GUERRINI, GABRIELLA

GUERRINI, GABRIELLA  

Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)  

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Risultati 1 - 20 di 85 (tempo di esecuzione: 0.031 secondi).
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'Proximity frequencies' a new parameter to evaluate the profile of GABAAR modulators 2021 Crocetti, Letizia; Guerrini, Gabriella; Cantini, Niccolò; Vergelli, Claudia; Melani, Fabrizio; Mascia, Maria Paola; Giovannoni, Maria Paola
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitors 2021 Cantini, Niccolo; Crocetti, Letizia; Guerrini, Gabriella; Vergelli, Claudia; Schepetkin, Igor A; Pallecchi, Marco; Bartolucci, Gian Luca; Quinn, Mark T; Teodori, Elisabetta; Paola Giovannoni, Maria
1H-pyrrolo[2,3-b]pyridine: a new scaffold for human neutrophil elastase (HNE) inhibitors 2018 Letizia Crocetti, Maria Paola Giovannoni, Igor A. Schepetkinb, Mark T. Quinn, Andrei I. Khlebnikovc, Niccolò Cantini, Gabriella Guerrini, Antonella Iacovone, Elisabetta Teodori, Claudia Vergelli
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists. 2016 Vergelli, C; Schepetkin, I.A; Ciciani, G; Cilibrizzi, A; Crocetti, L; Giovannoni, M.P; Guerrini, G; Iacovone, A; Kirpotina, L.N; Khlebnikov, A.I; Ye, R.D; Quinn, M.T.
2-Arylpyrazolo[1,5-a]pyrimidin-3-yl acetamides. New potent and selective Peripheral Benzodiazepine Receptor ligands 2001 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; B. COSTA; C. MARTINI
4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABAA Receptor Subtype 2023 Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola
8H-PYRAZOLO[5',1':2,3]PYRIMIDO[5,4-D][1,2]DIAZEPINE. A NEW TRICYCLIC SYSTEM. 1993 F. BRUNI; B. COSIMELLI; A. COSTANZO; G. GUERRINI; S. SELLERI
A combined crystallographic and computational study on dexketoprofen trometamol dihydrate salt 2020 Rossi P.; Paoli P.; Milazzo S.; Chelazzi L.; Giovannoni M.P.; Guerrini G.; Ienco A.; Valleri M.; Conti L.
A new class of pyrazolo[5,1-c][1,2,4]triazines as γ-aminobutyric type A (GABAA) receptor subtype ligand: synthesis and pharmacological evaluation 2018 Gabriella Guerrini, Giovanna Ciciani, Simona Daniele, Claudia Martini, Camilla Costagli, Chiara Guarino, Silvia Selleri
A New Entry to Pyrazolo[1,5-a]pyrido[3,4-e]pyrimidine Derivatives 1990 F.BRUNI; S. CHIMICHI; B.COSIMELLI; A.COSTANZO; G.GUERRINI; S.SELLERI
A novel selective GABA-A alpha1 receptor agonist displaying sedative and anxiolytic-like properties in rodents. 2005 S. SELLERI; F. BRUNI; C. COSTAGLI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. GRATTERI; F. BESNARD; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; M. MONTALI; J. FOHLIN
Antiproliferative and antimicrobial activities of pyrazolo[5,1-c][1,2,4]benzotriazines 5-oxides and their 5-deoxyderivatives. 1999 F. BRUNI; S. SELLERI; A. COSTANZO; G. GUERRINI; G. CICIANI; P. LA COLLA; R. DONATO; C. SACCO; C. MUSIU; C. MILIA; S. LONGU; C. MINNEI
BENZODIAZEPINE RECEPTOR (BZR) LIGANDS.5. NEW 3-ALKYLOXYCARBONYL-, 3-CYCLOALKYLOXYCARBONYL-,3-ARYLOXYCARBONYLDERIVATIVES OF PYRAZOLO [5,1-C][1,2,4]BENZOTRIAZINE 5-OXIDES: A STUDY ON THE 3-ESTER FUNCTION MODIFICATION 1999 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG; A. IPPONI; A. LUCACCHINI
Benzodiazepine receptor ligands. 4.Synthesis, and pharmacological evaluation of 3-hetroaryl-8-chloro pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides. 1999 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; S. SELLERI; B. COSTA; C. MARTINI; A. LUCACCHINI; P. MALMBERG AIELLO; A. IPPONI
Benzodiazepine receptor ligands. 6. New 3-(2-,3- or 4-substituted benzyloxycarbonyl) derivatives of 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide receptor affinity and In vivo testing C. Martini, P. Malmberg Aiello 2001 A. COSTANZO; G. GUERRINI; G. CICIANI; F. BRUNI; C. COSTAGLI; S. SELLERI; B. COSTA; C. MARTINI; P. MALMBERG AIELLO
BENZODIAZEPINE RECEPTOR LIGANDS. 7. SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF NEW 3-ESTERS OF THE 8-CHLOROPYRAZOLO[5,1-C][1,2,4]BENZOTRIAZINE 5-OXIDE. 3-(2- THIENYLMETHOXYCARBONYL) DERIVATIVE: AN ANXIOSELECTIVE AGENT IN RODENTS. 2002 F. BRUNI; P. MALMBERG; A. COSTANZO; G. CICIANI; G. GUERRINI; S. SELLERI; C. COSTAGLI; C. MARTINI; B. COSTA; F. BESNARD
Benzodiazepine receptor ligands. 8. Synthesis and pharamcological evaluation of new pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide 3- and 8-disubstituted: high affinity ligands endowed with inverse-agonist pharmacological efficacy. 2006 G. GUERRINI; A. COSTANZO; G. CICIANI; F. BRUNI; S. SELLERI; C. COSTAGLI; B. COSTA; C. MARTINI; G. DE SIENA; P. MALMBERG; F. BESNARD
BENZODIAZEPINE RECEPTOR LIGANDS. PART II. SYNTHESIS AND BIOLOGICAL EVALUATION OF PYRAZOLO[5,1-C][1,2,4]BENZOTRIAZINES 4-OXIDE. 1998 F. BRUNI; A. COSTANZO; G. CICIANI; G. GUERRINI; S. SELLERI; C. MARTINI; A. LUCACCHINI; B. COSTA; S. CAPPELLETTI
Benzodiazepine receptor ligands. Part III. Synthesis and biological evaluation of 2 and/or 3-substituted pyrazolo[5,1-c][1,2,4] benzotriazine 5-oxides. 1999 G. GUERRINI; A. COSTANZO; F. BRUNI; G. CICIANI; S. SELLERI; P. GRATTERI; B. COSTA; C. MARTINI; A. LUCACCHINI
BENZODIAZEPINE RECEPTOR LIGANDS. SYNTHESIS AND PHARMACOLOGICAL EVALUATION OF 3-, 7- AND 8-SUBSTITUTED [5,1-C][1,2,4]BENZOTRIAZINES AND 5-OXIDE DERIVATIVES. PART I. 1996 G. GUERRINI; A. COSTANZO; F. BRUNI; S. SELLERI; L. GIUSTI; A. LUCACCHINI; C. MARTINI