ANGELI, ANDREA
ANGELI, ANDREA
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy
2020 Kaproń, Barbara; Czarnomysy, Robert; Wysokiński, Mariusz; Andrys, Rudolf; Musilek, Kamil; Angeli, Andrea; Supuran, Claudiu T; Plech, Tomasz
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
2020 D'Ascenzio M.; Secci D.; Carradori S.; Zara S.; Guglielmi P.; Cirilli R.; Pierini M.; Poli G.; Tuccinardi T.; Angeli A.; Supuran C.T.
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity
2022 Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N.
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site
2020 Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V.
3-Functionalised benzenesulphonamide based 1,3,4-oxadiazoles as selective carbonic anhydrase XIII inhibitors: Design, synthesis and biological evaluation
2021 Swain B.; Abhay; Singh P.; Angeli A.; Aashritha K.; Nagesh N.; Supuran C.T.; Arifuddin M.
3-Hydroxy-1H-quinazoline-2,4-dione as a New Scaffold to Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII
2017 Falsini, Matteo; Squarcialupi, Lucia; Catarzi, Daniela; Varano, Flavia; Betti, Marco; Di Cesare Mannelli, Lorenzo; Tenci, Barbara; Ghelardini, Carla; Tanc, Muhammet; Angeli, Andrea; Supuran, Claudiu T.; Colotta, Vittoria
4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies
2022 Nada H.; Elkamhawy A.; Abdellattif M.H.; Angeli A.; Lee C.H.; Supuran C.T.; Lee K.
4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae
2021 Mancuso F.; De Luca L.; Bucolo F.; Vrabel M.; Angeli A.; Capasso C.; Supuran C.T.; Gitto R.
A novel small molecule that kills a subset of MLL-rearranged leukemia cells by inducing mitochondrial dysfunction
2019 Somers K.; Wen V.W.; Middlemiss S.M.C.; Osborne B.; Forgham H.; Jung M.S.; Karsa M.; Clifton M.; Bongers A.; Gao J.; Mayoh C.; Raoufi-Rad N.; Kusnadi E.P.; Hannan K.M.; Scott D.A.; Kwek A.; Liu B.; Flemming C.; Chudakova D.A.; Pandher R.; Failes T.W.; Lim J.; Angeli A.; Osterman A.L.; Imamura T.; Kees U.R.; Supuran C.T.; Pearson R.B.; Hannan R.D.; Davis T.P.; McCarroll J.; Kavallaris M.; Turner N.; Gudkov A.V.; Haber M.; Norris M.D.; Henderson M.J.
A structure-based approach towards the identification of novel antichagasic compounds: Trypanosoma cruzi carbonic anhydrase inhibitors
2020 Llanos M.A.; Sbaraglini M.L.; Villalba M.L.; Ruiz M.D.; Carrillo C.; Soto C.A.; Talevi A.; Angeli A.; Parkkila S.; Supuran C.T.; Gavernet L.
Activation Effects of Carnosine- and Histidine-Containing Dipeptides on Human Carbonic Anhydrases: A Comprehensive Study
2020 Vistoli, Giulio; Aldini, Giancarlo; Fumagalli, Laura; Dallanoce, Clelia; Angeli, Andrea; Supuran, Claudiu T.
Activation of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with amines and amino acids
2021 Angeli A.; Urbanski L.J.; Hytonen V.P.; Parkkila S.; Supuran C.T.
Activation of β- and γ-carbonic anhydrases from pathogenic bacteria with tripeptides
2018 Stefanucci A.; Angeli A.; Dimmito M.P.; Luisi G.; Del Prete S.; Capasso C.; Donald W.A.; Mollica A.; Supuran C.T.
Activation studies of the α- and β-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with amines and amino acids
2018 Angeli, Andrea; Del Prete, Sonia; Osman, Sameh M; Alasmary, Fatmah A S; Alothman, Zeid; Donald, William A; Capasso, Clemente; Supuran, Claudiu T
Activation studies of the β-carbonic anhydrases from Malassezia restricta with amines and amino acids
2020 Angeli A.; Prete S.D.; Ghobril C.; Hitce J.; Clavaud C.; Marrat X.; Donald W.A.; Capasso C.; Supuran C.T.
Activation studies of the γ-carbonic anhydrases from the antarctic marine bacteria pseudoalteromonas haloplanktis and colwellia psychrerythraea with amino acids and amines
2019 Angeli A.; Del Prete S.; Osman S.M.; AlOthman Z.; Donald W.A.; Capasso C.; Supuran C.T.
Activation studies with amines and amino acids of the α-carbonic anhydrase from the pathogenic protozoan Trypanosoma cruzi
2018 Angeli A.; Kuuslahti M.; Parkkila S.; Supuran C.T.
Activation studies with amines and amino acids of the β-carbonic anhydrase encoded by the Rv3273 gene from the pathogenic bacterium Mycobacterium tuberculosis
2018 Angeli, Andrea; Del Prete, Sonia; Osman, Sameh M; Alasmary, Fatmah A S; Alothman, Zeid; Donald, William A; Capasso, Clemente; Supuran, Claudiu T
Activation studies with amines and amino acids of the β-carbonic anhydrase from the pathogenic protozoan Leishmania donovani chagasi
2018 Angeli, Andrea; Donald, William A.; Parkkila, Seppo; Supuran, Claudiu T.
Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic anhydrase
2022 Angeli, Andrea; Urbański, Linda J; Capasso, Clemente; Parkkila, Seppo; Supuran, Claudiu T
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy | 2020 | Kaproń, Barbara; Czarnomysy, Robert; Wysokiński, Mariusz; Andrys, Rudolf; Musilek, Kamil; Angeli, Andrea; Supuran, Claudiu T; Plech, Tomasz | |
| 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors | 2020 | D'Ascenzio M.; Secci D.; Carradori S.; Zara S.; Guglielmi P.; Cirilli R.; Pierini M.; Poli G.; Tuccinardi T.; Angeli A.; Supuran C.T. | |
| 2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity | 2022 | Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N. | |
| 2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site | 2020 | Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V. | |
| 3-Functionalised benzenesulphonamide based 1,3,4-oxadiazoles as selective carbonic anhydrase XIII inhibitors: Design, synthesis and biological evaluation | 2021 | Swain B.; Abhay; Singh P.; Angeli A.; Aashritha K.; Nagesh N.; Supuran C.T.; Arifuddin M. | |
| 3-Hydroxy-1H-quinazoline-2,4-dione as a New Scaffold to Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII | 2017 | Falsini, Matteo; Squarcialupi, Lucia; Catarzi, Daniela; Varano, Flavia; Betti, Marco; Di Cesare Mannelli, Lorenzo; Tenci, Barbara; Ghelardini, Carla; Tanc, Muhammet; Angeli, Andrea; Supuran, Claudiu T.; Colotta, Vittoria | |
| 4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies | 2022 | Nada H.; Elkamhawy A.; Abdellattif M.H.; Angeli A.; Lee C.H.; Supuran C.T.; Lee K. | |
| 4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae | 2021 | Mancuso F.; De Luca L.; Bucolo F.; Vrabel M.; Angeli A.; Capasso C.; Supuran C.T.; Gitto R. | |
| A novel small molecule that kills a subset of MLL-rearranged leukemia cells by inducing mitochondrial dysfunction | 2019 | Somers K.; Wen V.W.; Middlemiss S.M.C.; Osborne B.; Forgham H.; Jung M.S.; Karsa M.; Clifton M.; Bongers A.; Gao J.; Mayoh C.; Raoufi-Rad N.; Kusnadi E.P.; Hannan K.M.; Scott D.A.; Kwek A.; Liu B.; Flemming C.; Chudakova D.A.; Pandher R.; Failes T.W.; Lim J.; Angeli A.; Osterman A.L.; Imamura T.; Kees U.R.; Supuran C.T.; Pearson R.B.; Hannan R.D.; Davis T.P.; McCarroll J.; Kavallaris M.; Turner N.; Gudkov A.V.; Haber M.; Norris M.D.; Henderson M.J. | |
| A structure-based approach towards the identification of novel antichagasic compounds: Trypanosoma cruzi carbonic anhydrase inhibitors | 2020 | Llanos M.A.; Sbaraglini M.L.; Villalba M.L.; Ruiz M.D.; Carrillo C.; Soto C.A.; Talevi A.; Angeli A.; Parkkila S.; Supuran C.T.; Gavernet L. | |
| Activation Effects of Carnosine- and Histidine-Containing Dipeptides on Human Carbonic Anhydrases: A Comprehensive Study | 2020 | Vistoli, Giulio; Aldini, Giancarlo; Fumagalli, Laura; Dallanoce, Clelia; Angeli, Andrea; Supuran, Claudiu T. | |
| Activation of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with amines and amino acids | 2021 | Angeli A.; Urbanski L.J.; Hytonen V.P.; Parkkila S.; Supuran C.T. | |
| Activation of β- and γ-carbonic anhydrases from pathogenic bacteria with tripeptides | 2018 | Stefanucci A.; Angeli A.; Dimmito M.P.; Luisi G.; Del Prete S.; Capasso C.; Donald W.A.; Mollica A.; Supuran C.T. | |
| Activation studies of the α- and β-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with amines and amino acids | 2018 | Angeli, Andrea; Del Prete, Sonia; Osman, Sameh M; Alasmary, Fatmah A S; Alothman, Zeid; Donald, William A; Capasso, Clemente; Supuran, Claudiu T | |
| Activation studies of the β-carbonic anhydrases from Malassezia restricta with amines and amino acids | 2020 | Angeli A.; Prete S.D.; Ghobril C.; Hitce J.; Clavaud C.; Marrat X.; Donald W.A.; Capasso C.; Supuran C.T. | |
| Activation studies of the γ-carbonic anhydrases from the antarctic marine bacteria pseudoalteromonas haloplanktis and colwellia psychrerythraea with amino acids and amines | 2019 | Angeli A.; Del Prete S.; Osman S.M.; AlOthman Z.; Donald W.A.; Capasso C.; Supuran C.T. | |
| Activation studies with amines and amino acids of the α-carbonic anhydrase from the pathogenic protozoan Trypanosoma cruzi | 2018 | Angeli A.; Kuuslahti M.; Parkkila S.; Supuran C.T. | |
| Activation studies with amines and amino acids of the β-carbonic anhydrase encoded by the Rv3273 gene from the pathogenic bacterium Mycobacterium tuberculosis | 2018 | Angeli, Andrea; Del Prete, Sonia; Osman, Sameh M; Alasmary, Fatmah A S; Alothman, Zeid; Donald, William A; Capasso, Clemente; Supuran, Claudiu T | |
| Activation studies with amines and amino acids of the β-carbonic anhydrase from the pathogenic protozoan Leishmania donovani chagasi | 2018 | Angeli, Andrea; Donald, William A.; Parkkila, Seppo; Supuran, Claudiu T. | |
| Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic anhydrase | 2022 | Angeli, Andrea; Urbański, Linda J; Capasso, Clemente; Parkkila, Seppo; Supuran, Claudiu T |