GIOVANNUZZI, SIMONE
GIOVANNUZZI, SIMONE
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
1,5-Diaryl-1,2,4-triazole Ureas as New SLC-0111 Analogues Endowed with Dual Carbonic Anhydrase and VEGFR-2 Inhibitory Activities
2023 Elsawi, Ahmed E.; Elbadawi, Mostafa M.; Nocentini, Alessio; Almahli, Hadia; Giovannuzzi, Simone; Shaldam, Moataz; Salem, Rofaida; Ibrahim, Tamer M.; Abdel-Aziz, Hatem A.; Supuran, Claudiu T.; Eldehna, Wagdy M.
4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors
2022 Abdoli, Morteza; Giovannuzzi, Simone; Supuran, Claudiu T; Žalubovskis, Raivis
Aromatic sulfonamides including a sulfonic acid tail: New membrane impermeant carbonic anhydrase inhibitors for targeting selectively the cancer‐associated isoforms
2022 Giovannuzzi S.; D'ambrosio M.; Luceri C.; Osman S.M.; Pallecchi M.; Bartolucci G.; Nocentini A.; Supuran C.T.
Benzoxaborinine, New Chemotype for Carbonic Anhydrase Inhibition: Ex Novo Synthesis, Crystallography, In Silico Studies, and Anti-Melanoma Cell Line Activity
2024 Giovannuzzi S.; Nikitjuka A.; Angeli A.; Smietana M.; Massardi M.-L.; Turati M.; Ronca R.; Bonardi A.; Nocentini A.; Ferraroni M.; Supuran C.T.; Winum J.-Y.
Boron-containing carbonic anhydrases inhibitors
2024 Giovannuzzi, Simone; Nikitjuka, Anna; Pereira Resende, Bruna Rafaela; Smietana, Michael; Nocentini, Alessio; Supuran, Claudiu T.; Winum, Jean-Yves
Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors
2023 Martínez-Montiel, Mónica; Romero-Hernández, Laura L; Giovannuzzi, Simone; Begines, Paloma; Puerta, Adrián; Ahuja-Casarín, Ana I; Fernandes, Miguel X; Merino-Montiel, Penélope; Montiel-Smith, Sara; Nocentini, Alessio; Padrón, José M; Supuran, Claudiu T; Fernández-Bolaños, José G; López, Óscar
Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII
2022 Giovannuzzi, Simone; Capasso, Clemente; Nocentini, Alessio; Supuran, Claudiu T
Coumarins effectively inhibit bacterial α-carbonic anhydrases
2022 Giovannuzzi S.; Hewitt C.S.; Nocentini A.; Capasso C.; Flaherty D.P.; Supuran C.T.
Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum
2022 Giovannuzzi S.; De Luca V.; Nocentini A.; Capasso C.; Supuran C.T.
Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies
2023 Begines, Paloma; Bonardi, Alessandro; Nocentini, Alessio; Gratteri, Paola; Giovannuzzi, Simone; Ronca, Roberto; Tavani, Camilla; Luisa Massardi, Maria; López, Óscar; Supuran, Claudiu T
Discovery of indolinone-bearing benzenesulfonamides as new dual carbonic anhydrase and VEGFR-2 inhibitors possessing anticancer and pro-apoptotic properties
2023 Saied, Samaa; Shaldam, Moataz; Elbadawi, Mostafa M.; Giovannuzzi, Simone; Nocentini, Alessio; Almahli, Hadia; Salem, Rofaida; Ibrahim, Tamer M.; Supuran, Claudiu T.; Eldehna, Wagdy M.
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors
2023 Giovannuzzi, Simone; Bonardi, Alessandro; Gratteri, Paola; Nocentini, Alessio; Supuran, Claudiu T
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae
2022 Giovannuzzi S.; Abutaleb N.S.; Hewitt C.S.; Carta F.; Nocentini A.; Seleem M.N.; Flaherty D.P.; Supuran C.T.
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction
2024 Giovannuzzi, Simone; Chavarria, Daniel; Provensi, Gustavo; Leri, Manuela; Bucciantini, Monica; Carradori, Simone; Bonardi, Alessandro; Gratteri, Paola; Borges, Fernanda; Nocentini, Alessio; Supuran, Claudiu T.
Elaborating 5-(4-chlorophenyl)-1,3,4-thiadiazole scaffold with a p-tolyl sulfonamide moiety enhances cytotoxic activity: Design, synthesis, in vitro cytotoxicity evaluation, radiolabelling, and in vivo pharmacokinetic study
2022 El-Masry, Rana; Shaarawy, Sahar; Kadry, Hanan; Shalaby, Azza; Supuran, Claudiu; Giovannuzzi, Simone; sakr, tamer; Amin, Mohamed; Korani, Mohamed
Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases
2024 Nocentini A.; Costa A.; Bonardi A.; Ammara A.; Giovannuzzi S.; Petreni A.; Bartolucci G.; Rani B.; Leri M.; Bucciantini M.; Fernandez-Bolanos J.G.; Lopez O.; Passani M.B.; Provensi G.; Gratteri P.; Supuran C.T.
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates
2023 Giovannuzzi, Simone; Marapaka, Anil Kumar; Abutaleb, Nader S.; Carta, Fabrizio; Liang, Hsin-Wen; Nocentini, Alessio; Pisano, Luigi; Seleem, Mohamed N.; Flaherty, Daniel P.; Supuran, Claudiu T.
Inhibition studies of bacterial α-carbonic anhydrases with phenols
2022 Giovannuzzi S.; Hewitt C.S.; Nocentini A.; Capasso C.; Costantino G.; Flaherty D.P.; Supuran C.T.
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ
2023 Giovannuzzi, Simone; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T
May Sulfonamide Inhibitors of Carbonic Anhydrases from Mammaliicoccus sciuri Prevent Antimicrobial Resistance Due to Gene Transfer to Other Harmful Staphylococci?
2022 De Luca, Viviana; Giovannuzzi, Simone; Supuran, Claudiu T; Capasso, Clemente
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1,5-Diaryl-1,2,4-triazole Ureas as New SLC-0111 Analogues Endowed with Dual Carbonic Anhydrase and VEGFR-2 Inhibitory Activities | 2023 | Elsawi, Ahmed E.; Elbadawi, Mostafa M.; Nocentini, Alessio; Almahli, Hadia; Giovannuzzi, Simone; Shaldam, Moataz; Salem, Rofaida; Ibrahim, Tamer M.; Abdel-Aziz, Hatem A.; Supuran, Claudiu T.; Eldehna, Wagdy M. | |
4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors | 2022 | Abdoli, Morteza; Giovannuzzi, Simone; Supuran, Claudiu T; Žalubovskis, Raivis | |
Aromatic sulfonamides including a sulfonic acid tail: New membrane impermeant carbonic anhydrase inhibitors for targeting selectively the cancer‐associated isoforms | 2022 | Giovannuzzi S.; D'ambrosio M.; Luceri C.; Osman S.M.; Pallecchi M.; Bartolucci G.; Nocentini A.; Supuran C.T. | |
Benzoxaborinine, New Chemotype for Carbonic Anhydrase Inhibition: Ex Novo Synthesis, Crystallography, In Silico Studies, and Anti-Melanoma Cell Line Activity | 2024 | Giovannuzzi S.; Nikitjuka A.; Angeli A.; Smietana M.; Massardi M.-L.; Turati M.; Ronca R.; Bonardi A.; Nocentini A.; Ferraroni M.; Supuran C.T.; Winum J.-Y. | |
Boron-containing carbonic anhydrases inhibitors | 2024 | Giovannuzzi, Simone; Nikitjuka, Anna; Pereira Resende, Bruna Rafaela; Smietana, Michael; Nocentini, Alessio; Supuran, Claudiu T.; Winum, Jean-Yves | |
Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors | 2023 | Martínez-Montiel, Mónica; Romero-Hernández, Laura L; Giovannuzzi, Simone; Begines, Paloma; Puerta, Adrián; Ahuja-Casarín, Ana I; Fernandes, Miguel X; Merino-Montiel, Penélope; Montiel-Smith, Sara; Nocentini, Alessio; Padrón, José M; Supuran, Claudiu T; Fernández-Bolaños, José G; López, Óscar | |
Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII | 2022 | Giovannuzzi, Simone; Capasso, Clemente; Nocentini, Alessio; Supuran, Claudiu T | |
Coumarins effectively inhibit bacterial α-carbonic anhydrases | 2022 | Giovannuzzi S.; Hewitt C.S.; Nocentini A.; Capasso C.; Flaherty D.P.; Supuran C.T. | |
Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum | 2022 | Giovannuzzi S.; De Luca V.; Nocentini A.; Capasso C.; Supuran C.T. | |
Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies | 2023 | Begines, Paloma; Bonardi, Alessandro; Nocentini, Alessio; Gratteri, Paola; Giovannuzzi, Simone; Ronca, Roberto; Tavani, Camilla; Luisa Massardi, Maria; López, Óscar; Supuran, Claudiu T | |
Discovery of indolinone-bearing benzenesulfonamides as new dual carbonic anhydrase and VEGFR-2 inhibitors possessing anticancer and pro-apoptotic properties | 2023 | Saied, Samaa; Shaldam, Moataz; Elbadawi, Mostafa M.; Giovannuzzi, Simone; Nocentini, Alessio; Almahli, Hadia; Salem, Rofaida; Ibrahim, Tamer M.; Supuran, Claudiu T.; Eldehna, Wagdy M. | |
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors | 2023 | Giovannuzzi, Simone; Bonardi, Alessandro; Gratteri, Paola; Nocentini, Alessio; Supuran, Claudiu T | |
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae | 2022 | Giovannuzzi S.; Abutaleb N.S.; Hewitt C.S.; Carta F.; Nocentini A.; Seleem M.N.; Flaherty D.P.; Supuran C.T. | |
Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction | 2024 | Giovannuzzi, Simone; Chavarria, Daniel; Provensi, Gustavo; Leri, Manuela; Bucciantini, Monica; Carradori, Simone; Bonardi, Alessandro; Gratteri, Paola; Borges, Fernanda; Nocentini, Alessio; Supuran, Claudiu T. | |
Elaborating 5-(4-chlorophenyl)-1,3,4-thiadiazole scaffold with a p-tolyl sulfonamide moiety enhances cytotoxic activity: Design, synthesis, in vitro cytotoxicity evaluation, radiolabelling, and in vivo pharmacokinetic study | 2022 | El-Masry, Rana; Shaarawy, Sahar; Kadry, Hanan; Shalaby, Azza; Supuran, Claudiu; Giovannuzzi, Simone; sakr, tamer; Amin, Mohamed; Korani, Mohamed | |
Enhanced Recognition Memory through Dual Modulation of Brain Carbonic Anhydrases and Cholinesterases | 2024 | Nocentini A.; Costa A.; Bonardi A.; Ammara A.; Giovannuzzi S.; Petreni A.; Bartolucci G.; Rani B.; Leri M.; Bucciantini M.; Fernandez-Bolanos J.G.; Lopez O.; Passani M.B.; Provensi G.; Gratteri P.; Supuran C.T. | |
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates | 2023 | Giovannuzzi, Simone; Marapaka, Anil Kumar; Abutaleb, Nader S.; Carta, Fabrizio; Liang, Hsin-Wen; Nocentini, Alessio; Pisano, Luigi; Seleem, Mohamed N.; Flaherty, Daniel P.; Supuran, Claudiu T. | |
Inhibition studies of bacterial α-carbonic anhydrases with phenols | 2022 | Giovannuzzi S.; Hewitt C.S.; Nocentini A.; Capasso C.; Costantino G.; Flaherty D.P.; Supuran C.T. | |
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ | 2023 | Giovannuzzi, Simone; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T | |
May Sulfonamide Inhibitors of Carbonic Anhydrases from Mammaliicoccus sciuri Prevent Antimicrobial Resistance Due to Gene Transfer to Other Harmful Staphylococci? | 2022 | De Luca, Viviana; Giovannuzzi, Simone; Supuran, Claudiu T; Capasso, Clemente |