BRACONI, LAURA
BRACONI, LAURA
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
1-benzyl-1,4-diazepane reduces the efflux of resistance-nodulation-cell division pumps in Escherichia coli
2020 Enrico Casalone, Tiziano Vignolini, Laura Braconi, Lucia Gardini, Marco Capitanio, Francesco S Pavone, Silvia Dei, Elisabetta Teodori
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity
2022 Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N.
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers
2020 Braconi L.; Bartolucci G.; Contino M.; Chiaramonte N.; Giampietro R.; Manetti D.; Perrone M.G.; Romanelli M.N.; Colabufo N.A.; Riganti C.; Dei S.; Teodori E.
Application of LEDA Algorithm for the characterization of Isomers in Simultaneous Degradation Study in Human Plasma by HPLC-MS/MS
2023 M. Pallecchi; L. Braconi; M. Menicatti; S. Giachetti; S. Dei; E. Teodori; Gian Luca Bartolucci
Application of LEDA algorithm for the recognition of P-glycoprotein and Carbonic Anhydrase hybrid inhibitors and evaluation of their plasma stability by HPLC-MS/MS analysis
2022 Pallecchi, Marco; Menicatti, Marta; Braconi, Laura; Supuran, Claudiu T; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca
Characterization of substituted piperazines able to reverse MDR in Escherichia coli strains overexpressing resistance-nodulation-cell division (RND) efflux pumps
2022 Casalone E.; Vignolini T.; Braconi L.; Gardini L.; Capitanio M.; Pavone F.S.; Giovannelli L.; Dei S.; Teodori E.
Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers
2019 Braconi L., Bartolucci G., Manetti D., Romanelli M.N., Dei S., Teodori E.
Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers
2019 Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Braconi L.; Manetti D.; Romanelli M.N.; Trezza A.; Athanasios A.; Spiga O.; Perrone M.G.; Giampietro R.; Gazzano E.; Salerno M.; Colabufo N.A.; Dei S.
Design, synthesis and characterization of new molecules which counteract drug resistance mechanisms
2022 Laura Braconi
Drug plasma stability study of multidrug resistance inhibitors by LC-MS/MS analysis
2018 Marta Menicatti, Matilde Maggini, Francesco Caponi, Donato Squillaci, Laura Braconi, Silvia Dei , Elisabetta Teodori, Gian Luca Bartolucci
Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold
2024 Braconi L.; Riganti C.; Parenti A.; Cecchi M.; Nocentini A.; Bartolucci G.; Menicatti M.; Contino M.; Colabufo N.A.; Manetti D.; Romanelli M.N.; Supuran C.T.; Teodori E.
Dual P-glycoprotein and CA XII inhibitors: A new strategy to reverse the P-gp Mediated Multidrug Resistance (MDR) in cancer cells y
2020 Teodori E.; Braconi L.; Bua S.; Lapucci A.; Bartolucci G.; Manetti D.; Romanelli M.N.; Dei S.; Supuran C.T.; Coronnello M.
ERMS EXPERIMENTS FOR RESOLUTION OF ISOBARIC COMPOUNDS: A CASE OF CIS/TRANS ISOMERISM
2018 Laura Braconi; Marta Menicatti; Silvia Dei; Elisabetta Teodori; Gian Luca Bartolucci
Isomers Recognition in HPLC-MS/MS Analysis of Human Plasma Samples by Using an Ion Trap Supported by a Linear Equations-Based Algorithm
2023 Pallecchi M.; Lucio L.; Braconi L.; Menicatti M.; Dei S.; Teodori E.; Bartolucci G.
Mass Spectrometry Study about In Vitro and In Vivo Reaction between Metformin and Glucose: A Preliminary Investigation on Alternative Biological Behavior
2024 Bartolucci, Gian Luca; Pallecchi, Marco; Braconi, Laura; Dei, Silvia; Teodori, Elisabetta; Lapolla, Annunziata; Sartore, Giovanni; Traldi, Pietro
Metformin reacts directly with glucose following the Maillard reaction pathway
2023 M. Pallecchi; G. Bartolucci; L. Braconi; S. Dei; E. Teodori; A. Lapolla; G. Sartore; P. Traldi;
Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug-resistance (MDR) modulators
2019 Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Marcella Coronnello, Niccolò Chiaramonte, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Chatchanok Udomtanakunchai, Nicola Antonio Colabufo, Gian luca Bartolucci, Ottavia Spiga, Milena Salerno, Elisabetta Teodori
New dual P-Glycoprotein (P-gp) and human carbonic anhydrase XII (hCA XII) inhibitors as Multidrug Resistance (MDR) reversers in cancer cells
2022 Braconi, Laura; Teodori, Elisabetta; Riganti, Chiara; Coronnello, Marcella; Nocentini, Alessio; Bartolucci, Gian Luca; Pallecchi, Marco; Contino, Marialessandra; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T; Dei, Silvia
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators
2022 Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N.
Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives
2022 Braconi L.; Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Manetti D.; Romanelli M.N.; Perrone M.G.; Colabufo N.A.; Guglielmo S.; Dei S.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1-benzyl-1,4-diazepane reduces the efflux of resistance-nodulation-cell division pumps in Escherichia coli | 2020 | Enrico Casalone, Tiziano Vignolini, Laura Braconi, Lucia Gardini, Marco Capitanio, Francesco S Pavone, Silvia Dei, Elisabetta Teodori | |
| 2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity | 2022 | Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N. | |
| 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers | 2020 | Braconi L.; Bartolucci G.; Contino M.; Chiaramonte N.; Giampietro R.; Manetti D.; Perrone M.G.; Romanelli M.N.; Colabufo N.A.; Riganti C.; Dei S.; Teodori E. | |
| Application of LEDA Algorithm for the characterization of Isomers in Simultaneous Degradation Study in Human Plasma by HPLC-MS/MS | 2023 | M. Pallecchi; L. Braconi; M. Menicatti; S. Giachetti; S. Dei; E. Teodori; Gian Luca Bartolucci | |
| Application of LEDA algorithm for the recognition of P-glycoprotein and Carbonic Anhydrase hybrid inhibitors and evaluation of their plasma stability by HPLC-MS/MS analysis | 2022 | Pallecchi, Marco; Menicatti, Marta; Braconi, Laura; Supuran, Claudiu T; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca | |
| Characterization of substituted piperazines able to reverse MDR in Escherichia coli strains overexpressing resistance-nodulation-cell division (RND) efflux pumps | 2022 | Casalone E.; Vignolini T.; Braconi L.; Gardini L.; Capitanio M.; Pavone F.S.; Giovannelli L.; Dei S.; Teodori E. | |
| Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers | 2019 | Braconi L., Bartolucci G., Manetti D., Romanelli M.N., Dei S., Teodori E. | |
| Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers | 2019 | Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Braconi L.; Manetti D.; Romanelli M.N.; Trezza A.; Athanasios A.; Spiga O.; Perrone M.G.; Giampietro R.; Gazzano E.; Salerno M.; Colabufo N.A.; Dei S. | |
| Design, synthesis and characterization of new molecules which counteract drug resistance mechanisms | 2022 | Laura Braconi | |
| Drug plasma stability study of multidrug resistance inhibitors by LC-MS/MS analysis | 2018 | Marta Menicatti, Matilde Maggini, Francesco Caponi, Donato Squillaci, Laura Braconi, Silvia Dei , Elisabetta Teodori, Gian Luca Bartolucci | |
| Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold | 2024 | Braconi L.; Riganti C.; Parenti A.; Cecchi M.; Nocentini A.; Bartolucci G.; Menicatti M.; Contino M.; Colabufo N.A.; Manetti D.; Romanelli M.N.; Supuran C.T.; Teodori E. | |
| Dual P-glycoprotein and CA XII inhibitors: A new strategy to reverse the P-gp Mediated Multidrug Resistance (MDR) in cancer cells y | 2020 | Teodori E.; Braconi L.; Bua S.; Lapucci A.; Bartolucci G.; Manetti D.; Romanelli M.N.; Dei S.; Supuran C.T.; Coronnello M. | |
| ERMS EXPERIMENTS FOR RESOLUTION OF ISOBARIC COMPOUNDS: A CASE OF CIS/TRANS ISOMERISM | 2018 | Laura Braconi; Marta Menicatti; Silvia Dei; Elisabetta Teodori; Gian Luca Bartolucci | |
| Isomers Recognition in HPLC-MS/MS Analysis of Human Plasma Samples by Using an Ion Trap Supported by a Linear Equations-Based Algorithm | 2023 | Pallecchi M.; Lucio L.; Braconi L.; Menicatti M.; Dei S.; Teodori E.; Bartolucci G. | |
| Mass Spectrometry Study about In Vitro and In Vivo Reaction between Metformin and Glucose: A Preliminary Investigation on Alternative Biological Behavior | 2024 | Bartolucci, Gian Luca; Pallecchi, Marco; Braconi, Laura; Dei, Silvia; Teodori, Elisabetta; Lapolla, Annunziata; Sartore, Giovanni; Traldi, Pietro | |
| Metformin reacts directly with glucose following the Maillard reaction pathway | 2023 | M. Pallecchi; G. Bartolucci; L. Braconi; S. Dei; E. Teodori; A. Lapolla; G. Sartore; P. Traldi; | |
| Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug-resistance (MDR) modulators | 2019 | Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Marcella Coronnello, Niccolò Chiaramonte, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Chatchanok Udomtanakunchai, Nicola Antonio Colabufo, Gian luca Bartolucci, Ottavia Spiga, Milena Salerno, Elisabetta Teodori | |
| New dual P-Glycoprotein (P-gp) and human carbonic anhydrase XII (hCA XII) inhibitors as Multidrug Resistance (MDR) reversers in cancer cells | 2022 | Braconi, Laura; Teodori, Elisabetta; Riganti, Chiara; Coronnello, Marcella; Nocentini, Alessio; Bartolucci, Gian Luca; Pallecchi, Marco; Contino, Marialessandra; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T; Dei, Silvia | |
| New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators | 2022 | Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N. | |
| Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives | 2022 | Braconi L.; Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Manetti D.; Romanelli M.N.; Perrone M.G.; Colabufo N.A.; Guglielmo S.; Dei S. |