BRACONI, LAURA
BRACONI, LAURA
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
1-benzyl-1,4-diazepane reduces the efflux of resistance-nodulation-cell division pumps in Escherichia coli
2020 Enrico Casalone, Tiziano Vignolini, Laura Braconi, Lucia Gardini, Marco Capitanio, Francesco S Pavone, Silvia Dei, Elisabetta Teodori
2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity
2022 Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N.
6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers
2020 Braconi L.; Bartolucci G.; Contino M.; Chiaramonte N.; Giampietro R.; Manetti D.; Perrone M.G.; Romanelli M.N.; Colabufo N.A.; Riganti C.; Dei S.; Teodori E.
Application of LEDA algorithm for the recognition of P-glycoprotein and Carbonic Anhydrase hybrid inhibitors and evaluation of their plasma stability by HPLC-MS/MS analysis
2022 Pallecchi, Marco; Menicatti, Marta; Braconi, Laura; Supuran, Claudiu T; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca
Characterization of substituted piperazines able to reverse MDR in Escherichia coli strains overexpressing resistance-nodulation-cell division (RND) efflux pumps
2022 Casalone E.; Vignolini T.; Braconi L.; Gardini L.; Capitanio M.; Pavone F.S.; Giovannelli L.; Dei S.; Teodori E.
Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers
2019 Braconi L., Bartolucci G., Manetti D., Romanelli M.N., Dei S., Teodori E.
Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers
2019 Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Braconi L.; Manetti D.; Romanelli M.N.; Trezza A.; Athanasios A.; Spiga O.; Perrone M.G.; Giampietro R.; Gazzano E.; Salerno M.; Colabufo N.A.; Dei S.
Design, synthesis and characterization of new molecules which counteract drug resistance mechanisms
2022 Laura Braconi
Drug plasma stability study of multidrug resistance inhibitors by LC-MS/MS analysis
2018 Marta Menicatti, Matilde Maggini, Francesco Caponi, Donato Squillaci, Laura Braconi, Silvia Dei , Elisabetta Teodori, Gian Luca Bartolucci
Dual P-glycoprotein and CA XII inhibitors: A new strategy to reverse the P-gp Mediated Multidrug Resistance (MDR) in cancer cells y
2020 Teodori E.; Braconi L.; Bua S.; Lapucci A.; Bartolucci G.; Manetti D.; Romanelli M.N.; Dei S.; Supuran C.T.; Coronnello M.
ERMS EXPERIMENTS FOR RESOLUTION OF ISOBARIC COMPOUNDS: A CASE OF CIS/TRANS ISOMERISM
2018 Laura Braconi; Marta Menicatti; Silvia Dei; Elisabetta Teodori; Gian Luca Bartolucci
Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug-resistance (MDR) modulators
2019 Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Marcella Coronnello, Niccolò Chiaramonte, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Chatchanok Udomtanakunchai, Nicola Antonio Colabufo, Gian luca Bartolucci, Ottavia Spiga, Milena Salerno, Elisabetta Teodori
New dual P-Glycoprotein (P-gp) and human carbonic anhydrase XII (hCA XII) inhibitors as Multidrug Resistance (MDR) reversers in cancer cells
2022 Braconi, Laura; Teodori, Elisabetta; Riganti, Chiara; Coronnello, Marcella; Nocentini, Alessio; Bartolucci, Gian Luca; Pallecchi, Marco; Contino, Marialessandra; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T; Dei, Silvia
New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators
2022 Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N.
Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives
2022 Braconi L.; Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Manetti D.; Romanelli M.N.; Perrone M.G.; Colabufo N.A.; Guglielmo S.; Dei S.
P-glycoprotein and carbonic anhydrases hybrid inhibitors: a new strategy to reverse multidrug resistance (MDR) in cancer cells
2018 E. Teodori, M. Coronnello, S. Bua, L. Braconi, D. Manetti, M.N. Romanelli, C. Supuran, S. Dei
Recent advances in the discovery of Nicotinic acetylcholine receptor allosteric modulators
2023 Dina Manetti , Silvia Dei, Hugo R. Arias, Laura Braconi, Alessio Gabellini, Elisabetta Teodori, Maria Romanelli
Recent advances in the search of BCRP- and dual P-gp/BCRP-based multidrug resistance modulators
2019 Silvia Dei, Laura Braconi, Maria Novella Romanelli, Elisabetta Teodori
Simultaneous Degradation Study of Isomers in Human Plasma by HPLC-MS/MS and Application of LEDA Algorithm for Their Characterization
2022 Pallecchi, Marco; Braconi, Laura; Menicatti, Marta; Giachetti, Sara; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca
Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors
2019 Niccolò Chiaramontea, Silvia Bua, Andrea Angeli, Marta Ferraroni, Ilaria Picchioni, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T. Supuran, Maria Novella Romanelli
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1-benzyl-1,4-diazepane reduces the efflux of resistance-nodulation-cell division pumps in Escherichia coli | 2020 | Enrico Casalone, Tiziano Vignolini, Laura Braconi, Lucia Gardini, Marco Capitanio, Francesco S Pavone, Silvia Dei, Elisabetta Teodori | |
| 2-(2-Hydroxyethyl)piperazine derivatives as potent human carbonic anhydrase inhibitors: Synthesis, enzyme inhibition, computational studies and antiglaucoma activity | 2022 | Chiaramonte N.; Angeli A.; Sgambellone S.; Bonardi A.; Nocentini A.; Bartolucci G.; Braconi L.; Dei S.; Lucarini L.; Teodori E.; Gratteri P.; Wunsch B.; Supuran C.T.; Romanelli M.N. | |
| 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers | 2020 | Braconi L.; Bartolucci G.; Contino M.; Chiaramonte N.; Giampietro R.; Manetti D.; Perrone M.G.; Romanelli M.N.; Colabufo N.A.; Riganti C.; Dei S.; Teodori E. | |
| Application of LEDA algorithm for the recognition of P-glycoprotein and Carbonic Anhydrase hybrid inhibitors and evaluation of their plasma stability by HPLC-MS/MS analysis | 2022 | Pallecchi, Marco; Menicatti, Marta; Braconi, Laura; Supuran, Claudiu T; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca | |
| Characterization of substituted piperazines able to reverse MDR in Escherichia coli strains overexpressing resistance-nodulation-cell division (RND) efflux pumps | 2022 | Casalone E.; Vignolini T.; Braconi L.; Gardini L.; Capitanio M.; Pavone F.S.; Giovannelli L.; Dei S.; Teodori E. | |
| Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers | 2019 | Braconi L., Bartolucci G., Manetti D., Romanelli M.N., Dei S., Teodori E. | |
| Design, synthesis and biological evaluation of stereo- and regioisomers of amino aryl esters as multidrug resistance (MDR) reversers | 2019 | Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Braconi L.; Manetti D.; Romanelli M.N.; Trezza A.; Athanasios A.; Spiga O.; Perrone M.G.; Giampietro R.; Gazzano E.; Salerno M.; Colabufo N.A.; Dei S. | |
| Design, synthesis and characterization of new molecules which counteract drug resistance mechanisms | 2022 | Laura Braconi | |
| Drug plasma stability study of multidrug resistance inhibitors by LC-MS/MS analysis | 2018 | Marta Menicatti, Matilde Maggini, Francesco Caponi, Donato Squillaci, Laura Braconi, Silvia Dei , Elisabetta Teodori, Gian Luca Bartolucci | |
| Dual P-glycoprotein and CA XII inhibitors: A new strategy to reverse the P-gp Mediated Multidrug Resistance (MDR) in cancer cells y | 2020 | Teodori E.; Braconi L.; Bua S.; Lapucci A.; Bartolucci G.; Manetti D.; Romanelli M.N.; Dei S.; Supuran C.T.; Coronnello M. | |
| ERMS EXPERIMENTS FOR RESOLUTION OF ISOBARIC COMPOUNDS: A CASE OF CIS/TRANS ISOMERISM | 2018 | Laura Braconi; Marta Menicatti; Silvia Dei; Elisabetta Teodori; Gian Luca Bartolucci | |
| Modulation of the spacer in N,N-bis(alkanol)amine aryl ester heterodimers led to the discovery of a series of highly potent P-glycoprotein-based multidrug-resistance (MDR) modulators | 2019 | Silvia Dei, Laura Braconi, Alfonso Trezza, Marta Menicatti, Marialessandra Contino, Marcella Coronnello, Niccolò Chiaramonte, Dina Manetti, Maria Grazia Perrone, Maria Novella Romanelli, Chatchanok Udomtanakunchai, Nicola Antonio Colabufo, Gian luca Bartolucci, Ottavia Spiga, Milena Salerno, Elisabetta Teodori | |
| New dual P-Glycoprotein (P-gp) and human carbonic anhydrase XII (hCA XII) inhibitors as Multidrug Resistance (MDR) reversers in cancer cells | 2022 | Braconi, Laura; Teodori, Elisabetta; Riganti, Chiara; Coronnello, Marcella; Nocentini, Alessio; Bartolucci, Gian Luca; Pallecchi, Marco; Contino, Marialessandra; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T; Dei, Silvia | |
| New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators | 2022 | Chiaramonte N.; Gabellini A.; Angeli A.; Bartolucci G.; Braconi L.; Dei S.; Teodori E.; Supuran C.T.; Romanelli M.N. | |
| Overcoming Multidrug Resistance (MDR): Design, Biological Evaluation and Molecular Modelling Studies of 2,4-Substituted Quinazoline Derivatives | 2022 | Braconi L.; Teodori E.; Contino M.; Riganti C.; Bartolucci G.; Manetti D.; Romanelli M.N.; Perrone M.G.; Colabufo N.A.; Guglielmo S.; Dei S. | |
| P-glycoprotein and carbonic anhydrases hybrid inhibitors: a new strategy to reverse multidrug resistance (MDR) in cancer cells | 2018 | E. Teodori, M. Coronnello, S. Bua, L. Braconi, D. Manetti, M.N. Romanelli, C. Supuran, S. Dei | |
| Recent advances in the discovery of Nicotinic acetylcholine receptor allosteric modulators | 2023 | Dina Manetti , Silvia Dei, Hugo R. Arias, Laura Braconi, Alessio Gabellini, Elisabetta Teodori, Maria Romanelli | |
| Recent advances in the search of BCRP- and dual P-gp/BCRP-based multidrug resistance modulators | 2019 | Silvia Dei, Laura Braconi, Maria Novella Romanelli, Elisabetta Teodori | |
| Simultaneous Degradation Study of Isomers in Human Plasma by HPLC-MS/MS and Application of LEDA Algorithm for Their Characterization | 2022 | Pallecchi, Marco; Braconi, Laura; Menicatti, Marta; Giachetti, Sara; Dei, Silvia; Teodori, Elisabetta; Bartolucci, Gian Luca | |
| Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors | 2019 | Niccolò Chiaramontea, Silvia Bua, Andrea Angeli, Marta Ferraroni, Ilaria Picchioni, Gianluca Bartolucci, Laura Braconi, Silvia Dei, Elisabetta Teodori, Claudiu T. Supuran, Maria Novella Romanelli |