OCCHIATO, ERNESTO GIOVANNI
 Distribuzione geografica
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Continente #
NA - Nord America 5.552
EU - Europa 3.461
AS - Asia 394
AF - Africa 17
SA - Sud America 3
Continente sconosciuto - Info sul continente non disponibili 1
Totale 9.428
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Nazione #
US - Stati Uniti d'America 5.538
PL - Polonia 1.366
IE - Irlanda 487
SE - Svezia 438
IT - Italia 391
UA - Ucraina 289
DE - Germania 193
HK - Hong Kong 183
FI - Finlandia 108
GB - Regno Unito 95
CN - Cina 86
JO - Giordania 45
TR - Turchia 30
FR - Francia 23
RU - Federazione Russa 20
VN - Vietnam 18
CA - Canada 13
SC - Seychelles 13
CH - Svizzera 12
BE - Belgio 11
ES - Italia 11
IN - India 11
SG - Singapore 11
AT - Austria 7
NL - Olanda 6
JP - Giappone 4
BR - Brasile 3
MY - Malesia 3
PK - Pakistan 3
CM - Camerun 2
MU - Mauritius 2
RO - Romania 2
EU - Europa 1
HU - Ungheria 1
MD - Moldavia 1
MX - Messico 1
Totale 9.428
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Città #
Warsaw 1.366
Fairfield 878
Chandler 534
Dublin 486
Jacksonville 453
Ashburn 450
Woodbridge 383
Seattle 350
Cambridge 349
Wilmington 309
Houston 304
Ann Arbor 145
Altamura 142
Princeton 135
Lawrence 130
Boardman 88
Florence 81
Hong Kong 81
Boston 73
Medford 71
San Diego 68
Buffalo 39
Beijing 38
New York 32
Shanghai 31
Izmir 27
Milan 23
Dong Ket 18
Falls Church 18
Norwalk 17
Auburn Hills 14
Frankfurt Am Main 14
Moscow 14
Hillsboro 13
Philadelphia 12
Barcelona 11
Brussels 11
Los Angeles 11
Bern 10
West Jordan 10
London 9
Scandicci 9
Toronto 9
Andover 8
Laurel 8
Washington 8
Bremen 7
Phoenix 7
Pune 7
Verona 7
Vienna 7
Torino 5
Düsseldorf 4
Nanjing 4
Ottawa 4
Redwood City 4
San Mateo 4
Singapore 4
Chengdu 3
Kajang 3
Muzaffargarh 3
Rome 3
Salerno 3
Tappahannock 3
Atsugi 2
Campinas 2
Dongying 2
Goleta 2
Hanover 2
Lucca 2
Mountain View 2
Muro Lucano 2
Naaldwijk 2
Ogarëv 2
Padova 2
Pisa 2
Prescot 2
Arnsberg 1
Augusta 1
Brentford 1
Budapest 1
Calvisano 1
Central 1
Chicago 1
Chisinau 1
Chiswick 1
Corato 1
Cork 1
Dallas 1
Delhi 1
Empoli 1
Fucecchio 1
Grevenbroich 1
Gunzenhausen 1
Hangzhou 1
Hefei 1
Islington 1
Istanbul 1
Kilburn 1
Laguna Niguel 1
Totale 7.421
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Nome #
Treatment with 8-OH-modified adenine (TLR7 ligand)-allergen conjugates decreases T helper type 2-oriented murine airway inflammation 242
A novel allergen-adjuvant conjugate suitable for specific immunotherapy of respiratory allergy 236
19-nor-10-azasteroids, a new class of steroid 5a-reductase inhibitors. 2. X-ray structure, molecular modeling, conformational analysis of 19-nor-10-azasteroids and comparison with 4-azasteroids and 6-azasteroids 232
Synthesis of benzo[c]quinolizin-3-ones: selective non steroidal inhibitors of steroid 5a-Reductase 1 229
Dermatophagoides pteronyssinus group 2 allergen bound to 8-OH modified adenine reduces the Th2-mediated airway inflammation without inducing a Th17 response and autoimmunity 218
5alpha-reductase ihnibitors, chemical and clinical models 191
19-nor-10-azasteroids: a novel class of inhibitors for human steroid 5alpha-reductases 1 and 2 187
Synthesis and conformational analysis of peptides embodying 2,3-methanopipecolic acids 185
Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1 184
Pharmacokinetics of 4-hydroxyandrostenedione in man after intramuscular injection of different formulations and the effect of this drug on plasma aromatizable androgens and 17beta-estradiol concentrations. 177
Stereodivergent synthesis of 5-aminopipecolic acids and application in the preparation of a cyclic RGD peptidomimetic as a nanomolar αvβ3 integrin ligand 125
5A-REDUCTASE INHIBITORS, CHEMICAL AND CLINICAL MODELS 109
PD(0)-CATALYZED CROSS COUPLING REACTIONS OF BORON DERIVATIVES WITH A LACTAM-DERIVED N-BOC ENOL TRIFLATE 100
Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity 100
BAKER'S YEAST REDUCTION OF PROCHIRAL G-NITROKETONES: ENANTIOSELECTIVE SYNTHESIS OF (S)-4-NITROALCOHOLS 99
STEREOSELECTIVE SYNTHESIS OF SPIROCYCLIC KETONES BY NAZAROV REACTION 99
ASYMMETRIC HYDROGENATION OF PROCHIRAL G-NITROKETONES BY RUTHENIUM COMPLEXES 97
Enantioselective Addition of Diethylzinc to Aldehydes using 1,4-Aminoalcohols as Chiral Ligands. 96
Bicyclic Compounds Derived from Tartaric Acid and -Amino Acids (BTAas): Synthesis of New Molecular Scaffolds Derived from the Combination of (R,R)-Tartaric Acid and L-Serine 94
Construction of Cyclopenta[b]indol-1-ones by a Tandem Gold(I)-Catalyzed Rearrangement/Nazarov Reaction and Application to the Synthesis of Bruceolline H 90
Density Functional Studies on the Nazarov Reaction Involving Cyclic Systems. 89
New Potent Fluorescent Analogues of Strigolactones: Synthesis and Biological Activity in Parasitic Weed Germination and Fungal Branching 89
Cyclopropane Pipecolic Acids as Templates for Linear and Cyclic Peptidomimetics: Application in the Synthesis of an Arg-Gly-Asp (RGD)-Containing Peptide as an αvβ3 Integrin Ligand 89
O-benzenedisulfonimide as a powerful and recyclable organocatalyst for the nazarov reaction 87
A Lactam-derived Vinyl Boronate as a Stable and Crystalline Reagent for the Synthesis of 2-substituted Piperidines by Pd-catalyzed Coupling Reactions 86
Effect of C-Ring Modifications in Benzo[c]quinolizin-3-ones, New Selective Inhibitors of Human 5a-Reductase 1 86
A SHORT AND EFFICIENT ROUTE TO ENANTIOPURE 3,5-DIARYLPYRROLIZIDINES 86
Cyclic RGD peptidomimetics containing 4- and 5-aminocyclopropane pipecolic acid (CPA) templates as dual aVb3 and a5b1 integrin ligands 86
Bicyclic compounds derived from Tartaric Acid and α-Amino acids (BTAas): Synthesis of New Molecular Scaffolds derived from the Combination of (R,R)-Tartaric Acid and L-Serine 85
New Synthetic Approach to Cyclopenta-Fused Heterocycles Based Upon a Mild Nazarov Reaction. Part 2: Further Studies on the Torquoselectivity 84
Suzuki Reaction of Vinyl Triflates from Six- and Seven-Membered N-Alkoxycarbonyl Lactams with Boronic Acids and Esters 84
Preparation of Cyclopenta-fused N-, O-, and S-Heterocycles by Lewis Acid-Catalyzed Nazarov Reaction 82
Complementary and Stereodivergent Approaches to the Synthesis of 5-Hydroxy- and 4,5-Dihydroxypipecolic Acids from Enantiopure Hydroxylated Lactams 82
Synthesis of Indenes by Tandem Gold(I)-Catalyzed Claisen Rearrangement/Hydroarylation Reaction of Propargyl Vinyl Ethers 82
Oligomers of enantiopure bicyclic g/d-amino acids (BTAa). 1. Synthesis and conformational analysis of 3-Aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid oligomers (PolyBTG) 81
Stereochemical Assignment of Strigolactone Analogues Confirms Their Selective Biological Activity 81
One-Pot Pictet-Spengler Reaction and Esterification for the Preparation of a Key Tadalafil Synthetic Intermediate 81
New Synthetic Approach to Cyclopenta-Fused Heterocycles Based upon a Mild Nazarov Reaction. 81
Synthesis of Weinreb amides via Pd-Catalyzed Aminocarbonylation of Heterocyclic-derived Triflates 80
Preparation and Cycloaddition Reactions of enantiopure 2-(N-acylamino)-1,3-dienes for the synthesis of octahydroquinoline derivatives 80
Pentannulation Reaction by Tandem Gold(I)-Catalyzed Propargyl Claisen Rearrangement/Nazarov Cyclization of Enynyl Vinyl Ethers 80
Stereoselective Synthesis of (2S,4R)-4-Hydroxypipecolic Acid 79
Remote Stereocontrol in the Nazarov Reaction: A New Approach to the Core of Roseophilin 79
Total Synthesis of Bruceolline I 79
Strigolactone Analogs as Molecular Probes in Chasing the (SLs) Receptor/s: Design and Synthesis of Fluorescent Labeled Molecules 79
A novel allergen-adjuvant conjugate suitable for allergen-specific Th2 redirection 78
Predicting Reactivity and Stereoselectivity in the Nazarov Reaction: A Combined Computational and Experimental Study 77
Synthesis of a-Acyl Functionalized Azacycles by Pd-Catalyzed Cross-Coupling Reactions of a-Alkoxyboronates with Lactam-derived Vinyl Triflates 76
Baker's yeast reduction of prochiral g-nitro ketones. II. Straightforward enantioselective synthesis of 2,7-dimethyl-1,6-dioxaspiro[4.4]nonanes 76
Stereoselective Meisenheimer Rearrangement using BTAa's as Chiral Auxiliaries 76
MODIFICATION OF THE AZA-ROBINSON ANNULATION FOR THE SYNTHESIS OF 4-METHYL-BENZO[C]QUINOLIZIN-3-ONES, POTENT INHIBITORS OF STEROID 5A-REDUCTASE 1 75
Lactam-derived vinyl triflates and phosphates in the synthesis of N-heterocycles 75
The Lewis Acid-catalyzed Nazarov Reaction of 2-(N-methoxycarbonylamino)-1,4-pentadien-3-ones 75
A short and convenient synthesis of enantiopure cis- and trans-4-hydroxypipecolic acid 75
Carbonylative Palladium-Catalyzed Reactions of Lactam-, Lactone-, and Thiolactone-Derived Vinyl Triflates and Phosphates for the Synthesis of N-, O-, and S-Heterocycles 75
Pentannulation of Heterocycles by Virtue of Precious Metal Catalysis 74
Carbonylative Suzuki-Miyaura Coupling Reaction of Lactam-, Lactone-, and Thiolactone-derived Enol Triflates for the Synthesis of Unsymmetrical Dienones. 73
Chemistry of lactam-derived vinyl phosphates: stereoselective synthesis of (+)-fagomine 73
19-NOR-10-AZASTEROIDS. 5.1 A SYNTHETIC STRATEGY FOR THE PREPARATION OF (+)-17-(3-PYRIDYL)-(5B)-10-AZAESTRA-1,16-DIEN-3-ONE, A NOVEL POTENTIAL INHIBITOR FOR HUMAN CYTOCHROME P45017A (17A-HYDROXYLASE/C17,20-LYASE) 72
Selective Nonsteroidal Inhibitors of 5a-Reductase Type 1 71
ENANTIOSELECTIVE SYNTHESIS OF INDOLIZINE DERIVATIVES BY REARRANGEMENT-CYCLIZATION OF ISOXAZOLINE-5-SPIROCYCLOPROPANES 71
Preparation and Suzuki-Miyaura Coupling Reactions of Tetrahydropyridine-2-boronic Acid Pinacol Esters 71
Diastereodivergent synthesis of 4-hydroxy-2,3-methanopipecolic acid derivatives as conformationally constrained homoserine analogues 71
Annulated N-Heterocycles by Tandem Gold(I)-catalyzed [3,3]-Rearrangement/Nazarov Reaction of Propargylic Ester Derivatives: an Experimental and Computational Study 71
A New, practical, and efficient method for protecting alcohols as tert-butyl ethers 70
Synthesis of Both Enantiomers of the Streptomyces Alkaloid 4-epi-SS20846A 68
PS1-076. Redirection of allergen-specific TH2 cells by a modified adenine chemically coupled to allergenic molecule(s) 68
N-Bridgehead polycyclic compounds by sequential rearrangement-annulation of isoxazoline-5-spirocyclopropanes. 6. A general synthetic method of 5,6-dihydro-7(8H)- and 2,3,5,6-tetrahydro-7(1H)-indolizinones 67
A new class of conjugated strigolactone analogues with fluorescent properties: synthesis and biological activity 67
Structure-Function Relations of Strigolactone Analogs: Activity as Plant Hormones and Plant Interactions 67
A modified adenine chemically coupled to allergenic molecule(s) as inducer of allergen-specific Th2 cells redirection 67
Synthesis and reactivity of bicycles derived from tartaric acids and alfa-amino acids: a novel class of conformationally constrained dipeptide isosteres based upon enantiopure 3-aza-6,8-dioxabicyclo[3.2.1]octane-7-carboxylic acid 66
N-Substituent effects on the diethylzinc addition to benzaldehyde catalysed by bicyclic 1,4-aminoalcohols 65
A modified adenine chemically coupled to allergenic molecule(s) as inducer of allergen-specific Th2 cells redirection 65
A CONCISE ROUTE TO 19-NOR-10-AZASTEROIDS, A NEW CLASS OF STEROID 5-REDUCTASE INHIBITORS. 3.1 SYNTHESIS OF (+)-19-NOR-10-AZATESTOSTERONE AND (+)-17B-ACETYLOXY-(5B)-10-AZAESTR-1-EN-3-ONE 64
SYNTHESIS OF ENANTIOPURE 2,7-DIARYL-1,6-DIOXASPIRO[4.4]NONANES VIA ENANTIOSELECTIVE REDUCTION OF PROCHIRAL G-NITROKETONES BY DIISOPINOCAMPHEYLCHLOROBORANE (DIP-CLTM) 64
From synthetic control to natural products: a focus on N-heterocycles 64
Synthesis, biological activity, and three-dimensional quantitative structure-activity relationship model for a series of benzo[c]quinolizin-3-ones, nonsteroidal inhibitors of human steroid 5alpha-reductase 1 64
Analoghi sintetici degli strigolattoni, loro usi e metodi per la loro preparazione 63
Gold-catalyzed Synthesis of Exocyclic Vinylogous Amides and beta-Amino Ketones. A Detailed Study on the 5-exo/6-endo dig Selectivity, Methodology and Scope 63
A Gold(I)-Catalyzed Oxidative Rearrangement of Heterocycle-Derived 1,3-Enynes Provides an Efficient and Selective Route to Divinyl Ketones 62
LIC-KOR PROMOTED FORMATION OF CONJUGATE DIENES AS USEFUL BUILDING BLOCKS IN PALLADIUM-CATALYZED SYNTHESES 61
STEREOSELECTIVITY IN THE TICL4-CATALYSED REEACTION OF DANISHEFSKY¿S DIENE WITH A N-(ACYLOXY)IMINIUM ION: SYNTHESIS OF 5A VERSUS 5B D1(2)-19-NOR-10-AZASTEROIDS. PART 4 60
A modified adenine chemically coupled to the allergen molecule of Dermatophagoides pteronyssinus redirects allergen-specific Th2 cells 60
Tailoring Fluorescent Strigolactones for in vivo Investigations: a computational and experimental study 60
Enantiodivergent chemoenzymatic synthesis of 4-hydroxypiperidine alkaloids 59
A modified adenines chemically coupled to allergen molecule of dermatophagoides pteronyssinus down-regulates allergen-specific Th2 cells responses 57
Recent Advances in the Synthesis of Indenes 57
Pentannulation of N-heterocycles by a tandem gold-catalyzed [3,3]-rearrangement/Nazarov reaction of propargyl ester derivatives: A computational study on the crucial role of the nitrogen atom 55
PROBING ENZYME STEREOSPECIFICITY. INHIBITION OF A-CHYMOTRYPSIN AND SUBTILISIN CARLSBERG BY CHIRAL AMINE- AND AMINOALCOHOL-DERIVATIVES 54
Synthesis of 17b-N-Substituted 19-Nor-10-Azasteroids as Inhibitors of Human 5a-Reductase I and II 53
3-Aza-6,8-dioxabicyclo (3,2,1) octanes and analogues and combinatorial libraries 52
A modified adenine chemically coupled to allergen molecole redirects allergen-specific Th2 cells 51
Process for the synthesis of (1H)-benzo[c]quinolizin-3-ones derivatives 51
Synthesis of Vinylogous Amides by Gold(I)-Catalyzed Cyclization of N‑Boc-Protected 6‑Alkynyl-3,4-dihydro‑2H‑pyridines 51
Synthesis and Conformational Analysis of Small Peptides Containing 6-endo-BT(t)L Scaffolds as Reverse Turns Mimetics 50
Oxidation of diazenyl-protected N-heterocycles – a new entry to functionalized lactams 50
Synthesis and activity of 8-substituted benzo[c]quinolizin-3-ones as dual inhibitors of human 5alpha-reductases 1 and 2 49
Short synthesis of racemic 5-hydroxy-6-hydroxymethylpiperidin-2-one 49
Introduction of the New Dipeptide Isostere 7-Endo-BtA as Reverse Turn Inducer in a Bowman-Birk Proteinase Inhibitor: Synthesis and Conformational Analysis 49
Totale 8.714
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Categoria #
all - tutte 26.290
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 26.290
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019616 0 0 0 0 0 0 0 0 0 0 342 274
2019/20202.219 164 192 56 229 236 278 221 301 205 114 188 35
2020/20211.466 137 99 117 165 39 179 37 140 119 238 78 118
2021/2022882 52 98 76 28 41 32 39 44 44 29 181 218
2022/20232.215 236 389 69 184 190 422 301 120 192 12 57 43
2023/2024635 43 81 126 47 43 104 34 111 16 30 0 0
Totale 9.585