CARTA, FABRIZIO
CARTA, FABRIZIO
Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA)
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site
2020 Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V.
4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies
2016 Cornelio, Benedetta; Laronze Cochard, Marie; Ceruso, Mariangela; Ferraroni, Marta; Rance, Graham A.; Carta, Fabrizio; Khlobystov, Andrei N.; Fontana, Antonella; Supuran, CLAUDIU TRANDAFIR; Sapi, Janos
5- and 6-membered (thio)lactones are prodrug type carbonic anhydrase inhibitors.
2012 F. Carta;A. Maresca;A. Scozzafava;C. T. Supuran
6-Substituted 1,2-benzoxathiine-2,2-dioxides are isoform-selective inhibitors of human carbonic anhydrases IX, XII and VA.
2015 M. Tanc;F. Carta;A. Scozzafava;C. T. Supuran
6-substituted sulfocoumarins are selective carbonic anhdydrase IX and XII Inhibitors with significant cytotoxicity against colorectal cancer cells
2015 Grandane, Aiga; Tanc, Muhammet; Di Cesare Mannelli, Lorenzo; Carta, Fabrizio; Ghelardini, Carla; Žalubovskis, Raivis; Supuran, Claudiu T.
7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring.
2015 Vullo, Daniela*; Isik, Semra; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T.
7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII
2016 Nocentini, Alessio; Ceruso, Mariangela; Carta, Fabrizio; Supuran, Claudiu T.
7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors.
2013 M. Tanc;F. Carta;M. Bozdag;A. Scozzafava;C. T. Supuran
[(Cp-R)M(CO)(3) ] (M=Re or (99m) Tc) Arylsulfonamide, Arylsulfamide, and Arylsulfamate Conjugates for Selective Targeting of Human Carbonic Anhydrase IX.
2012 D. Can;B. Spingler;P. Schmutz;F. Mendes;P. Raposinho;C. Fernandes;F. Carta;A. Innocenti;I. Santos;C. T. Supuran;R. Alberto
A CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE
2013 CLAUDIU SUPURAN; ANDREA SCOZZAFAVA; EMANUELA MASINI; FABRIZIO CARTA; ERIK OLAI PETTERSEN; PETER EBBERSEN
A class of 4-Sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects.
2014 M. Bozdag;M. Pinard;F. Carta;E. Masini;A. Scozzafava;R. McKenna;C. T. Supuran
A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects
2015 Carta, Fabrizio; Di Cesare Mannelli, Lorenzo; Pinard, Melissa; Ghelardini, Carla; Scozzafava, Andrea; Mckenna, Robert; Supuran, Claudiu T.
A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors
2019 Costa G.; Carta F.; Ambrosio F.A.; Artese A.; Ortuso F.; Moraca F.; Rocca R.; Romeo I.; Lupia A.; Maruca A.; Bagetta D.; Catalano R.; Vullo D.; Alcaro S.; Supuran C.T.
A deadly spillover: SARS-CoV-2 outbreak
2020 Mori M.; Capasso C.; Carta F.; Donald W.A.; Supuran C.T.
A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
2023 Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran
A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease
2019 Gustavo Provensi, Fabrizio Carta, Alessio Nocentini, Claudiu T. Supuran, Fiorella Casamenti, Maria Beatrice Passani, Silvia Fossati
A non-catalytic function of carbonic anhydrase IX contributes to the glycolytic phenotype and pH regulation in human breast cancer cells
2019 Mboge M.Y.; Chen Z.; Khokhar D.; Wolff A.; Ai L.; Heldermon C.D.; Bozdag M.; Carta F.; Supuran C.T.; Brown K.D.; McKenna R.; Frost C.J.; Frost S.C.
A potentiated cooperation of carbonic anhydrase IX and histone deacetylase inhibitors against cancer
2020 Ruzzolini J, Laurenzana A, Andreucci E, Peppicelli S, Bianchini F, Carta F, Supuran CT, Romanelli MN, Nediani C, Calorini L.
Acyl selenoureido benzensulfonamides show potent inhibitory activity against carbonic anhydrases from the pathogenic bacterium Vibrio cholerae
2017 Angeli, Andrea; Abbas, Ghulam; Del Prete, Sonia; Carta, Fabrizio; Capasso, Clemente; Supuran, Claudiu T.
Advances in New Psychoactive Substances Identification: The U.R.I.To.N Consortium
2017 Bertol, Elisabetta; Vaiano, Fabio; Mari, Francesco; Di Milia, Maria Grazia; Bua, Silvia; Supuran, Claudiu Trandafir; Carta, Fabrizio
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site | 2020 | Bozdag M.; Supuran C.T.; Esposito D.; Angeli A.; Carta F.; Monti S.M.; De Simone G.; Alterio V. | |
| 4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies | 2016 | Cornelio, Benedetta; Laronze Cochard, Marie; Ceruso, Mariangela; Ferraroni, Marta; Rance, Graham A.; Carta, Fabrizio; Khlobystov, Andrei N.; Fontana, Antonella; Supuran, CLAUDIU TRANDAFIR; Sapi, Janos | |
| 5- and 6-membered (thio)lactones are prodrug type carbonic anhydrase inhibitors. | 2012 | F. Carta;A. Maresca;A. Scozzafava;C. T. Supuran | |
| 6-Substituted 1,2-benzoxathiine-2,2-dioxides are isoform-selective inhibitors of human carbonic anhydrases IX, XII and VA. | 2015 | M. Tanc;F. Carta;A. Scozzafava;C. T. Supuran | |
| 6-substituted sulfocoumarins are selective carbonic anhdydrase IX and XII Inhibitors with significant cytotoxicity against colorectal cancer cells | 2015 | Grandane, Aiga; Tanc, Muhammet; Di Cesare Mannelli, Lorenzo; Carta, Fabrizio; Ghelardini, Carla; Žalubovskis, Raivis; Supuran, Claudiu T. | |
| 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibits α-carbonic anhydrases without hydrolysis of the lactam ring. | 2015 | Vullo, Daniela*; Isik, Semra; Bozdag, Murat; Carta, Fabrizio; Supuran, Claudiu T. | |
| 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII | 2016 | Nocentini, Alessio; Ceruso, Mariangela; Carta, Fabrizio; Supuran, Claudiu T. | |
| 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors. | 2013 | M. Tanc;F. Carta;M. Bozdag;A. Scozzafava;C. T. Supuran | |
| [(Cp-R)M(CO)(3) ] (M=Re or (99m) Tc) Arylsulfonamide, Arylsulfamide, and Arylsulfamate Conjugates for Selective Targeting of Human Carbonic Anhydrase IX. | 2012 | D. Can;B. Spingler;P. Schmutz;F. Mendes;P. Raposinho;C. Fernandes;F. Carta;A. Innocenti;I. Santos;C. T. Supuran;R. Alberto | |
| A CARBONIC ANHYDRASE INHIBITOR COMPRISING A DITHIOCARBAMATE | 2013 | CLAUDIU SUPURAN; ANDREA SCOZZAFAVA; EMANUELA MASINI; FABRIZIO CARTA; ERIK OLAI PETTERSEN; PETER EBBERSEN | |
| A class of 4-Sulfamoylphenyl-ω-aminoalkyl ethers with effective carbonic anhydrase inhibitory action and antiglaucoma effects. | 2014 | M. Bozdag;M. Pinard;F. Carta;E. Masini;A. Scozzafava;R. McKenna;C. T. Supuran | |
| A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects | 2015 | Carta, Fabrizio; Di Cesare Mannelli, Lorenzo; Pinard, Melissa; Ghelardini, Carla; Scozzafava, Andrea; Mckenna, Robert; Supuran, Claudiu T. | |
| A computer-assisted discovery of novel potential anti-obesity compounds as selective carbonic anhydrase VA inhibitors | 2019 | Costa G.; Carta F.; Ambrosio F.A.; Artese A.; Ortuso F.; Moraca F.; Rocca R.; Romeo I.; Lupia A.; Maruca A.; Bagetta D.; Catalano R.; Vullo D.; Alcaro S.; Supuran C.T. | |
| A deadly spillover: SARS-CoV-2 outbreak | 2020 | Mori M.; Capasso C.; Carta F.; Donald W.A.; Supuran C.T. | |
| A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration | 2023 | Emanuela Berrino; Simone Carradori; Fabrizio Carta; Francesco Melfi; Marialucia Gallorini; Giulio Poli; Tiziano Tuccinardi; José G. Fernández-Bolaños; Óscar López; Jacobus P. Petzer; Anél Petzer; Paolo Guglielmi; Daniela Secci; Claudiu T. Supuran | |
| A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease | 2019 | Gustavo Provensi, Fabrizio Carta, Alessio Nocentini, Claudiu T. Supuran, Fiorella Casamenti, Maria Beatrice Passani, Silvia Fossati | |
| A non-catalytic function of carbonic anhydrase IX contributes to the glycolytic phenotype and pH regulation in human breast cancer cells | 2019 | Mboge M.Y.; Chen Z.; Khokhar D.; Wolff A.; Ai L.; Heldermon C.D.; Bozdag M.; Carta F.; Supuran C.T.; Brown K.D.; McKenna R.; Frost C.J.; Frost S.C. | |
| A potentiated cooperation of carbonic anhydrase IX and histone deacetylase inhibitors against cancer | 2020 | Ruzzolini J, Laurenzana A, Andreucci E, Peppicelli S, Bianchini F, Carta F, Supuran CT, Romanelli MN, Nediani C, Calorini L. | |
| Acyl selenoureido benzensulfonamides show potent inhibitory activity against carbonic anhydrases from the pathogenic bacterium Vibrio cholerae | 2017 | Angeli, Andrea; Abbas, Ghulam; Del Prete, Sonia; Carta, Fabrizio; Capasso, Clemente; Supuran, Claudiu T. | |
| Advances in New Psychoactive Substances Identification: The U.R.I.To.N Consortium | 2017 | Bertol, Elisabetta; Vaiano, Fabio; Mari, Francesco; Di Milia, Maria Grazia; Bua, Silvia; Supuran, Claudiu Trandafir; Carta, Fabrizio |