CARTA, FABRIZIO
CARTA, FABRIZIO
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site
2020 Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V.
2-Substituted-4,7-dihydro-4-ethylpyrazolo[1,5-a]pyrimidin-7-ones alleviate LPS-induced inflammation by modulating cell metabolism via CD73 upon macrophage polarization
2024 Ricci A.; Zara S.; Carta F.; Di Valerio V.; Sancilio S.; Cataldi A.; Selleri S.; Supuran C.T.; Carradori S.; Gallorini M.
4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies
2016 Cornelio, Benedetta; Laronze Cochard, Marie; Ceruso, Mariangela; Ferraroni, Marta; Rance, Graham A.; Carta, Fabrizio; Khlobystov, Andrei N.; Fontana, Antonella; Supuran, CLAUDIU TRANDAFIR; Sapi, Janos
5- and 6-membered (thio)lactones are prodrug type carbonic anhydrase inhibitors.
2012 F. Carta;A. Maresca;A. Scozzafava;C. T. Supuran
6-Substituted 1,2-benzoxathiine-2,2-dioxides are isoform-selective inhibitors of human carbonic anhydrases IX, XII and VA.
2015 M. Tanc;F. Carta;A. Scozzafava;C. T. Supuran
6-substituted sulfocoumarins are selective carbonic anhdydrase IX and XII Inhibitors with significant cytotoxicity against colorectal cancer cells
2015 Grandane, Aiga; Tanc, Muhammet; Di Cesare Mannelli, Lorenzo; Carta, Fabrizio; Ghelardini, Carla; Žalubovskis, Raivis; Supuran, Claudiu T.
7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring.
2015 Vullo, Daniela*; Isik, Semra; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T.
7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII
2016 Nocentini, Alessio; Ceruso, Mariangela; Carta, Fabrizio; Supuran, Claudiu T.
7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors.
2013 M. Tanc;F. Carta;M. Bozdag;A. Scozzafava;C. T. Supuran
[(Cp-R)M(CO)(3) ] (M=Re or (99m) Tc) Arylsulfonamide, Arylsulfamide, and Arylsulfamate Conjugates for Selective Targeting of Human Carbonic Anhydrase IX.
2012 D. Can;B. Spingler;P. Schmutz;F. Mendes;P. Raposinho;C. Fernandes;F. Carta;A. Innocenti;I. Santos;C. T. Supuran;R. Alberto
A CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE
2013 CLAUDIU SUPURAN; ANDREA SCOZZAFAVA; EMANUELA MASINI; FABRIZIO CARTA; ERIK OLAI PETTERSEN; PETER EBBERSEN
A cheminformatics and network pharmacology approach to elucidate the mechanism of action of Mycobacterium tuberculosis γ-carbonic anhydrase inhibitors
2024 Manaithiya A.; Bhowmik R.; Bhattacharya K.; Ray R.; Shyamal S.S.; Carta F.; Supuran C.T.; Parkkila S.; Aspatwar A.
A class of 4-Sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.
2014 M. Bozdag;M. Pinard;F. Carta;E. Masini;A. Scozzafava;R. McKenna;C. T. Supuran
A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects
2015 Carta, Fabrizio; Di Cesare Mannelli, Lorenzo; Pinard, Melissa; Ghelardini, Carla; Scozzafava, Andrea; Mckenna, Robert; Supuran, Claudiu T.
A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors
2019 Costa G.; Carta F.; Ambrosio F.A.; Artese A.; Ortuso F.; Moraca F.; Rocca R.; Romeo I.; Lupia A.; Maruca A.; Bagetta D.; Catalano R.; Vullo D.; Alcaro S.; Supuran C.T.
A data and knowledge-driven integrated modeling approach to organ-specific Tuberculosis subtype discovery: A one health paradigm
2024 Ray, Rajarshi; Bhowmik, Ratul; Shyamal, Sagar Singh; Manaithiya, Ajay; Carta, Fabrizio; Supuran, Claudiu T; Parkkila, Seppo; Aspatwar, Ashok
A deadly spillover: SARS-CoV-2 outbreak
2020 Mori M.; Capasso C.; Carta F.; Donald W.A.; Supuran C.T.
A multi-dimensional systems biology approach to elucidate the mechanism of action of Mycobacterium tuberculosis γ-carbonic anhydrase inhibitors
2024 Manaithiya, Ajay; Bhowmik, Ratul; Bhattacharya, Kunal; Ray, Rajarshi; Shyamal, Sagar Singh; Carta, Fabrizio; Supuran, Claudiu; Parkkila, Seppo; Aspatwar, Ashok
A multidimensional network-based approach to elucidate the molecular mechanism underlying tuberculosis and HIV coinfection
2024 Bhowmik, Ratul; Shyamal, Sagar Singh; Ray, Rajarshi; Carta, Fabrizio; Supuran, Claudiu T.; Parkkila, Seppo; Aspatwar, Ashok
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site | 2020 | Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V. | |
| 2-Substituted-4,7-dihydro-4-ethylpyrazolo[1,5-a]pyrimidin-7-ones alleviate LPS-induced inflammation by modulating cell metabolism via CD73 upon macrophage polarization | 2024 | Ricci A.; Zara S.; Carta F.; Di Valerio V.; Sancilio S.; Cataldi A.; Selleri S.; Supuran C.T.; Carradori S.; Gallorini M. | |
| 4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies | 2016 | Cornelio, Benedetta; Laronze Cochard, Marie; Ceruso, Mariangela; Ferraroni, Marta; Rance, Graham A.; Carta, Fabrizio; Khlobystov, Andrei N.; Fontana, Antonella; Supuran, CLAUDIU TRANDAFIR; Sapi, Janos | |
| 5- and 6-membered (thio)lactones are prodrug type carbonic anhydrase inhibitors. | 2012 | F. Carta;A. Maresca;A. Scozzafava;C. T. Supuran | |
| 6-Substituted 1,2-benzoxathiine-2,2-dioxides are isoform-selective inhibitors of human carbonic anhydrases IX, XII and VA. | 2015 | M. Tanc;F. Carta;A. Scozzafava;C. T. Supuran | |
| 6-substituted sulfocoumarins are selective carbonic anhdydrase IX and XII Inhibitors with significant cytotoxicity against colorectal cancer cells | 2015 | Grandane, Aiga; Tanc, Muhammet; Di Cesare Mannelli, Lorenzo; Carta, Fabrizio; Ghelardini, Carla; Žalubovskis, Raivis; Supuran, Claudiu T. | |
| 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. | 2015 | Vullo, Daniela*; Isik, Semra; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T. | |
| 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII | 2016 | Nocentini, Alessio; Ceruso, Mariangela; Carta, Fabrizio; Supuran, Claudiu T. | |
| 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors. | 2013 | M. Tanc;F. Carta;M. Bozdag;A. Scozzafava;C. T. Supuran | |
| [(Cp-R)M(CO)(3) ] (M=Re or (99m) Tc) Arylsulfonamide, Arylsulfamide, and Arylsulfamate Conjugates for Selective Targeting of Human Carbonic Anhydrase IX. | 2012 | D. Can;B. Spingler;P. Schmutz;F. Mendes;P. Raposinho;C. Fernandes;F. Carta;A. Innocenti;I. Santos;C. T. Supuran;R. Alberto | |
| A CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE | 2013 | CLAUDIU SUPURAN; ANDREA SCOZZAFAVA; EMANUELA MASINI; FABRIZIO CARTA; ERIK OLAI PETTERSEN; PETER EBBERSEN | |
| A cheminformatics and network pharmacology approach to elucidate the mechanism of action of Mycobacterium tuberculosis γ-carbonic anhydrase inhibitors | 2024 | Manaithiya A.; Bhowmik R.; Bhattacharya K.; Ray R.; Shyamal S.S.; Carta F.; Supuran C.T.; Parkkila S.; Aspatwar A. | |
| A class of 4-Sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects. | 2014 | M. Bozdag;M. Pinard;F. Carta;E. Masini;A. Scozzafava;R. McKenna;C. T. Supuran | |
| A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects | 2015 | Carta, Fabrizio; Di Cesare Mannelli, Lorenzo; Pinard, Melissa; Ghelardini, Carla; Scozzafava, Andrea; Mckenna, Robert; Supuran, Claudiu T. | |
| A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors | 2019 | Costa G.; Carta F.; Ambrosio F.A.; Artese A.; Ortuso F.; Moraca F.; Rocca R.; Romeo I.; Lupia A.; Maruca A.; Bagetta D.; Catalano R.; Vullo D.; Alcaro S.; Supuran C.T. | |
| A data and knowledge-driven integrated modeling approach to organ-specific Tuberculosis subtype discovery: A one health paradigm | 2024 | Ray, Rajarshi; Bhowmik, Ratul; Shyamal, Sagar Singh; Manaithiya, Ajay; Carta, Fabrizio; Supuran, Claudiu T; Parkkila, Seppo; Aspatwar, Ashok | |
| A deadly spillover: SARS-CoV-2 outbreak | 2020 | Mori M.; Capasso C.; Carta F.; Donald W.A.; Supuran C.T. | |
| A multi-dimensional systems biology approach to elucidate the mechanism of action of Mycobacterium tuberculosis γ-carbonic anhydrase inhibitors | 2024 | Manaithiya, Ajay; Bhowmik, Ratul; Bhattacharya, Kunal; Ray, Rajarshi; Shyamal, Sagar Singh; Carta, Fabrizio; Supuran, Claudiu; Parkkila, Seppo; Aspatwar, Ashok | |
| A multidimensional network-based approach to elucidate the molecular mechanism underlying tuberculosis and HIV coinfection | 2024 | Bhowmik, Ratul; Shyamal, Sagar Singh; Ray, Rajarshi; Carta, Fabrizio; Supuran, Claudiu T.; Parkkila, Seppo; Aspatwar, Ashok | |
| A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran |