna Ciciani, Simona Daniele, Claudia Martini, Camilla Costagli, Chiara Guarino, Silvia Selleri | |
A New Entry to Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine Derivatives | 1990 | F.BRUNI; S. CHIMICHI; B.COSIMELLI; A.COSTANZO; G.GUERRINI; S.SELLERI | |
A novel selective GABA-A alpha1 receptor agonist displaying sedative and anxiolytic-like properties in rodents. | 2005 | S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. GRATTERI; F. BESNARD; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; M. MONTALI; J. FOHLIN | |
Anti-Inflammatory Activity of Pyrazolo[1,5-a]quinazolines | 2024 | Crocetti, Letizia; Khlebnikov, Andrei I.; Guerrini, Gabriella; Schepetkin, Igor A.; Melani, Fabrizio; Giovannoni, Maria Paola; Quinn, Mark T. | |
Antiproliferative and antimicrobial activities of pyrazolo[5,1-c][1,2,4]benzotriazines 5-oxides and their 5-deoxyderivatives. | 1999 | F. BRUNI; S. SELLERI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. LA COLLA; R. DONATO; C. SACCO; C. MUSIU; C. MILIA; S. LONGU; C. MINNEI | |
BENZODIAZEPINE RECEPTOR (BZR) LIGANDS.5. NEW 3-ALKYLOXYCARBONYL-, 3-CYCLOALKYLOXYCARBONYL-,3-ARYLOXYCARBONYLDERIVATIVES OF PYRAZOLO [5,1-C][1,2,4]BENZOTRIAZINE 5-OXIDES: A STUDY ON THE 3-ESTER FUNCTION MODIFICATION | 1999 | A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG; A. IPPONI; A. LUCACCHINI | |
Benzodiazepine receptor ligands. 4.Synthesis, and pharmacological evaluation of 3-hetroaryl-8-chloro pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides. | 1999 | A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; S. SELLERI; B. COSTA; C. MARTINI; A. LUCACCHINI; P. MALMBERG AIELLO; A. IPPONI | |
Benzodiazepine receptor ligands. 6. New 3-(2-,3- or 4-substituted benzyloxycarbonyl) derivatives of 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide receptor affinity and In vivo testing C. Martini, P. Malmberg Aiello | 2001 | A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; C. COSTAGLI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG AIELLO | |
BENZODIAZEPINE RECEPTOR LIGANDS. 7. SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF NEW 3-ESTERS OF THE 8-CHLOROPYRAZOLO[5,1-C][1,2,4]BENZOTRIAZINE 5-OXIDE. 3-(2- THIENYLMETHOXYCARBONYL) DERIVATIVE: AN ANXIOSELECTIVE AGENT IN RODENTS. | 2002 | F. BRUNI; P. MALMBERG; A. COSTANZO; G. CICIANI; G. GUERRINI; S. SELLERI; C. COSTAGLI; C. MARTINI; B. COSTA; F. BESNARD | |
Benzodiazepine receptor ligands. 8. Synthesis and pharamcological evaluation of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide 3- and 8-disubstituted: high affinity ligands endowed with inverse-agonist pharmacological efficacy. | 2006 | G. GUERRINI; A. COSTANZO; G. CICIANI; F. BRUNI; S. SELLERI; C. COSTAGLI; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; F. BESNARD | |
BENZODIAZEPINE RECEPTOR LIGANDS. PART II. SYNTHESIS AND BIOLOGICAL EVALUATION OF PYRAZOLO[5,1-C][1,2,4]BENZOTRIAZINES 4-OXIDE. | 1998 | F. BRUNI; A. COSTANZO; G. CICIANI; G. GUERRINI; S. SELLERI; C. MARTINI; A. LUCACCHINI; B. COSTA; S. CAPPELLETTI |