MACHETTI, FABRIZIO
 Distribuzione geografica
Salva come PNG Salva come JPEG
Continente #
NA - Nord America 3.895
EU - Europa 2.395
AS - Asia 541
OC - Oceania 45
AF - Africa 19
SA - Sud America 3
Totale 6.898
Salva come PNG Salva come JPEG
Nazione #
US - Stati Uniti d'America 3.884
RU - Federazione Russa 703
PL - Polonia 396
SE - Svezia 311
IE - Irlanda 266
IT - Italia 221
UA - Ucraina 177
SG - Singapore 140
DE - Germania 130
HK - Hong Kong 124
VN - Vietnam 78
CN - Cina 65
FI - Finlandia 65
GB - Regno Unito 65
IN - India 46
AU - Australia 45
JO - Giordania 35
FR - Francia 25
TR - Turchia 17
KR - Corea 16
BE - Belgio 12
CI - Costa d'Avorio 11
CH - Svizzera 7
CA - Canada 6
ES - Italia 6
JP - Giappone 6
SC - Seychelles 6
IQ - Iraq 5
MX - Messico 5
AT - Austria 4
ID - Indonesia 4
MY - Malesia 3
NL - Olanda 3
BR - Brasile 2
MD - Moldavia 2
AE - Emirati Arabi Uniti 1
EG - Egitto 1
LU - Lussemburgo 1
MU - Mauritius 1
PE - Perù 1
RO - Romania 1
TW - Taiwan 1
Totale 6.898
Salva come PNG Salva come JPEG
Città #
Santa Clara 1.122
Warsaw 395
Fairfield 351
Chandler 296
Jacksonville 287
Dublin 260
Woodbridge 159
Cambridge 156
Ashburn 155
Seattle 145
Wilmington 123
Houston 120
Singapore 103
Ann Arbor 95
Dong Ket 78
Hong Kong 71
Florence 62
Princeton 61
Altamura 44
Melbourne 44
Lawrence 42
Medford 42
Boardman 41
Boston 34
Buffalo 34
Menlo Park 34
Mumbai 32
San Diego 25
Beijing 23
Shanghai 21
Moscow 18
West Jordan 17
Milan 16
Frankfurt Am Main 13
Kent 13
Norwalk 13
Brussels 12
Abidjan 11
Auburn Hills 11
Andover 9
Falls Church 9
Izmir 9
Los Angeles 9
Helsinki 8
Bern 7
New York 7
Pune 6
Yubileyny 6
Philadelphia 5
Regensburg 5
Villeurbanne 5
Acerra 4
Charlottesville 4
Jakarta 4
Kolkata 4
London 4
Toronto 4
Verona 4
Vienna 4
Ankara 3
Barcelona 3
Bologna 3
Cuernavaca 3
Erbil 3
Hillsboro 3
Kajang 3
Nanjing 3
Salerno 3
Seveso 3
Tokyo 3
Bellante 2
Changsha 2
Chisinau 2
Columbia 2
Düsseldorf 2
Jaipur 2
Kilburn 2
Lappeenranta 2
Madrid 2
Mentor 2
Mosul 2
Ogarëv 2
Redmond 2
Rome 2
Romola 2
Saint Petersburg 2
Siena 2
Victoria 2
Washington 2
Aachen 1
Bursa 1
Campinas 1
Cedar Knolls 1
Cerveteri 1
Chongqing 1
Cork 1
Damietta 1
Dubai 1
Edinburgh 1
Follonica 1
Totale 4.778
Salva come PNG Salva come JPEG
Nome #
19-nor-10-azasteroids, a new class of steroid 5a-reductase inhibitors. 2. X-ray structure, molecular modeling, conformational analysis of 19-nor-10-azasteroids and comparison with 4-azasteroids and 6-azasteroids 270
19-nor-10-azasteroids: a novel class of inhibitors for human steroid 5alpha-reductases 1 and 2 227
Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1 225
1,2,5-Oxadiazole (Furazan) derivatives from benzoylnitromethane and dipolarophiles in the presence of DABCO: structure and intermediates. 200
1,4-Diazabicyclo[2.2.2]octane (DABCO) as an efficient reagent for the synthesis of isoxazole derivatives from primary nitro compounds and dipolarophiles: The role of the base 168
A New Bicyclic Dipeptide Isostere with Pyrrolizidinone Skeleton 153
4,5-Dihydroisoxazoles by copper(II)-catalysed condensation of primary nitroalkanes with dipolarophiles 141
4.03 - Isoxazoles 138
Multiwalled carbon nanotubes for combination therapy: a biodistribution and efficacy pilot study 137
Bicyclic Compounds Derived from Tartaric Acid and -Amino Acids (BTAas): Synthesis of New Molecular Scaffolds Derived from the Combination of (R,R)-Tartaric Acid and L-Serine 133
SYNTHESIS OF TAURINE ANALOGUES. PART 1: 2-AMINOSULFONIC ACIDS FROM ALKENE-SULFUR MONOCHLORIDE ADDUCTS 128
Identification of Inhibitors of Drug-Resistant Candida albicans Strains from a Library of Bicyclic Peptidomimetic Compounds 128
Effect of C-Ring Modifications in Benzo[c]quinolizin-3-ones, New Selective Inhibitors of Human 5a-Reductase 1 127
Synthesis of Taurine Analogues from Alkenes 127
Base- and Copper-Catalysed Condensation of Primary Activated Nitro Compounds with Enolisable Compounds 125
Isoxazoline derivatives from activated primary nitro compounds and tertiary diamines 124
Synthesis of 4,5-dihydroisoxazoles by condensation of primary nitro compounds with alkenes by using a copper/base catalytic system. 122
31.5.7 - Five-Membered Ring Systems: With O and N Atoms 120
Reactivity of [60]Fullerene with Primary Nitro Compounds: Addition or Catalysed Condensation to Isoxazolo[60]fullerenes 119
Competitive Copper Catalysis in the Condensation of Primary Nitro Compounds with Terminal Alkynes: Synthesis of Isoxazoles 119
Conversion of a nitrosocarbonyl hetero Diels-Alder cycloadduct to useful isoxazoline-carbocyclic aminols 118
Bicyclic compounds derived from Tartaric Acid and α-Amino acids (BTAas): Synthesis of New Molecular Scaffolds derived from the Combination of (R,R)-Tartaric Acid and L-Serine 116
Inhibition of rabbit brain 4-aminobutyrate transaminase by some taurine analogues: a kinetic analysis. 115
32.5.7 - Five-Membered Ring Systems: With O and N Atoms 112
Oligomers of enantiopure bicyclic g/d-amino acids (BTAa). 1. Synthesis and conformational analysis of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid oligomers (PolyBTG) 111
MODIFICATION OF THE AZA-ROBINSON ANNULATION FOR THE SYNTHESIS OF 4-METHYL-BENZO[C]QUINOLIZIN-3-ONES, POTENT INHIBITORS OF STEROID 5A-REDUCTASE 1 109
The Synthesis of 4-Hydroxypipecolic Acids by Stereoselective Cycloaddition of Configurationally Stable Nitrones 109
Synthesis and X-ray study of hexahydro- and tetrahydrophospholo[2,3-d]isoxazoles, a new class of heterocycles of potential fungicidal activity 109
19-NOR-10-AZASTEROIDS. 5.1 A SYNTHETIC STRATEGY FOR THE PREPARATION OF (+)-17-(3-PYRIDYL)-(5B)-10-AZAESTRA-1,16-DIEN-3-ONE, A NOVEL POTENTIAL INHIBITOR FOR HUMAN CYTOCHROME P45017A (17A-HYDROXYLASE/C17,20-LYASE) 109
Enantiospecific synthesis of 3-aza-6,8-dioxa-bicyclo[3.2.1]octane carboxylic acids from erythrose 106
A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5-REDUCTASE INHIBITORS. 3.1 SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-17B-ACETYLOXY-(5B)-10-AZAESTR-1-EN-3-ONE 105
Design and Synthesis of a New Bicyclic Dipeptide Isostere 104
New Synthesis of (Methoxycarbonyl)-indolizidine-7-one and -quinolizidine-2-one: an Access to β-Aminoacids with Indolizidine and Quinolizidine Backbone 103
Synthesis and reactivity of bicycles derived from tartaric acids and alfa-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid 103
Practical synthesis of both enantiomers of protected 4-oxopipecolic acid. 103
PYRROLIZINONE DERIVATIVES AS NEW BICYCLIC GLY-PRO DIPEPTIDE ISOSTERS 101
Parallel Synthesis of an Amide Library Based on the 6,8-Dioxa-3-azabicyclo[3.2.1]octane Scaffold by Direct Aminolysis of Methyl Esters. 101
Design, Synthesis and Applications of 3-Aza-6,8-Dioxa-Bicyclo[3.2.1]Octane-Based Scaffolds for peptidominetic Chemistry 100
Synthesis of Bicyclic Molecular Scaffolds (BTAa) for the Development of New Matrix Metalloproteinases Inhibitors 100
STEREOSELECTIVITY IN THE TICL4-CATALYSED REEACTION OF DANISHEFSKY¿S DIENE WITH A N-(ACYLOXY)IMINIUM ION: SYNTHESIS OF 5A VERSUS 5B D1(2)-19-NOR-10-AZASTEROIDS. PART 4 97
A New Synthesis of (2S)-4-Oxopipecolic Acid by Thermal Rearrangement ofEnantiopure Spirocyclopropaneisoxazolidine 97
Neat reaction of carboxylic acid methyl esters and amines for efficient parallel synthesis of scaffold amide libraries. 96
Isoxazoles 92
Michael Addition versus Cycloaddition-Condensation of Ethyl Nitroacetate with Electron-deficient Olefins 90
Five membered heterocycles: 1,3 azoles 88
Acid–Base-Catalysed Condensation Reaction in Water: Isoxazolines andIsoxazoles from Nitroacetates and Dipolarophiles 88
Synthesis of New Enantiopure Bicycles gamma/delta-Amino Acid (BTKa), Derived from Tartaric Acid and alfa-Aminoacetophenone 87
3-Aza-6,8-dioxabicyclo (3,2,1) octanes and analogues and combinatorial libraries 87
Synthesis of free and Nalpha-Fmoc/Ngamma-Boc protected (2S, 4S)- and (2S, 4R)-4-aminopipecolic acids 83
Synthesis of Taurine Analogues, Part 2. Amino-Sulfonation of Alkenes by a Three Component Reaction 79
Studies Towards the Synthesis of Enantiopure 4-Substituted Pipecolic Acids 77
Synthesis of benzo[c]quinolizin-3-ones: discovery and development of novel inhibitors of human steroid 5alpha-reductase 74
Synthesis and Structure-Activity Relationship of 19-Nor-10-azasteroids, a New Class of 5α -Reductase Inhibitors in Human Prostate. 73
XIV Convegno nazionale sulle reazioni pericicliche e sintesi di etero e carbocicli 73
BICYCLIC DIPEPTIDE ISOSTERES, THEIR PREPARATION AND USE AS BETA-TURN MIMICS 70
33.5.7 - Five-Membered Ring Systems: With O and N Atoms 69
STUDIO DELLE CARATTERISTICHE ANALITICHE ED APPLICATIVE DI ALCUNI TANNINI VEGETALI E SINTETICI PER LA CONCIA DEL CUOIO. 67
DETERMINATION OF ABSOLUTE CONFIGURATION OF BICYCLIC LACTAMIC PROLINES USING THEIR MTPA ESTERS 67
35.5.7 - Five-membered ring systems with O and N atoms 66
Isoxazoles and Isoxazolines by 1,3-dipolar Cycloaddition (1,3-DC). Base-Catalyzed Condensation of Primary Nitro compounds with Dipolarophiles to Isoxazole Derivatives. 65
Emerging drugs for the third millenium. Discovery and development of the inhibitors of steroids 5alpha-reductase as drugs for the androgen-dependant diaseas 64
34.5.7 - Five-membered ring systems with O and N atoms 60
5-(Benzoyloxymethyl)isoxazole-3-carboxylic Acid Ethyl Ester 42
Synthesis of 2-Azetidinones via Cycloaddition Approaches: An Update 33
Totale 6.949
Salva come PNG Salva come JPEG
Categoria #
all - tutte 17.875
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 17.875
Salva come PNG Salva come JPEG


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020449 0 0 0 0 0 0 86 134 77 46 85 21
2020/2021731 56 30 69 75 13 88 13 85 44 86 37 135
2021/2022476 15 43 32 54 41 17 15 25 20 12 101 101
2022/20231.163 109 153 53 114 94 240 155 79 109 4 32 21
2023/2024413 14 52 65 19 25 58 24 73 5 33 30 15
2024/20252.253 86 259 164 406 842 486 10 0 0 0 0 0
Totale 6.949