BRACONI, LAURA

BRACONI, LAURA  

Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)  

Mostra records
Risultati 1 - 20 di 26 (tempo di esecuzione: 0.041 secondi).
Titolo Data di pubblicazione Autore(i) File
1-benzyl-1,4-diazepane reduces the efflux of resistance-nodulation-cell division pumps in Escherichia coli 2020 Enrico Casalone, Tiziano Vignolini, Laura Braconi, Lucia Gardini, Marco Capitanio, Francesco S Pavone, Silvia Dei, Elisabetta Teodori
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity 2022 Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N.
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers 2020 Braconi L.; Bartolucci G.; Contino M.; Chiaramonte N.; Giampietro R.; Manetti D.; Perrone M.G.; Romanelli M.N.; Colabufo N.A.; Riganti C.; Dei S.; Teodori E.
Application of LEDA algorithm for the recognition of P-glycoprotein and Carbonic Anhydrase hybrid inhibitors and evaluation of their plasma stability by HPLC-MS/MS analysis 2022 Pallecchi, Marco; Menicatti, Marta; Braconi, Laura; Supuran, Claudiu T; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca
Characterization of substituted piperazines able to reverse MDR in Escherichia coli strains overexpressing resistance-nodulation-cell division (RND) efflux pumps 2022 Casalone E.; Vignolini T.; Braconi L.; Gardini L.; Capitanio M.; Pavone F.S.; Giovannelli L.; Dei S.; Teodori E.
Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers 2019 Braconi L., Bartolucci G., Manetti D., Romanelli M.N., Dei S., Teodori E.
Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers 2019 Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Braconi L.; Manetti D.; Romanelli M.N.; Trezza A.; Athanasios A.; Spiga O.; Perrone M.G.; Giampietro R.; Gazzano E.; Salerno M.; Colabufo N.A.; Dei S.
Design, synthesis and characterization of new molecules which counteract drug resistance mechanisms 2022 Laura Braconi
Drug plasma stability study of multidrug resistance inhibitors by LC-MS/MS analysis 2018 Marta Menicatti, Matilde Maggini, Francesco Caponi, Donato Squillaci, Laura Braconi, Silvia Dei , Elisabetta Teodori, Gian Luca Bartolucci
Dual P-glycoprotein and CA XII inhibitors: A new strategy to reverse the P-gp Mediated Multidrug Resistance (MDR) in cancer cells y 2020 Teodori E.; Braconi L.; Bua S.; Lapucci A.; Bartolucci G.; Manetti D.; Romanelli M.N.; Dei S.; Supuran C.T.; Coronnello M.
ERMS EXPERIMENTS FOR RESOLUTION OF ISOBARIC COMPOUNDS: A CASE OF CIS/TRANS ISOMERISM 2018 Laura Braconi; Marta Menicatti; Silvia Dei; Elisabetta Teodori; Gian Luca Bartolucci
Isomers Recognition in HPLC-MS/MS Analysis of Human Plasma Samples by Using an Ion Trap Supported by a Linear Equations-Based Algorithm 2023 Pallecchi M.; Lucio L.; Braconi L.; Menicatti M.; Dei S.; Teodori E.; Bartolucci G.
Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug-resistance (MDR) modulators 2019 Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Marcella Coronnello, Niccolò Chiaramonte, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Chatchanok Udomtanakunchai, Nicola Antonio Colabufo, Gian luca Bartolucci, Ottavia Spiga, Milena Salerno, Elisabetta Teodori
New dual P-Glycoprotein (P-gp) and human carbonic anhydrase XII (hCA XII) inhibitors as Multidrug Resistance (MDR) reversers in cancer cells 2022 Braconi, Laura; Teodori, Elisabetta; Riganti, Chiara; Coronnello, Marcella; Nocentini, Alessio; Bartolucci, Gian Luca; Pallecchi, Marco; Contino, Marialessandra; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T; Dei, Silvia
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators 2022 Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N.
Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives 2022 Braconi L.; Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Manetti D.; Romanelli M.N.; Perrone M.G.; Colabufo N.A.; Guglielmo S.; Dei S.
P-glycoprotein and carbonic anhydrases hybrid inhibitors: a new strategy to reverse multidrug resistance (MDR) in cancer cells 2018 E. Teodori, M. Coronnello, S. Bua, L. Braconi, D. Manetti, M.N. Romanelli, C. Supuran, S. Dei
Recent advances in the discovery of Nicotinic acetylcholine receptor allosteric modulators 2023 Dina Manetti , Silvia Dei, Hugo R. Arias, Laura Braconi, Alessio Gabellini, Elisabetta Teodori, Maria Romanelli
Recent advances in the search of BCRP- and dual P-gp/BCRP-based multidrug resistance modulators 2019 Silvia Dei, Laura Braconi, Maria Novella Romanelli, Elisabetta Teodori
Simultaneous Degradation Study of Isomers in Human Plasma by HPLC-MS/MS and Application of LEDA Algorithm for Their Characterization 2022 Pallecchi, Marco; Braconi, Laura; Menicatti, Marta; Giachetti, Sara; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca