MACHETTI, FABRIZIO
 Distribuzione geografica
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Continente #
NA - Nord America 2.592
EU - Europa 1.677
AS - Asia 321
AF - Africa 8
SA - Sud America 2
OC - Oceania 1
Totale 4.601
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Nazione #
US - Stati Uniti d'America 2.584
PL - Polonia 396
SE - Svezia 311
IE - Irlanda 266
IT - Italia 210
UA - Ucraina 176
DE - Germania 127
HK - Hong Kong 110
VN - Vietnam 78
GB - Regno Unito 65
FI - Finlandia 55
CN - Cina 45
JO - Giordania 35
FR - Francia 25
KR - Corea 15
IN - India 13
TR - Turchia 13
BE - Belgio 12
RU - Federazione Russa 12
CH - Svizzera 7
ES - Italia 6
SC - Seychelles 6
AT - Austria 4
CA - Canada 4
MX - Messico 4
IQ - Iraq 3
JP - Giappone 3
MY - Malesia 3
SG - Singapore 3
BR - Brasile 2
NL - Olanda 2
AU - Australia 1
EG - Egitto 1
LU - Lussemburgo 1
MD - Moldavia 1
MU - Mauritius 1
RO - Romania 1
Totale 4.601
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Città #
Warsaw 395
Fairfield 351
Chandler 296
Jacksonville 287
Dublin 260
Woodbridge 159
Cambridge 156
Ashburn 155
Seattle 145
Wilmington 123
Houston 120
Ann Arbor 95
Dong Ket 78
Princeton 61
Hong Kong 57
Florence 54
Altamura 44
Lawrence 42
Medford 42
Boardman 38
Boston 34
Buffalo 34
Menlo Park 34
San Diego 25
Beijing 23
West Jordan 17
Shanghai 16
Milan 15
Frankfurt Am Main 13
Norwalk 13
Brussels 12
Auburn Hills 11
Andover 9
Falls Church 9
Izmir 9
Los Angeles 8
Bern 7
New York 7
Pune 6
Moscow 5
Philadelphia 5
Regensburg 5
Villeurbanne 5
Acerra 4
Kolkata 4
London 4
Toronto 4
Verona 4
Vienna 4
Barcelona 3
Bologna 3
Cuernavaca 3
Erbil 3
Hillsboro 3
Kajang 3
Salerno 3
Seveso 3
Bellante 2
Changsha 2
Charlottesville 2
Düsseldorf 2
Jaipur 2
Kilburn 2
Madrid 2
Mentor 2
Ogarëv 2
Redmond 2
Rome 2
Saint Petersburg 2
Siena 2
Washington 2
Campinas 1
Cedar Knolls 1
Cerveteri 1
Chisinau 1
Cork 1
Damietta 1
Edinburgh 1
Follonica 1
Gustavo Adolfo Madero 1
Hanover 1
Huntsville 1
Laguna Niguel 1
Landshut 1
Lodz 1
Luxembourg 1
Mascalucia 1
Messina 1
Nanjing 1
Napoli 1
Phoenix 1
Praia A Mare 1
Rosignano Marittimo 1
Salamanca 1
San Mateo 1
Sansepolcro 1
Singapore 1
St Petersburg 1
State College 1
Sydney 1
Totale 3.385
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Nome #
19-nor-10-azasteroids, a new class of steroid 5a-reductase inhibitors. 2. X-ray structure, molecular modeling, conformational analysis of 19-nor-10-azasteroids and comparison with 4-azasteroids and 6-azasteroids 232
19-nor-10-azasteroids: a novel class of inhibitors for human steroid 5alpha-reductases 1 and 2 187
Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1 184
1,2,5-Oxadiazole (Furazan) derivatives from benzoylnitromethane and dipolarophiles in the presence of DABCO: structure and intermediates. 141
1,4-Diazabicyclo[2.2.2]octane (DABCO) as an efficient reagent for the synthesis of isoxazole derivatives from primary nitro compounds and dipolarophiles: The role of the base 127
4,5-Dihydroisoxazoles by copper(II)-catalysed condensation of primary nitroalkanes with dipolarophiles 105
A New Bicyclic Dipeptide Isostere with Pyrrolizidinone Skeleton 103
Identification of Inhibitors of Drug-Resistant Candida albicans Strains from a Library of Bicyclic Peptidomimetic Compounds 99
Bicyclic Compounds Derived from Tartaric Acid and -Amino Acids (BTAas): Synthesis of New Molecular Scaffolds Derived from the Combination of (R,R)-Tartaric Acid and L-Serine 94
SYNTHESIS OF TAURINE ANALOGUES. PART 1: 2-AMINOSULFONIC ACIDS FROM ALKENE-SULFUR MONOCHLORIDE ADDUCTS 93
Isoxazoline derivatives from activated primary nitro compounds and tertiary diamines 92
Multiwalled carbon nanotubes for combination therapy: a biodistribution and efficacy pilot study 92
Synthesis of Taurine Analogues from Alkenes 89
Inhibition of rabbit brain 4-aminobutyrate transaminase by some taurine analogues: a kinetic analysis. 89
Synthesis of 4,5-dihydroisoxazoles by condensation of primary nitro compounds with alkenes by using a copper/base catalytic system. 87
Effect of C-Ring Modifications in Benzo[c]quinolizin-3-ones, New Selective Inhibitors of Human 5a-Reductase 1 86
Bicyclic compounds derived from Tartaric Acid and α-Amino acids (BTAas): Synthesis of New Molecular Scaffolds derived from the Combination of (R,R)-Tartaric Acid and L-Serine 85
Competitive Copper Catalysis in the Condensation of Primary Nitro Compounds with Terminal Alkynes: Synthesis of Isoxazoles 85
Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition or Catalysed Condensation to Isoxazolo[60]fullerenes 84
Conversion of a nitrosocarbonyl hetero Diels-Alder cycloadduct to useful isoxazoline-carbocyclic aminols 84
Oligomers of enantiopure bicyclic g/d-amino acids (BTAa). 1. Synthesis and conformational analysis of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid oligomers (PolyBTG) 81
Base- and Copper-Catalysed Condensation of Primary Activated Nitro Compounds with Enolisable Compounds 81
4.03 - Isoxazoles 81
The Synthesis of 4-Hydroxypipecolic Acids by Stereoselective Cycloaddition of Configurationally Stable Nitrones 79
Synthesis and X-ray study of hexahydro- and tetrahydrophospholo[2,3-d]isoxazoles, a new class of heterocycles of potential fungicidal activity 78
31.5.7 - Five-Membered Ring Systems: With O and N Atoms 76
MODIFICATION OF THE AZA-ROBINSON ANNULATION FOR THE SYNTHESIS OF 4-METHYL-BENZO[C]QUINOLIZIN-3-ONES, POTENT INHIBITORS OF STEROID 5A-REDUCTASE 1 75
Enantiospecific synthesis of 3-aza-6,8-dioxa-bicyclo[3.2.1]octane carboxylic acids from erythrose 74
Parallel Synthesis of an Amide Library Based on the 6,8-Dioxa-3-azabicyclo[3.2.1]octane Scaffold by Direct Aminolysis of Methyl Esters. 73
19-NOR-10-AZASTEROIDS. 5.1 A SYNTHETIC STRATEGY FOR THE PREPARATION OF (+)-17-(3-PYRIDYL)-(5B)-10-AZAESTRA-1,16-DIEN-3-ONE, A NOVEL POTENTIAL INHIBITOR FOR HUMAN CYTOCHROME P45017A (17A-HYDROXYLASE/C17,20-LYASE) 72
Practical synthesis of both enantiomers of protected 4-oxopipecolic acid. 72
Neat reaction of carboxylic acid methyl esters and amines for efficient parallel synthesis of scaffold amide libraries. 69
32.5.7 - Five-Membered Ring Systems: With O and N Atoms 68
Design and Synthesis of a New Bicyclic Dipeptide Isostere 67
Synthesis and reactivity of bicycles derived from tartaric acids and alfa-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid 66
A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5-REDUCTASE INHIBITORS. 3.1 SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-17B-ACETYLOXY-(5B)-10-AZAESTR-1-EN-3-ONE 64
Design, Synthesis and Applications of 3-Aza-6,8-Dioxa-Bicyclo[3.2.1]Octane-Based Scaffolds for peptidominetic Chemistry 64
Synthesis of Bicyclic Molecular Scaffolds (BTAa) for the Development of New Matrix Metalloproteinases Inhibitors 64
New Synthesis of (Methoxycarbonyl)-indolizidine-7-one and -quinolizidine-2-one: an Access to β-Aminoacids with Indolizidine and Quinolizidine Backbone 63
Michael Addition versus Cycloaddition-Condensation of Ethyl Nitroacetate with Electron-deficient Olefins 61
Five membered heterocycles: 1,3 azoles 61
STEREOSELECTIVITY IN THE TICL4-CATALYSED REEACTION OF DANISHEFSKY¿S DIENE WITH A N-(ACYLOXY)IMINIUM ION: SYNTHESIS OF 5A VERSUS 5B D1(2)-19-NOR-10-AZASTEROIDS. PART 4 60
PYRROLIZINONE DERIVATIVES AS NEW BICYCLIC GLY-PRO DIPEPTIDE ISOSTERS 57
Acid–Base-Catalysed Condensation Reaction in Water: Isoxazolines andIsoxazoles from Nitroacetates and Dipolarophiles 57
A New Synthesis of (2S)-4-Oxopipecolic Acid by Thermal Rearrangement ofEnantiopure Spirocyclopropaneisoxazolidine 55
Isoxazoles 54
3-Aza-6,8-dioxabicyclo (3,2,1) octanes and analogues and combinatorial libraries 52
Studies Towards the Synthesis of Enantiopure 4-Substituted Pipecolic Acids 50
Synthesis of New Enantiopure Bicycles gamma/delta-Amino Acid (BTKa), Derived from Tartaric Acid and alfa-Aminoacetophenone 48
Synthesis of benzo[c]quinolizin-3-ones: discovery and development of novel inhibitors of human steroid 5alpha-reductase 46
Synthesis and Structure-Activity Relationship of 19-Nor-10-azasteroids, a New Class of 5α -Reductase Inhibitors in Human Prostate. 46
Synthesis of free and Nalpha-Fmoc/Ngamma-Boc protected (2S, 4S)- and (2S, 4R)-4-aminopipecolic acids 46
DETERMINATION OF ABSOLUTE CONFIGURATION OF BICYCLIC LACTAMIC PROLINES USING THEIR MTPA ESTERS 44
XIV Convegno nazionale sulle reazioni pericicliche e sintesi di etero e carbocicli 43
BICYCLIC DIPEPTIDE ISOSTERES, THEIR PREPARATION AND USE AS BETA-TURN MIMICS 40
STUDIO DELLE CARATTERISTICHE ANALITICHE ED APPLICATIVE DI ALCUNI TANNINI VEGETALI E SINTETICI PER LA CONCIA DEL CUOIO. 40
Synthesis of Taurine Analogues, Part 2. Amino-Sulfonation of Alkenes by a Three Component Reaction 40
Isoxazoles and Isoxazolines by 1,3-dipolar Cycloaddition (1,3-DC). Base-Catalyzed Condensation of Primary Nitro compounds with Dipolarophiles to Isoxazole Derivatives. 38
Emerging drugs for the third millenium. Discovery and development of the inhibitors of steroids 5alpha-reductase as drugs for the androgen-dependant diaseas 36
33.5.7 - Five-Membered Ring Systems: With O and N Atoms 27
35.5.7 - Five-membered ring systems with O and N atoms 24
34.5.7 - Five-membered ring systems with O and N atoms 18
5-(Benzoyloxymethyl)isoxazole-3-carboxylic Acid Ethyl Ester 3
Totale 4.651
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Categoria #
all - tutte 12.254
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 12.254
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019328 0 0 0 0 0 0 0 0 0 70 134 124
2019/2020949 83 90 27 95 85 120 86 134 77 46 85 21
2020/2021731 56 30 69 75 13 88 13 85 44 86 37 135
2021/2022476 15 43 32 54 41 17 15 25 20 12 101 101
2022/20231.163 109 153 53 114 94 240 155 79 109 4 32 21
2023/2024368 14 52 65 19 25 58 24 73 5 33 0 0
Totale 4.651