GIOVANNUZZI, SIMONE
GIOVANNUZZI, SIMONE
Neuroscienze, Area del Farmaco e Salute del Bambino (NEUROFARBA)
4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors
2022 Abdoli, Morteza; Giovannuzzi, Simone; Supuran, Claudiu T; Žalubovskis, Raivis
Aromatic sulfonamides including a sulfonic acid tail: New membrane impermeant carbonic anhydrase inhibitors for targeting selectively the cancer‐associated isoforms
2022 Giovannuzzi S.; D'ambrosio M.; Luceri C.; Osman S.M.; Pallecchi M.; Bartolucci G.; Nocentini A.; Supuran C.T.
Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII
2022 Giovannuzzi, Simone; Capasso, Clemente; Nocentini, Alessio; Supuran, Claudiu T
Coumarins effectively inhibit bacterial α-carbonic anhydrases
2022 Giovannuzzi S.; Hewitt C.S.; Nocentini A.; Capasso C.; Flaherty D.P.; Supuran C.T.
Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum
2022 Giovannuzzi S.; De Luca V.; Nocentini A.; Capasso C.; Supuran C.T.
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors
2023 Giovannuzzi, Simone; Bonardi, Alessandro; Gratteri, Paola; Nocentini, Alessio; Supuran, Claudiu T
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae
2022 Giovannuzzi S.; Abutaleb N.S.; Hewitt C.S.; Carta F.; Nocentini A.; Seleem M.N.; Flaherty D.P.; Supuran C.T.
Elaborating 5-(4-chlorophenyl)-1,3,4-thiadiazole scaffold with a p-tolyl sulfonamide moiety enhances cytotoxic activity: Design, synthesis, in vitro cytotoxicity evaluation, radiolabelling, and in vivo pharmacokinetic study
2022 El-Masry, Rana; Shaarawy, Sahar; Kadry, Hanan; Shalaby, Azza; Supuran, Claudiu; Giovannuzzi, Simone; sakr, tamer; Amin, Mohamed; Korani, Mohamed
Inhibition studies of bacterial α-carbonic anhydrases with phenols
2022 Giovannuzzi S.; Hewitt C.S.; Nocentini A.; Capasso C.; Costantino G.; Flaherty D.P.; Supuran C.T.
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ
2023 Giovannuzzi, Simone; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T
May Sulfonamide Inhibitors of Carbonic Anhydrases from Mammaliicoccus sciuri Prevent Antimicrobial Resistance Due to Gene Transfer to Other Harmful Staphylococci?
2022 De Luca, Viviana; Giovannuzzi, Simone; Supuran, Claudiu T; Capasso, Clemente
Pyrrolyl and Indolyl alpha-gamma-Diketo Acid Derivatives Acting as Selective Inhibitors of Human Carbonic Anhydrases IX and XII
2023 Ialongo, D; Messore, A; Madia, VN; Tudino, V; Nocentini, A; Gratteri, P; Giovannuzzi, S; Supuran, CT; Nicolai, A; Scarpa, S; Taurone, S; Camarda, M; Artico, M; Papa, V; Saccoliti, F; Scipione, L; Di Santo, R; Costi, R
Sulfonamides linked to sulfonate esters via hydrazone functionality: synthesis, human carbonic anhydrase inhibitory activities, and molecular modeling studies
2023 Han, MI; Gunduz, MG; Alci, G; Giovannuzzi, S; Yuvali, D; Supuran, CT; Dogan, SD